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2-[(5-methyl-1H-1,3-benzodiazol-2-yl)sulfanyl]-N-[1-(pyridin-3-yl)propan-2-yl]acetamide
4-methyl-1-{3-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}pentan-1-one
N-cyclooctyl-2-{[2-(pyrrolidine-1-sulfonyl)ethyl]amino}acetamide
1-[6-(dimethylamino)pyridine-3-carbonyl]-4-(4-fluorophenyl)piperidin-4-ol
(3aR,7aS)-2-{1H-pyrrolo[2,3-b]pyridin-6-yl}-2,3,3a,4,7,7a-hexahydro-1H-isoindole
6-chloro-N-[4-(5-methylfuran-3-amido)phenyl]pyridine-2-carboxamide
4-cyano-N-(4-methoxy-2-methylphenyl)piperidine-1-carboxamide
2-(dimethylamino)-2-(2-fluorophenyl)-N-[2-(4-hydroxyphenyl)-2-oxoethyl]-N-methylacetamide
3-(5-amino-1H-1,2,4-triazol-3-yl)-N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
2-{8-methylimidazo[1,2-a]pyridin-3-yl}-N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)acetamide
3-chloro-4-methyl-N-{[1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]methyl}benzamide
3-{[(1R,3S,5S)-3-(4-fluoro-3-methylphenyl)-8-azabicyclo[3.2.1]octan-8-yl]methyl}pyridin-2-amine
[(1,5-dimethyl-1H-indol-2-yl)methyl](methyl)(pyrazin-2-ylmethyl)amine
2-{[5-(1-methyl-1H-1,3-benzodiazol-2-yl)furan-2-yl]methyl}-1,2,3,4-tetrahydroisoquinolin-4-ol
(2S)-4-{[3-(4-fluorophenyl)-1H-pyrazol-5-yl]formamido}-2-hydroxybutanoic acid
(3S,4R)-4-(3-methylthiophen-2-yl)-1-(4,5,6,7-tetrahydro-1,3-benzothiazole-2-carbonyl)piperidin-3-ol
N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}furan-3-carboxamide
N-(1-butyl-4-methyl-1H-pyrazol-5-yl)-2-(2-methyl-2,3-dihydro-1H-indol-1-yl)-2-oxoacetamide
5-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1H-1,2,3-benzotriazole
(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)-N-(2-phenylethyl)piperidine-1-carboxamide
5-{furo[3,2-c]pyridin-4-yl}-2,4-dimethoxypyrimidine
(1R,7S)-3-(4-fluorophenyl)-N-methyl-4-oxo-N-[2-(pyridin-2-yl)ethyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
(1R,3S)-3-ethoxy-7-(2-methyl-4-phenylpyridine-3-carbonyl)-7-azaspiro[3.5]nonan-1-ol
3-amino-1-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}pyrrolidine-3-carboxylic acid
N-{4-[2-(cyclopropylcarbamoyl)ethyl]phenyl}-3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carboxamide
1-[(3,4-dimethoxyphenyl)methyl]-4-[2-(thiomorpholine-4-carbonyl)-1-benzofuran-5-yl]piperidin-4-ol
N-(2-methanesulfonamidoethyl)-2-methyl-4-oxo-1,4-dihydroquinoline-8-carboxamide
5-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-N,N,4-trimethylpyrimidin-2-amine
N-[3-chloro-4-(2,2-dimethylpropanamido)phenyl]-1H-imidazole-5-carboxamide
3-methyl-N-(2-{1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}ethyl)furan-2-carboxamide
5-chloro-1,3-dimethyl-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-1H-pyrazole-4-sulfonamide
N-[(2,4-difluorophenyl)methyl]-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
1-[3-({4-[(4-fluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenyl]ethan-1-one
7-(3-chlorophenyl)-4-(2-methyl-1,3-thiazole-4-carbonyl)-9-(oxan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-(5-propyl-1,2,4-oxadiazol-3-yl)piperazine-2-carboxylic acid
N-methyl-3-[3-(oxan-4-yl)-1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]propanamide
N-cyclopropyl-2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}acetamide
butyl(methyl)({5-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)amine
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[3-(pyridin-3-yloxy)propyl]benzamide
N-(furan-2-ylmethyl)-N-{[2-(morpholin-4-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-3-(1H-pyrazol-5-yl)piperidine
N-[1-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-2,3-dihydro-1-benzofuran-5-carboxamide
9-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[(5-fluoro-2-methylphenyl)methyl]-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
ethyl 1-(2-acetylbenzoyl)-4-[(4-chlorophenyl)methyl]piperidine-4-carboxylate
4-(1-ethyl-1H-pyrazole-5-carbonyl)-1-[(4-methylphenyl)methyl]piperazin-2-one
2-[4-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperazin-1-yl]-1,3-benzothiazole
N-[2-(cyclohex-1-en-1-yl)ethyl]-5-methyl-6-(4-methylpiperazine-1-carbonyl)thieno[2,3-d]pyrimidin-4-amine
N,N-dimethyl-5-({4-[(3-methylphenyl)methyl]piperazin-1-yl}methyl)pyridin-2-amine
(3R,4S)-1-(5-methylpyrazine-2-carbonyl)-4-propylpyrrolidin-3-amine