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3-methyl-4-[3-(propan-2-yl)-1,2-oxazol-5-yl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-cyclopropyl-2-(dimethylamino)-2-(2-fluorophenyl)-N-(pyridin-3-ylmethyl)acetamide
2-(4-cyclohexyl-1,4-diazepane-1-carbonyl)-5-methoxy-1-methyl-1H-indole
(1S,6R)-9-{2,3-dimethyl-5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carbonyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
5-(2-{[(3-methylphenyl)methyl]amino}ethyl)-1-[3-(methylsulfanyl)propyl]pyrrolidin-2-one
2,7-dimethyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}pyrazolo[1,5-a]pyrimidine-5-carboxamide
5-{[(butan-2-yl)(cyclopentyl)amino]methyl}-N-ethylpyrimidin-2-amine
4-(5-methyl-1,2,4-oxadiazol-3-yl)-1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperidine
4-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrole-1-carbonyl]-2,6-dimethylquinoline
3-(oxolan-3-yl)-5-(2,4,5-trimethoxyphenyl)-1,2,4-oxadiazole
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[2-(4-hydroxypiperidin-1-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-3,5-dimethoxybenzamide
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-1-phenyl-1H-pyrazole-4-carboxamide
(3R,4S)-1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-amine
3-(2-fluorophenyl)-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)propanamide
8-(2,3-difluoro-4-methoxybenzoyl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-1,4-oxazepan-5-one
N,2-dimethyl-6-(piperidin-3-yl)-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}pyrimidin-4-amine
5-{furo[3,2-c]pyridin-4-yl}-N-(2-hydroxyethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
4-benzyl-3-{1-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
6-methyl-2-(2-phenylethyl)-1-(pyridin-2-ylmethyl)-3-(pyrrolidine-1-carbonyl)-1,4-dihydropyridin-4-one
methyl (3aS,6aS)-2-methyl-5-[2-methyl-2-(morpholin-4-yl)propyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylate
N3-{2-[5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-yl]ethyl}piperidine-1,3-dicarboxamide
1-cycloheptyl-5-[4-(3-methoxypropyl)piperidine-1-carbonyl]piperidin-2-one
N-(1H-1,3-benzodiazol-2-ylmethyl)-N-methyl-1,2,3,4-tetrahydronaphthalene-2-carboxamide
2-{3-cyclopentyl-5-[3-(1H-1,2,3,4-tetrazol-1-yl)phenoxymethyl]-1H-1,2,4-triazol-1-yl}acetic acid
methyl 4-({1-[2-(3-fluorophenyl)ethyl]-6-oxopiperidin-3-yl}formamido)butanoate
1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
(2S,4R)-4-amino-N-ethyl-1-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)pyrrolidine-2-carboxamide
N-{4-[(benzyloxy)methyl]-7-methoxy-2-oxo-1,2,3,4-tetrahydroquinolin-6-yl}-2,2-dimethylpropanamide
N-{2-methyl-1-[7-(3-phenylpropyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]propyl}methanesulfonamide
(4aS,7aR)-1-[(3-cyclohexyl-1,2-oxazol-5-yl)methyl]-4-ethyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]-4-(pyrimidin-2-yl)-1,4-diazepane
3-{[(4-fluorophenyl)methyl]sulfanyl}-N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)propanamide
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-1-(oxan-4-yl)piperidine
1-{1-[(3-ethyl-1,2-oxazol-5-yl)methyl]-4-phenylpiperidin-4-yl}ethan-1-one
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-3-(2-fluorophenyl)-3-phenylpropanamide
N-{2-[2-(benzyloxy)acetamido]-5-methoxyphenyl}-2-methylpropanamide
[(1-cyclopentylpiperidin-4-yl)methyl]({[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl})(oxolan-2-ylmethyl)amine
2-(2-chlorophenyl)-2-hydroxy-1-(4-{[1,2,4]triazolo[4,3-a]pyrimidin-5-yl}piperazin-1-yl)ethan-1-one
(3S,4R)-1-(4-chloro-1H-pyrazole-3-carbonyl)-4-(3-methylthiophen-2-yl)piperidin-3-ol
methyl 3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxylate
2-cyclopropyl-9-(pyrimidin-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
5-acetyl-N-[3-methyl-1-(pyridin-3-yl)butyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
6-ethyl-3-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3H,4H-thieno[2,3-d]pyrimidin-4-one
2-[1-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)pyrrolidin-2-yl]pyridine
4-(4-chlorobenzoyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-[4-(furan-2-ylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
2-[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-3-yl]-1H-1,3-benzodiazole
5-(4-{2-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl}phenyl)-1H-pyrazole