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8-methoxy-2-{[4-(oxan-4-yl)piperazin-1-yl]methyl}quinoline
2-[2-(morpholin-4-yl)ethyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-3-methylpyrazine
2-(cyclopentylmethyl)-6-methyl-3-(4-phenylazepane-1-carbonyl)-1-(pyridin-3-ylmethyl)-1,4-dihydropyridin-4-one
7,8-dimethyl-4-(2-methylpyrrolidine-1-carbonyl)-2-(1-propyl-1H-pyrazol-4-yl)quinoline
1-{3-[2-(4-fluoropiperidin-1-yl)-2-oxoethyl]morpholin-4-yl}-3-(pyridin-3-yl)propan-1-one
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
1-[(4S)-4-hydroxy-3,3,4-trimethylpiperidin-1-yl]-3-(2-methyl-1H-1,3-benzodiazol-1-yl)propan-1-one
4-methoxy-2-{[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]methyl}phenol
({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)[(4-methoxyphenyl)methyl]methylamine
N-[1-(cyclohex-1-en-1-yl)ethyl]-1-(propan-2-yl)-1H-pyrazole-5-carboxamide
5-methoxy-2-{[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-4H-pyran-4-one
N-[(1-benzylpiperidin-4-yl)methyl]-N-methylmorpholine-2-carboxamide
3,5-dimethyl-4-(1-{5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl}pyrrolidin-2-yl)-1,2-oxazole
3-{3-[({2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}amino)methyl]-1H-indol-1-yl}propanamide
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N-methyl-1-[(4-methylphenyl)methyl]-5-oxopyrrolidine-3-carboxamide
[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl](methyl)[1-(pyridin-3-yl)ethyl]amine
8-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-3-(2-phenylpropyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-[(dimethylamino)methyl]-N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}benzamide
N-(1-cyclopentyl-4-methyl-1H-pyrazol-5-yl)-3-methoxypropanamide
N-(1-cyclopropanecarbonylpiperidin-3-yl)-6-(propan-2-yl)pyrimidin-4-amine
4-{3-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}-6-methyl-1,2-dihydroquinolin-2-one
1-(cyclohex-1-en-1-ylmethyl)-3-[6-(dimethylamino)-1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl]urea
1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-(hydroxymethyl)azepan-4-ol
3-({2-[1-(3-methylthiophene-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
5-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidine-1-carbonyl}-3-methyl-2,3-dihydro-1,3-benzoxazol-2-one
N-{[5-(4-chlorophenyl)-1,2-oxazol-3-yl]methyl}-3-(1-methylpiperidin-2-yl)propanamide
2-cyclopropyl-5-[4-(3-phenylpropyl)-1,4-diazepane-1-carbonyl]-3,4-dihydropyrimidin-4-one
N-(3-hydroxy-2,2-dimethylpropyl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
4-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-2-ethyl-1-(propan-2-yl)piperazine
N-(furan-2-ylmethyl)-4-methyl-3-(2-oxoimidazolidin-1-yl)-N-(prop-2-en-1-yl)benzamide
1-(1H-imidazol-2-ylmethyl)-4-(quinolin-6-yloxy)piperidine-4-carboxylic acid
3-[(4-cyclopentylpyrimidin-2-yl)(methyl)amino]-2,2-dimethylpropan-1-ol
3-{[1-butyl-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]methyl}-2,3-dihydro-1H-isoindol-1-one
ethyl 3-(3-phenylpropyl)-1-[2-(1H-pyrazol-1-yl)acetyl]piperidine-3-carboxylate
N-cyclobutyl-5-[1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)pyrrolidin-2-yl]thiophene-2-carboxamide
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-[(3R,4R)-3-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]ethan-1-one
1-(but-3-enoyl)-N-[3-(1H-indol-2-yl)phenyl]piperidine-3-carboxamide
(3aR,6aR)-2-methanesulfonyl-5-(pyridin-3-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[(1S,5R)-3-(2,6-dimethylpyrimidine-4-carbonyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
3-(2-ethoxypyridin-3-yl)-6-methylpyridin-2-amine
2-[4-(4-ethoxyphenyl)-1H-imidazol-2-yl]-4-methoxyphenol
2-(4-fluorophenyl)-N-[3-(propan-2-yloxy)propyl]imidazo[1,2-a]pyridine-6-carboxamide
N-({3-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)acetamide
1-(1-ethyl-1H-pyrazole-3-carbonyl)-3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine
3,5-dimethyl-4-{1-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]pyrrolidin-2-yl}-1,2-oxazole
1-(2,3-dihydro-1-benzofuran-5-ylmethyl)-N-[2-(pyridin-3-yloxy)phenyl]piperidine-3-carboxamide
N-(2,3-dimethylphenyl)-2-{2-[2-(pyridin-2-yl)pyrimidin-5-yl]-1H-imidazol-1-yl}acetamide
1-(2-{[(5-fluoro-3-methyl-1H-indol-2-yl)methyl](methyl)amino}ethyl)piperidin-2-one
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-[2-(3-oxopiperazin-1-yl)acetyl]-decahydro-1,6-naphthyridin-2-one