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N-({5-[(3-ethenylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)methanesulfonamide
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-4-{octahydropyrrolo[1,2-a]piperazine-2-carbonyl}-1,3-oxazole
5,5-dimethyl-1-(2-oxo-2-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethyl)imidazolidine-2,4-dione
5-[benzyl(methyl)amino]-2-(oxan-2-ylmethyl)-2,3-dihydropyridazin-3-one
N-methyl-N-(quinolin-6-ylmethyl)cyclobutanecarboxamide
2-[3-(3,4-dimethyl-1H-pyrazol-5-yl)propanamido]-N-(2,6-dimethylphenyl)benzamide
N-methyl-2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]acetamide
3-chloro-4-hydroxy-N-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}benzamide
N-[(4-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethoxy}-3-methoxyphenyl)methyl]-N-[(3S)-2-oxoazepan-3-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
(3S,4S)-1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
6-[3-(4-fluorophenyl)pyrrolidin-1-yl]-9H-purin-2-amine
ethyl 4-{2-[1-methyl-2,5-dioxo-3-(4-phenylphenyl)pyrrolidin-3-yl]acetyl}piperazine-1-carboxylate
2-(2-hydroxyethyl)-8-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
4-({3-[2-(1-cyclobutanecarbonylpiperidin-2-yl)ethoxy]-4-methoxyphenyl}methyl)morpholine
6-(3-methylpiperazin-1-yl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
4-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]morpholine-2-carboxylic acid
(3S,5S)-N-(2,3-dihydro-1H-inden-2-yl)-1-(propan-2-yl)-5-{4-[3-(trifluoromethyl)phenyl]piperazine-1-carbonyl}pyrrolidin-3-amine
8-fluoro-3-{4-[2-(methylsulfanyl)ethyl]piperazine-1-carbonyl}-1,4-dihydroquinolin-4-one
5,5-dimethyl-3-(2-oxo-2-{spiro[indene-1,4'-piperidine]-1'-yl}ethyl)-1,3-oxazolidine-2,4-dione
2-(1-methyl-1H-pyrazole-5-carbonyl)-7-(pyrrolidine-1-sulfonyl)-1,2,3,4-tetrahydroisoquinoline
(3aR,6aR)-2-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-5-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[({3-cyclopropyl-1-[(4-fluorophenyl)methyl]-1H-1,2,4-triazol-5-yl}methyl)sulfanyl]pyrimidine
1-(3-chloro-4-methoxybenzoyl)-2-(3-methoxypropyl)piperidine
N-[(3-methoxyphenyl)methyl]-N-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}cyclopropanamine
1-{8-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decane
N,3-dimethyl-5-propyl-N-(1,3-thiazol-2-ylmethyl)-1-benzofuran-2-carboxamide
1-{1-[4-(methylsulfanyl)butan-2-yl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
1-({6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}sulfonyl)-4-hydroxypiperidine-4-carboxylic acid
N-[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-2-(phenylamino)pyrimidine-5-carboxamide
4-(4-{[2-(aminomethyl)morpholin-4-yl]methyl}-2-methylphenoxy)thiane-4-carboxylic acid
4-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(4aS,7aR)-4-ethyl-N-[3-(methylsulfanyl)phenyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
7-[(3-propylmorpholin-4-yl)methyl]-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-4-hydroxy-3-methylbenzamide
N,N,4-trimethyl-3-({[3-(pyridin-4-yl)propyl]carbamoyl}methyl)-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-{1H-pyrrolo[2,3-b]pyridin-6-yl}piperazine
N-(1-{5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}-2-phenylethyl)-3-methylthiophene-2-carboxamide
1-methyl-4-(2-methyl-1,8-naphthyridine-3-carbonyl)piperazine-2-carboxylic acid
2-(1-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}-3-oxopiperazin-2-yl)-N-methylacetamide
3-acetyl-N-{2-[(trifluoromethyl)sulfanyl]ethyl}-1H-pyrazole-5-carboxamide
3-ethoxy-1-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[2-(pyridin-4-yl)ethyl]propanamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]pyrrolidin-3-yl]-2,4-dimethyl-1,3-oxazole-5-carboxamide
1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine
({5-[1-(2,1,3-benzoxadiazole-5-carbonyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
N-{[6,7-dimethoxy-2-(3-methoxyphenyl)quinolin-3-yl]methyl}-2-(3-methyl-1H-pyrazol-1-yl)-N-(oxolan-2-ylmethyl)acetamide
N-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl][(3-methylthiophen-2-yl)methyl](pyridin-2-ylmethyl)amine
7-(3,6-dimethylpyrazin-2-yl)-4-[2-(pyrrolidin-1-yl)ethyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol