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2-{[(1R,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-5-methoxy-4H-pyran-4-one
4-(4-{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)phenol
8-[2-(4-chloro-1H-pyrazol-1-yl)acetyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
1-{3-[(4-methoxyphenyl)methyl]-5-[(methylsulfanyl)methyl]-1H-1,2,4-triazol-1-yl}butan-2-ol
6-methyl-2-[6-oxo-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-2-yl]pyridine-3-carbonitrile
6-chloro-4-[2-(3-methyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]-2-(1H-pyrazol-4-yl)quinoline
2-(3-methoxypropyl)-9-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
2-methoxy-N-{1-[4-(3-propoxypiperidine-1-carbonyl)phenyl]-1H-pyrazol-4-yl}acetamide
N-benzyl-4-(3-methylpyridin-4-yl)piperazine-1-sulfonamide
1-[2-(4-methoxyphenyl)ethyl]-N-[(3-methyloxetan-3-yl)methyl]-6-oxopiperidine-3-carboxamide
2-tert-butyl-6-(3,5-difluoro-4-methoxybenzoyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
N-[2-(dimethylamino)ethyl]-5-(isoquinolin-1-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
6-[4-methoxy-2-(1H-pyrazol-1-yl)phenyl]pyridine-2-carboxamide
(4aS,8aR)-6-[(1-methyl-1H-imidazol-2-yl)methyl]-1-(2-phenylethyl)-decahydro-1,6-naphthyridin-2-one
N-[(1-methyl-1H-imidazol-2-yl)(phenyl)methyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
N-{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-1-(pyridin-3-ylmethyl)piperidin-4-amine
4-{1-[1-(2-fluorophenyl)-1H-1,2,4-triazol-5-yl]propyl}morpholine
{[2-(adamantan-1-yl)-1,3-thiazol-4-yl]methyl}[2-(1H-1,2,4-triazol-1-yl)propyl]amine
3-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]-1-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidine
N-[2-(1,3-benzothiazol-2-yl)ethyl]-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
2-[methyl({4-methyl-5-[1-(1H-1,2,4-triazole-5-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)amino]ethan-1-ol
1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidine
6-ethyl-4-(piperidine-1-carbonyl)-2-(1H-pyrazol-4-yl)quinoline
2-methoxy-1-{1'-[(2-methoxy-4-methylphenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
9-cyclopropanecarbonyl-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
N-(1-{1-[3-(5-methylfuran-2-yl)butyl]piperidin-4-yl}-1H-pyrazol-5-yl)pyridine-3-carboxamide
2-({[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)-1,3-thiazole-4-carboxamide
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-[2-(4-fluorophenyl)ethyl]piperidine
1-[1-(3-methoxypropanoyl)piperidin-4-yl]-N-(2-phenylethyl)piperidine-4-carboxamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-[2-(1H-imidazol-1-yl)acetyl]pyrrolidin-3-yl]-5-methyl-1,3-oxazole-4-carboxamide
methyl 4-({methyl[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]amino}methyl)-1H-pyrazole-3-carboxylate
2-[2-chloro-4-({[(3-ethyl-1,2-oxazol-5-yl)methyl](methyl)amino}methyl)phenoxy]acetamide
3-(2-ethyl-1H-imidazol-1-yl)-1-[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]propan-1-one
4-{2-amino-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl}-6-fluoro-1,2-dihydroquinolin-2-one
5-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-N,N-dimethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-{2-[(3,5-dimethyladamantan-1-yl)oxy]ethyl}-4H-1,2,4-triazole
N-[(3R,4S)-1-acetyl-4-cyclopropylpyrrolidin-3-yl]-2-(2,2,6,6-tetramethylpiperidin-4-yl)acetamide
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(1H-imidazol-2-ylmethyl)-N-methylacetamide
N-(2,3-dihydro-1H-inden-2-yl)-5-(methoxymethyl)-N-propylfuran-2-carboxamide
2-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}quinoxaline
2-(4-{[5-(2-chlorophenyl)furan-2-yl]methyl}-1-(1-methylpiperidin-4-yl)piperazin-2-yl)ethan-1-ol
1-(3,4-dihydro-2H-1-benzopyran-3-yl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
3-{3-[cyclohexyl(methyl)amino]propyl}-8-(3-hydroxypropyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(2S)-2-amino-N-[(4-ethylphenyl)methyl]-N-(2-methoxyethyl)-3-(1,3-thiazol-4-yl)propanamide
(4aS,8aR)-1-(3-methoxypropyl)-6-(2-methoxypyridine-4-carbonyl)-decahydro-1,6-naphthyridin-2-one
N-[2-(1H-indol-1-yl)ethyl]-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
N-[2-(1,3-thiazol-4-yl)ethyl]-1-(4,6,7-trimethylquinazolin-2-yl)piperidin-4-amine
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-(pyrrolidine-1-carbonyl)-decahydro-1,6-naphthyridin-2-one