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4-[(2-ethyl-1H-imidazol-1-yl)methyl]-5-methyl-2-(2-methylphenyl)-1,3-oxazole
1-{[5-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
(2S,4S)-1-benzyl-N-ethyl-4-{[(3-methylphenyl)methyl]amino}pyrrolidine-2-carboxamide
1-(4-{[(5-methylthiophen-2-yl)methyl]amino}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
(2S)-2-amino-3-(1H-imidazol-4-yl)-N-[2-(3-phenylpropoxy)phenyl]propanamide
2,3-dimethoxy-N-{[1-(1H-pyrazol-3-ylmethyl)piperidin-3-yl]methyl}benzamide
2-(dimethylamino)-N-[2-(1-hydroxycyclopentyl)ethyl]-N-methyl-2-(2-methylphenyl)acetamide
3,4,7-trimethyl-2-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]-1H-indole
N-[(1-cyclohexylpyrrolidin-3-yl)methyl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
(3S,4S)-1-(4-cyclopentylpyrimidin-2-yl)-4-(morpholin-4-yl)pyrrolidin-3-ol
1-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-[2-(trifluoromethyl)phenyl]ethan-1-one
4-(2-cyclopropylpyrimidine-5-carbonyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-(4-{3-azaspiro[5.5]undecan-9-yl}-1,4-diazepan-1-yl)-2-methoxyethan-1-one
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-1H-imidazole-2-carboxamide
methyl 2-[8-(1H-indol-3-ylmethyl)-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetate
4-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-4-oxobutanamide
3-methoxy-N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)propanamide
N-[3-(1H-1,2,3-triazol-1-yl)propyl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
N-{[7-(5-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-[4-(methylsulfanyl)phenyl]acetamide
1-methyl-4-[2-(morpholin-4-yl)-2-oxoethyl]-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
3-{2-[4-(methoxymethyl)piperidin-1-yl]-2-oxoethyl}-4-(3-methylbutyl)piperazin-2-one
2-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methoxy]-N-[(1-methylpiperidin-3-yl)methyl]acetamide
N-{[2-(difluoromethoxy)phenyl]methyl}-1-(pyrimidin-2-yl)piperidin-3-amine
ethyl 4-(2-methoxyethyl)-1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidine-4-carboxylate
3-benzyl-1-methyl-3-[3-oxo-3-(thiomorpholin-4-yl)propyl]-2,3-dihydro-1H-indol-2-one
3-chloro-4-fluoro-N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-1-benzothiophene-2-carboxamide
2-(pyridin-4-ylmethyl)-9-(3,3,3-trifluoro-2-methylpropyl)-2,9-diazaspiro[5.5]undecan-3-one
N4-[2-(4-fluorobenzenesulfonyl)ethyl]-6-methyl-5-(prop-2-en-1-yl)pyrimidine-2,4-diamine
8-chloro-2-(furan-2-yl)-4-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]quinoline
(3R,5S)-1-benzyl-N,N-dimethyl-5-{[(6-methylpyridin-3-yl)oxy]methyl}piperidine-3-carboxamide
6-({1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}methyl)-3-methanesulfonylpyrazolo[1,5-a]pyrimidine
1'-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carbonyl}spiro[indene-1,4'-piperidine]
8-[(2,6-dimethylphenyl)methyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-(dimethyl-1,3-thiazole-5-carbonyl)-3-(1-ethyl-1H-imidazol-2-yl)piperidine
2-fluoro-N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]-5-sulfamoylbenzamide
5-(4-acetylphenoxymethyl)-N-ethyl-N-(propan-2-yl)-1,2-oxazole-3-carboxamide
N-{1-[1-(1H-indol-2-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}pyridine-3-carboxamide
1-(1-{1-[(trimethylpyrazin-2-yl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)propan-2-ol
4-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]-1-(4-methylphenyl)piperazin-2-one
2-({5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)ethan-1-ol
(1-{[2,5-dimethyl-1-(pyridin-3-yl)-1H-pyrrol-3-yl]methyl}pyrrolidin-3-yl)methanamine
(4S)-3,3,4-trimethyl-1-[3-(5-methylfuran-2-yl)benzoyl]piperidin-4-ol
4-ethyl-1-[(2E)-3-(4-fluorophenyl)prop-2-enoyl]-1,4-diazepan-5-one
2-chloro-5-(4-phenyl-1H-imidazol-5-yl)pyridine
2-(4-chloro-1H-pyrazol-1-yl)-1-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}propan-1-one
{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)(oxolan-3-ylmethyl)amine
2-[4-(2H-1,3-benzodioxol-4-ylmethyl)-1-[(2-fluorophenyl)methyl]piperazin-2-yl]ethan-1-ol
2-(aminomethyl)-N-(3-methanesulfonamidophenyl)piperidine-1-carboxamide
6-ethyl-N-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]pyrimidin-4-amine
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}(furan-3-ylmethyl)(oxolan-2-ylmethyl)amine