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N-{[1-(3-chlorophenyl)-1H-pyrazol-4-yl]methyl}-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
3-(3-chloro-1,2-oxazol-5-yl)-1-{5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}propan-1-one
1-(5-acetyl-2,4-dimethyl-1H-pyrrole-3-carbonyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-[1-(5-aminopyrazin-2-yl)-4-methyl-1H-1,3-benzodiazol-2-yl]ethan-1-ol
8-methyl-N-{2-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}imidazo[1,2-a]pyridine-2-carboxamide
1-[1'-(3-fluoro-4-methylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
N-[1-methyl-3-(pyridin-3-yl)-1H-pyrazol-5-yl]-2-[4-(4-methylphenyl)-1H-pyrazol-1-yl]acetamide
1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-4-(thian-4-yl)piperazine
1-[5-(4-chloro-3,5-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]azocane
{3-[(4-fluorophenyl)methyl]-1-(6-methoxypyrimidin-4-yl)piperidin-3-yl}methanol
ethyl 1-{2-[(1,3-thiazol-2-yl)carbamoyl]ethyl}piperidine-2-carboxylate
ethyl 1-{2-[3-(2-chlorophenyl)-1-methyl-2,5-dioxopyrrolidin-3-yl]acetyl}piperidine-2-carboxylate
(4S,4aS,8aS)-1-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-4-phenyl-decahydroquinolin-4-ol
(4aS,8aR)-6-[(3-ethyl-1,2-oxazol-5-yl)methyl]-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
4-[2-(4-fluorophenyl)azetidine-1-carbonyl]-2,8-dimethylquinoline
(2E)-3-(1H-imidazol-4-yl)-1-{3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}prop-2-en-1-one
1-[(4-methylphenyl)methyl]-N-(1-methylpiperidin-4-yl)-5-oxopyrrolidine-3-carboxamide
8-methyl-2-(5-propyl-1,3,4-oxadiazol-2-yl)-2,8-diazaspiro[4.5]decane
4-[4-(prop-2-en-1-yl)benzoyl]-2-(trifluoromethyl)morpholine
4-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]benzonitrile
N-cyclopropyl-1-[1-(1-methyl-2-oxo-1,2-dihydropyridine-3-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
(3S,4R)-1-[(2,4-dimethoxy-3-methylphenyl)methyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
4-[5-(hydroxymethyl)furan-2-yl]-1-phenyl-3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
(3S,5R)-N3-(2-acetamidoethyl)-N5-(4-fluorophenyl)-1-(2-methylpropyl)piperidine-3,5-dicarboxamide
3-(2-phenylpropyl)-N-[2-(1,3-thiazol-4-yl)ethyl]-1,2-oxazole-5-carboxamide
2-(1H-indol-3-yl)-N-methyl-N-{2-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}acetamide
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-3-(2-methoxyphenyl)-1H-pyrazole-5-carboxamide
dimethyl(3-{2-[1-(propan-2-yl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)amine
6-[4-chloro-2-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]pyrazine-2-carboxylic acid
dimethyl[3-(2-{1-[3-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}-1H-imidazol-1-yl)propyl]amine
2-(3-chloro-5-fluorophenyl)-1-(oxan-4-ylmethyl)-1H-imidazole
4-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-3-methyl-1-(2-methylpropyl)piperazin-2-one
2-(3-methylbutyl)-8-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-2,8-diazaspiro[5.5]undecan-3-one
ethyl[(2-ethylpyrimidin-4-yl)methyl][2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]amine
2-{1-[(4Z)-hept-4-en-1-yl]azetidin-3-yl}-1H-1,3-benzodiazole
(2S,4S)-4-amino-1-(3-cyclopentylpropanoyl)-N-methylpyrrolidine-2-carboxamide
N-butyl-5-methyl-4-[(oxolan-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidine
1-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(pyridin-2-yl)propan-1-one
2-{1-[1-(methoxymethyl)cyclobutanecarbonyl]pyrrolidin-3-yl}benzoic acid
4-[6-(5-chloro-2-ethoxyphenyl)pyridazin-3-yl]thiomorpholine
2-cyclopropanecarbonyl-8-(6-ethylpyrimidin-4-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1'-[(1-ethyl-1H-pyrazol-4-yl)methyl]-5-(3-methylbut-2-en-1-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-{2-[(E)-2-phenylethenyl]pyrimidin-4-yl}pyrrolidin-3-ol
4-ethyl-3-[(1-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}piperidin-4-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(morpholin-4-yl)-2-{4-[({[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}amino)methyl]phenoxy}ethan-1-one
2-(4-{[(2-hydroxyethyl)(methyl)amino]methyl}phenyl)-5-methyl-6-(trifluoromethyl)-3,4-dihydropyrimidin-4-one
2-{4-[(2-chlorophenyl)methyl]-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
(4aS,7aR)-1-(3-methoxy-2-methylbenzoyl)-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-({[(3R,4R)-4-(hydroxymethyl)-1-[2-(trifluoromethyl)-1H-1,3-benzodiazole-5-carbonyl]pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol