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4-[(4-fluorophenyl)methyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
dimethyl({[4-({2-phenylimidazo[1,2-a]pyrimidin-3-yl}methyl)-1,4-oxazepan-6-yl]methyl})amine
5-(1-{4-[1-(4-methoxyphenyl)-1H-imidazol-2-yl]-1H-1,2,3-triazol-1-yl}ethyl)-1,3,4-thiadiazol-2-amine
4-(2H-1,3-benzodioxol-4-ylmethyl)-7-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-[(4aS,8aR)-decahydroisoquinolin-2-ylmethyl]-N-(1,5-dimethyl-1H-pyrazol-4-yl)benzamide
1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]-2-(1-propylpiperidin-4-yl)ethan-1-one
1-(1-cyclopropanecarbonylpiperidin-4-yl)-2-(3,4-dimethoxyphenyl)-5-fluoro-1H-1,3-benzodiazole
N-butyl-2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-(furan-2-ylmethyl)acetamide
6-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carboxylic acid
N-benzyl-N-(cyclobutylmethyl)-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
2-(dimethyl-1,3-thiazol-5-yl)-N-methyl-N-[1-(pyridin-2-yl)ethyl]acetamide
N-[(4-fluorophenyl)methyl]-N-(oxolan-2-ylmethyl)-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
4-methyl-1-{3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}pentane-1,2-dione
N-methyl-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]-N-[1-(pyridin-4-yl)ethyl]acetamide
5-chloro-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-4-ylmethyl)furan-2-carboxamide
1-(5-methanesulfonyl-2-methylphenyl)-3-{2-[(trifluoromethyl)sulfanyl]ethyl}urea
(3aS,6aR)-3-[2-(3-chlorophenyl)ethyl]-5-(9H-purin-6-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-[({3-[2-hydroxy-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propoxy]phenyl}methyl)amino]propane-1,3-diol
3-(1-ethyl-1H-1,2,3,4-tetrazol-5-yl)-1-{2-[3-(trifluoromethyl)phenyl]ethyl}urea
dimethyl[3-({5-[2-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]pyridin-2-yl}oxy)propyl]amine
(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-6-[(3-phenyl-1,2-oxazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
3,5,7-trimethyl-2-[4-(thian-4-yl)piperazine-1-carbonyl]-1H-indole
{[5-(1-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}piperidin-4-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}dimethylamine
(1R,5S)-3-{[2-(4-chlorophenyl)pyrimidin-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[5-(2-hydroxyethyl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl]benzoic acid
1-methyl-4-({[4-(trifluoromethyl)pyridin-2-yl]amino}methyl)piperidin-4-ol
1-({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-4-(piperidin-1-yl)piperidine-4-carboxamide
3-{[3-(2-methylpropyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-3,4-dihydroquinazolin-4-one
4-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]-1-(4-methylphenyl)pyrrolidin-2-one
N-(3-methoxypropyl)-N-(1-methylpiperidin-4-yl)-3-(pyridin-4-yl)propanamide
6-(oxolane-2-carbonyl)-N-(3-phenylpropyl)-6-azaspiro[2.5]octane-1-carboxamide
4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]-1-[2-(pyrrolidin-3-yl)benzoyl]piperidine
1-{3-[(3,4-difluorophenyl)amino]piperidin-1-yl}-4-phenylbutane-1,4-dione
2-(4-methyl-1,2,5-oxadiazol-3-yl)-N-[(6-methylquinolin-5-yl)methyl]acetamide
3-(2,3-dihydro-1H-isoindol-2-yl)-1-{8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}propan-1-one
1-{1-[(8-methoxy-2H-chromen-3-yl)methyl]piperidin-3-yl}-4-(2-methylphenyl)piperazine
3-[5-(morpholin-4-ylmethyl)pyridin-2-yl]benzoic acid
N-(2-hydroxyethyl)-2-methyl-N-{[4-(methylsulfanyl)phenyl]methyl}pyridine-3-carboxamide
2-methyl-N-[2-(1-oxo-1,2-dihydrophthalazin-2-yl)ethyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
(3R,4S)-1-(4-chloro-1-methyl-1H-pyrrole-2-carbonyl)-4-propylpyrrolidin-3-amine
4-{[(4aS,7aR)-4-(2-hydroxyethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]methyl}benzonitrile
2-(1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carbonyl)-1,2,3,4-tetrahydroisoquinoline
7-({4-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)-2,7-diazaspiro[4.4]nonane-1,3-dione
N-cyclopentyl-6-[4-(2-methoxyethyl)piperazine-1-carbonyl]-5-methylthieno[2,3-d]pyrimidin-4-amine
5-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyrazin-2-ol
(1S,5R)-6-(cyclobutylmethyl)-3-(3-hydroxy-2-methylbenzoyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
8-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
2-{[3-(3-chlorobenzoyl)piperidin-1-yl]methyl}-4-methoxyphenol
3-[(2-fluorophenyl)formamido]-N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}propanamide
2-{[(1R,2R,4R)-bicyclo[2.2.1]hept-5-en-2-ylformamido]methyl}-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide