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9-(5-methanesulfonyl-2-methylpyrimidin-4-yl)-5-methoxy-1-oxa-9-azaspiro[5.5]undecane
N-[(2,3-dimethylphenyl)methyl]-5-(3-fluorophenoxymethyl)-1H-pyrazole-3-carboxamide
6-[(3-methoxyphenyl)methoxy]-1-(2-phenylethyl)-4-(pyridine-4-carbonyl)-1,4-diazepan-2-one
N-cyclopropyl-1-[2-(4-methoxyphenyl)ethyl]-6-oxopiperidine-3-carboxamide
1-benzoyl-4-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperazine
(2R)-2-[5-(2,4-diethoxy-3-methylphenyl)-4-phenyl-1H-imidazol-1-yl]propanamide
N-cyclopropyl-3-{1-[4-(2-oxopiperidin-1-yl)butanoyl]piperidin-4-yl}propanamide
N-[(5-ethylpyridin-2-yl)methyl]-2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
2-acetamido-N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}acetamide
2-{2-[1-(1-cyclopropyl-5-oxopyrrolidine-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
2-(2-hydroxyphenyl)-1-{3-oxa-9-azaspiro[5.5]undecan-9-yl}ethan-1-one
1-[1-(methoxymethyl)cyclobutanecarbonyl]-4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine
N-(3-chloro-4-fluorophenyl)-3-[1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)piperidin-4-yl]propanamide
N-[1-(3-phenylpropyl)piperidin-3-yl]pyridine-4-carboxamide
4-methyl-2-{4-[3-(2-methylphenyl)piperidine-1-carbonyl]piperidin-1-yl}quinazoline
2-cyclopropanecarbonyl-8-(6-cyclopropylpyrimidin-4-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(3aR,6aR)-2-(cyclopentylcarbamoyl)-5-(pyridin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-methyl-N-[3-(4-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}phenoxy)propyl]benzamide
3-methyl-1-{1-oxa-7-azaspiro[3.5]nonan-7-yl}-3-phenylbutan-1-one
5-{1-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]piperidin-4-yl}-5-(pyridin-3-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
2-[3-(1-methyl-1H-pyrazol-5-yl)phenyl]-5-(pyrrolidin-1-ylmethyl)pyridine
1-(2-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}-2-oxoethyl)pyrrolidin-2-one
methyl 4-({[5-(2,6-dimethylphenoxymethyl)-1,2-oxazol-3-yl]formamido}methyl)benzoate
1-{[5-(1-cyclopropanecarbonylpiperidin-4-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}-4-methylpiperazine
3-hexyl-8-[2-(morpholin-4-yl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[5-(4-cyclohexylphenyl)-1,2,4-triazin-3-yl]-4-(piperidin-1-yl)piperidine-4-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[1-(4-methyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]piperazine
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-cyclopropyl-3-(1H-pyrazol-1-ylmethyl)benzamide
(3S,4R)-1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-N,N-dimethyl-4-(4-methylphenyl)pyrrolidin-3-amine
3-(4-fluorophenyl)-N,N-bis(1,3-oxazol-4-ylmethyl)-1H-pyrazole-5-carboxamide
8-(2-methoxyacetyl)-3-(2-phenylpropyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-1-(pyridin-4-ylmethyl)pyrrolidin-2-one
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(3-cyclopentylpropyl)acetamide
4-(1-{[5-(4-ethoxyphenyl)furan-2-yl]methyl}piperidin-3-yl)pyrimidine
N-[(2-fluoro-4-methoxyphenyl)methyl]-1-(pyrimidin-2-yl)piperidin-3-amine
N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-1,9-dioxaspiro[5.5]undecan-4-amine
(4aR,6R,8aS)-2-(1H-imidazol-4-ylmethyl)-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinoline
6-fluoro-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
N-tert-butyl-2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
2-methyl-N-(3-methyl-1,2,4-thiadiazol-5-yl)pyrrolidine-1-carboxamide
2-[2-(3-methoxyphenyl)azetidine-1-carbonyl]-3,4,7-trimethyl-1H-indole
3-[2-(2-methyl-2,3-dihydro-1-benzofuran-5-yl)-1H-imidazol-1-yl]pyridine
N-cyclopropyl-3-{1-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperidin-4-yl}propanamide
N-methyl-N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
methyl 5-{2-[(2,4-dimethylphenyl)carbamoyl]acetyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
4-ethyl-1-methyl-3-(1-{2-[(2-methylphenyl)sulfanyl]acetyl}piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-methyl-5-({5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-1,4-dihydropyridin-4-one
(1S,5R)-6-(4-chloro-2-methylbenzoyl)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-(4,6-dimethyl-2-oxo-1,2-dihydropyridin-1-yl)-3-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-4-yl)propanamide
1-methyl-N-{2-[(pyridin-3-yl)amino]ethyl}-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carboxamide