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N-ethyl-5-(2-methoxyphenoxymethyl)-N-methyl-1H-pyrazole-3-carboxamide
N-(2-hydroxyethyl)-N-[(2E)-3-phenylprop-2-en-1-yl]-2-(pyridin-3-yloxy)acetamide
3-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-1-(2-ethyl-2-methyl-4-oxo-3,4-dihydro-2H-1-benzopyran-6-yl)urea
N-(1,3-benzothiazol-2-ylmethyl)-3,6,7-trimethyl-1-benzofuran-2-carboxamide
N-(1-{3-azaspiro[5.5]undecan-9-yl}piperidin-4-yl)methanesulfonamide
N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-4-(pyridin-3-yl)pyrimidin-2-amine
2-[(2-phenylethyl)(pyridin-3-ylmethyl)amino]butan-1-ol
2-(4,5-dimethyl-1H-imidazol-1-yl)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one
5-amino-N-[(3S,5S)-5-(diethylcarbamoyl)-1-(2,2-dimethylpropanoyl)pyrrolidin-3-yl]-1H-pyrazole-3-carboxamide
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-[(4-hydroxypiperidin-1-yl)methyl]piperidin-2-one
2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]-N-(1-propylpiperidin-4-yl)acetamide
1-(3-{3-[4-(trifluoromethyl)pyrimidin-2-yl]phenyl}-1H-pyrazol-1-yl)butan-2-ol
4-{6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-2-methyl-1-(propan-2-yl)piperazine
[(2-fluorophenyl)[1-(6-methylpyridin-2-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]methyl]dimethylamine
N-methyl-N-[(2-phenyl-1,3-thiazol-5-yl)methyl]-2-propyl-1,3-thiazole-4-carboxamide
3-{[4-(4,6-dimethylpyrimidin-2-yl)piperazin-1-yl]methyl}-3-hydroxy-1-(2-methoxyethyl)piperidin-2-one
N-methyl-5-phenoxy-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}furan-2-carboxamide
1-methyl-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-{[3-(cyclopentyloxy)propyl]sulfamoyl}-N-(propan-2-yl)benzamide
2-({4-[3-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)ethan-1-ol
5-(dimethylamino)-2-[2-(3-methoxypiperidin-1-yl)-2-oxoethyl]-2,3-dihydropyridazin-3-one
N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}-2,5,7-trimethylpyrazolo[1,5-a]pyrimidine-3-carboxamide
4-{1-[3-(trifluoromethyl)benzenesulfonyl]azetidin-3-yl}pyridine
N-[3-(oxolan-3-yl)propyl]-2,3-dihydro-1H-inden-2-amine
1-(2-methoxyethyl)-1-[(5-methylthiophen-2-yl)methyl]-3-{[1,2,4]triazolo[4,3-a]pyridin-8-yl}urea
3,5-dimethyl-2-{4-[2-(1H-pyrrol-1-yl)ethyl]piperazine-1-carbonyl}-1H-indole
2-(4-fluorophenyl)-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}imidazo[1,2-a]pyridine-6-carboxamide
[7-(1H-indazol-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
1-methyl-9-[2-(3-phenylpyrrolidin-1-yl)acetyl]-1,4,9-triazaspiro[5.5]undecan-5-one
5-{1-[1-(cyclohex-1-en-1-yl)ethyl]-1H-1,2,3-triazol-4-yl}-2-(pyridin-2-yl)pyrimidine
4-[2-(1H-pyrazol-1-yl)ethyl]-1-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperidine
2-methylpropyl 9-[(3-cyanophenyl)methyl]-3,9-diazaspiro[5.5]undecane-3-carboxylate
{[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}[1-(3-methoxyphenyl)ethyl]methylamine
N-[(1R,3S)-3-(morpholine-4-carbonyl)cyclopentyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
2-(2-acetyl-4,5-dimethoxyphenyl)-1-[(3S)-3-ethylmorpholin-4-yl]ethan-1-one
N,1-dimethyl-N-[2-(1H-pyrazol-4-yl)ethyl]-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2,5-dimethylpyrazine
(3R,4R)-N-ethyl-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1-methyl-N-(oxan-4-ylmethyl)pyrrolidine-3-carboxamide
3-(3-chlorophenyl)-1-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]propan-1-one
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-4,6-dimethylpyrimidin-2-amine
1-(cyclopropylmethyl)-3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidine
4-methyl-N-{2-[4-(oxan-4-yl)morpholin-2-yl]ethyl}pyridine-3-carboxamide
N-(propan-2-yl)-1-{1-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]piperidin-4-yl}piperidine-4-carboxamide
N-[(2R,3R)-2-methoxy-1'-(2-oxo-2H-pyran-5-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenylacetamide
N-(2-hydroxy-1-phenylethyl)-2-(2,2,6,6-tetramethylpiperidin-4-yl)acetamide
3-[(3R,4S)-1-[3-chloro-4-(pyrrolidin-1-yl)benzoyl]-4-(dimethylamino)piperidin-3-yl]propan-1-ol
N-(2-methoxyethyl)-2,7-dimethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]imidazo[1,2-a]pyridine-3-carboxamide
(2S,4S)-4-amino-N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-1-methylpyrrolidine-2-carboxamide
1-[(2R,3S,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(pyridin-2-yl)ethan-1-one
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-5-methoxy-N,1-dimethyl-1H-indole-2-carboxamide