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9-(1-methyl-6-oxo-1,6-dihydropyridine-3-carbonyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
(3R,4R)-1-(6-aminopyrimidin-4-yl)-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-3-ol
3-(1-cyclohexyl-1H-pyrazol-5-yl)-1-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]urea
3-[1-(cyclopropylmethyl)-1H-pyrazol-5-yl]-1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)urea
1-(2-{[1-(6-ethyl-2-methylpyrimidin-4-yl)piperidin-4-yl]amino}ethyl)-4,6-dimethyl-1,2-dihydropyrimidin-2-one
4-(3-fluorophenyl)-N-{[3-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)benzamide
7-cyclopropanecarbonyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
3-chloro-N-(2,2-dimethylpropyl)-4-[(1-methanesulfonylpiperidin-4-yl)oxy]benzamide
8-fluoro-3-[2-(2-hydroxyethoxy)ethyl]-3,4-dihydroquinazolin-4-one
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-5-(3-hydroxy-3-methylbut-1-yn-1-yl)furan-2-carboxamide
1-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-3-[3-(3-methyl-2-oxoimidazolidin-1-yl)phenyl]urea
3-[(1-methylpiperidin-4-yl)methyl]-3H,4H-pyrido[4,3-d]pyrimidin-4-one
1-(4-{[(1S)-2-hydroxy-1-phenylethyl]amino}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
2-{[({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)amino]methyl}-3-methoxyphenol
3-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-1-(4-oxo-4H-chromen-6-yl)urea
(2S,4S)-4-amino-1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-benzyl-2-[2-(dimethylamino)ethyl]-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
(4S)-1-[2-(benzyloxy)benzoyl]-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]({[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
1-({4-[(2R,5S)-2,5-dimethylpyrrolidine-1-carbonyl]-1,3-oxazol-2-yl}methyl)-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine
(1S,5R)-3-[(4-methoxyphenyl)methyl]-6-(1H-pyrazole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-4-(thiophen-2-ylmethyl)piperazine
methyl 1-[2-(1H-indol-3-yl)ethyl]-3-(3-methoxypropanamido)-5-{[(6-methylpyridin-2-yl)methyl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
8-{4-[(butylsulfanyl)methyl]-5-methylfuran-2-carbonyl}-2-methyl-2,8-diazaspiro[4.5]decan-3-one
3-{[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]methyl}-1-(2-methyl-1H-1,3-benzodiazol-6-yl)urea
3,3,3-trifluoro-N-[(3R,4S)-1-[(3-methylpyrazin-2-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]propanamide
1-methyl-4-{1-[1-(1,3-thiazole-4-carbonyl)piperidin-4-yl]piperidine-3-carbonyl}piperazine
1-[benzyl(methyl)amino]-3-(4-{[(naphthalen-1-ylmethyl)amino]methyl}phenoxy)propan-2-ol
8-[2-(2-chlorophenyl)-2-hydroxyacetyl]-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-(1H-indol-3-yl)acetamide
4-methoxy-1-{2-phenyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidine
2-(4-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-1H-pyrazol-1-yl)propanamide
5-{[1-(4-phenylpiperazine-1-carbonyl)-6-azaspiro[2.5]octan-6-yl]methyl}-2,1,3-benzothiadiazole
N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(1H-imidazol-2-yl)benzamide
1-[(3R,4S)-3-amino-4-propylpyrrolidine-1-carbonyl]naphthalen-2-ol
1-{[2-(4-chlorophenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}piperidin-3-ol
ethyl 1-(4-acetylbenzenesulfonyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
1'-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)-5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-({[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}amino)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
5-acetamido-1-ethyl-2-(2-fluorophenyl)-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-1H-1,3-benzodiazole-7-carboxamide
5-methyl-3-[3-methyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]-4,5,6,7-tetrahydro-2H-indazole
2-[2-(morpholin-4-yl)ethyl]-N-(naphthalen-1-yl)piperidine-1-carboxamide
(2S,4S)-4-amino-1-(8-hydroxy-5,7-dimethylquinoline-2-carbonyl)-N-methylpyrrolidine-2-carboxamide
7-(cyclohexylmethyl)-2-[(3-hydroxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
6,7-dimethoxy-2-[3-(pyridin-3-yl)propyl]quinazolin-4-amine
ethyl 4-[({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(2-methoxyethyl)amino]piperidine-1-carboxylate
3,5-dimethyl-N-[4-(pyridin-2-yl)butyl]-1,2-oxazole-4-carboxamide
1-cyclopentyl-N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-6-oxopiperidine-3-carboxamide
2-(1H-pyrazol-1-ylmethyl)-4-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}-1,4-oxazepane
(9aR)-8-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione