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7-methanesulfonyl-4-methyl-2-(3-methylpiperidin-1-yl)quinazoline
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
7-(1-benzothiophen-3-yl)-4-(furan-3-carbonyl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(6-methoxynaphthalen-2-yl)-4-(6-methylpyridazin-3-yl)morpholine
2-{[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]methyl}-1H-indole
3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-2-methoxypyridine
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-(5-propyl-1,2-oxazole-3-carbonyl)piperazine
(3R,5S)-5-[(4-methylpiperazin-1-yl)methyl]-N,1-bis(2-methylpropyl)piperidine-3-carboxamide
N-cyclopentyl-4-[6-(thiomorpholin-4-yl)pyridazin-3-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
4-[7-(2,4-difluorobenzoyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]morpholine
4-methyl-N-propyl-N-(pyridin-3-ylmethyl)benzamide
1-(carbamoylmethyl)-N-ethyl-N-[2-hydroxy-2-(3-hydroxyphenyl)ethyl]piperidine-4-carboxamide
1-{3-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-4-phenylbutan-1-one
8-(2,5-dichlorobenzenesulfonyl)-1-oxa-8-azaspiro[4.5]decane
N-cyclopropyl-N-(1H-indol-5-ylmethyl)-4-(1H-pyrazol-4-yl)butanamide
2-(4-{[(1,4-dioxan-2-ylmethyl)(methyl)amino]methyl}phenyl)-6-(pyridin-2-yl)-3,4-dihydropyrimidin-4-one
2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-hydroxyethyl)-N-propylacetamide
1-(1-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}piperidin-4-yl)piperidin-3-ol
3-{5-[1-(4-fluorobenzenesulfonyl)pyrrolidin-2-yl]-1,2,4-oxadiazol-3-yl}pyridazine
[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl})amine
N-[(2,3-dimethylphenyl)methyl]-2-(1H-indazol-3-yl)acetamide
7-(1,3-benzothiazol-2-yl)-4-(5-methylpyrazine-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-2-(pyridin-3-yl)morpholine
N-[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
ethyl 1-[1-(6-methylpyridin-2-yl)propan-2-yl]-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-(2-methylpropyl)-decahydro-1,6-naphthyridin-2-one
methyl 3-[(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)carbamoyl]propanoate
1-({3-[(1-cyclohexanecarbonylpiperidin-4-yl)oxy]phenyl}methyl)-4-(pyridin-2-yl)piperazine
3-{1-[2-(diethylamino)ethyl]-1H-imidazol-2-yl}benzonitrile
2-methyl-9-(morpholine-4-carbonyl)-4-phenyl-2,9-diazaspiro[5.5]undecane
[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]({[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
5-chloro-6-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]pyridine-3-carboxylic acid
4-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,3λ6,4-oxathiazinane-3,3-dione
2-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]acetamide
1-[(3,4-dimethylphenyl)methyl]-4-[2-methyl-3-(pyrrolidin-1-yl)propanoyl]piperazin-2-one
N,N-dimethyl-2-[(1S,5R)-6-(5-methylpyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-[(3-methoxyphenyl)methyl]-3-[1-(4-phenylbutanoyl)piperidin-3-yl]propanamide
3-methoxy-1-{6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carbonyl}piperidine
N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-1-phenyl-1H-1,2,3-triazole-4-carboxamide
1-{4-[(oxolan-3-yl)amino]-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}cyclopropanecarboxamide
4-[(5-methylfuran-2-yl)methyl]-3-(2-oxo-2-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-yl}ethyl)piperazin-2-one
2-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
N-{[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]methyl}-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propanamide
6-ethoxy-3-(1,2,3,6-tetrahydropyridin-1-ylmethyl)-1,2-dihydroquinolin-2-one
2-(dimethyl-1,2-oxazol-4-yl)-1-[3-(4-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}phenoxymethyl)piperidin-1-yl]ethan-1-one
1-{2-[(3R,4R)-3-hydroxy-4-methyl-3-(propan-2-yl)pyrrolidin-1-yl]-2-oxoethyl}-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
(4aR,8aR)-7-[(5-cyclopentylthiophen-2-yl)methyl]-4a-hydroxy-N,N-dimethyl-decahydro-2,7-naphthyridine-2-carboxamide
N-cyclopropyl-2-({1-[(5-ethylfuran-2-yl)methyl]piperidin-4-yl}oxy)-4-methoxybenzamide