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N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]oxane-4-carboxamide
3-{[2-(4-methoxy-2,3-dimethylphenyl)-1H-imidazol-1-yl]methyl}-1,2,4-oxadiazole-5-carboxamide
methyl (2S,4R)-1-methyl-4-[3-(pyridin-3-yl)propanamido]pyrrolidine-2-carboxylate
1-[1-(2-cyclohexylacetyl)piperidin-4-yl]-N-cyclopentyl-1H-1,2,3-triazole-4-carboxamide
[(3R,4R)-4-[(dimethylamino)methyl]-1-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-yl]methanol
1-cyclopropanecarbonyl-N-methyl-N-[1-(1,3-thiazol-5-yl)ethyl]piperidine-4-carboxamide
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-[2-(methylsulfanyl)pyrimidine-5-carbonyl]pyrrolidin-3-yl]methanol
1-(2,3-dihydro-1H-inden-2-yl)-3-methyl-5-(1H-1,2,3-triazol-5-yl)-1H-1,2,4-triazole
2-methyl-4-[4-({2-methyl-2,7-diazaspiro[4.5]decan-7-yl}methyl)phenyl]butan-2-ol
3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-[4-(1H-pyrazol-1-yl)benzoyl]piperidine
2-{2-oxo-2-[3-(pyridine-2-carbonyl)piperidin-1-yl]ethyl}-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}cyclobutanamine
4-[3-(1H-imidazol-1-yl)pyrrolidin-1-yl]-1-[3-(1H-pyrazol-5-yl)phenyl]piperidine
(4aS,8aR)-1-(2-aminoethyl)-6-(isoquinoline-1-carbonyl)-decahydro-1,6-naphthyridin-2-one
4-{[5-(3-chlorophenyl)furan-2-yl]methyl}-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
[2,2-dimethyl-3-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)propyl]dimethylamine
2-{1-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]-1H-imidazol-2-yl}benzoic acid
3-(but-2-yn-1-yl)-5-[1-(1H-indol-2-ylmethyl)piperidin-4-yl]-5-(3-phenylpropyl)imidazolidine-2,4-dione
4-[(4-acetylphenyl)methyl]-1-(3-methoxyphenyl)piperazin-2-one
2-(2H-1,3-benzodioxol-5-yloxy)-1-[4-(1H-imidazol-2-yl)piperidin-1-yl]propan-1-one
N-[cyclopropyl(6-methylpyridin-2-yl)methyl]-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
4-methyl-2-{[methyl({[4-(1H-pyrazol-1-yl)phenyl]methyl})amino]methyl}phenol
N-({5-[(3-methyl-1-phenyl-1H-pyrazol-4-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
2-{3-cyclopropyl-5-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,4-triazol-1-yl}pyridine
1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-4-(oxolan-2-ylmethyl)piperazine
5-(azepane-1-carbonyl)-1-(butan-2-yl)-4-oxo-N-[3-(pyridin-4-yl)propyl]-1,4-dihydropyridine-3-carboxamide
5-acetyl-2,4-dimethyl-N-[1-(3-methylphenyl)-5-oxopyrrolidin-3-yl]-1H-pyrrole-3-carboxamide
ethyl 2-(3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-methylpropanamido)acetate
1-[4-(3-chlorophenyl)-2-methyl-5-oxopiperazin-1-yl]-2-phenylethane-1,2-dione
N-cyclopentyl-5-fluoro-N-{[4-methoxy-3-(propan-2-yloxy)phenyl]methyl}-2-methylbenzene-1-sulfonamide
5-[methyl(2-phenylethyl)amino]-2-[2-(phenylsulfanyl)ethyl]-2,3-dihydropyridazin-3-one
4-(2-amino-6-fluoro-1,3-benzothiazol-4-yl)phenol
3-[(1,1-dioxo-1λ6-thiolan-3-yl)(methyl)amino]-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]propanamide
1-{[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}azetidin-3-ol
(1S,4S)-5-(4,6-dimethylpyrimidin-2-yl)-2-(2-methoxy-5-phenylphenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
3-(2-fluorophenyl)-N-[2-(6-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-1H-pyrazole-5-carboxamide
1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-3-(3-methoxybenzoyl)piperidine
1-ethyl-5-({[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}amino)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
methyl 4-{[3-(3-chlorobenzoyl)piperidin-1-yl]methyl}benzoate
N5-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-N3,N3-dimethyl-1,2,4-thiadiazole-3,5-diamine
2-ethyl-9-(4-methoxy-3-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
(1S,5R)-6-(cyclopropanesulfonyl)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonane
N-{3-[(2S)-2-aminopropanamido]phenyl}-4-methylbenzamide
2-{4-[(2-butyl-1H-imidazol-4-yl)methyl]morpholin-3-yl}acetic acid
4-(4-cyclohexanecarbonylpiperazine-1-carbonyl)-6-ethyl-2-methylquinoline
1-[4-(3-methoxyphenyl)piperazin-1-yl]-3-(1-methylpiperidin-2-yl)propan-1-one
2-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-8-methoxy-4-methylquinoline
1-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-2-(2,5,7-trimethyl-1H-indol-3-yl)ethan-1-one
2-hydroxy-5-(1-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1H-imidazol-2-yl)benzoic acid
1-(1-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)-1,4-diazepan-5-one