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(3S,4R)-1-(2,5-dimethylfuran-3-carbonyl)-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
2-{1-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]-N-methylformamido}-2-(pyridin-3-yl)acetic acid
1-ethyl-3-[(3-methoxyphenyl)methyl]-8-[(1-methyl-1H-indol-3-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(dimethylamino)-2-(4-fluorophenyl)-N-{3-[(1-methylpiperidin-4-yl)oxy]propyl}acetamide
6-ethyl-4-({[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]amino}methyl)-2H-chromen-2-one
(1R,5S,6S)-N-(adamantan-1-yl)-3-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-azabicyclo[3.1.0]hexane-6-carboxamide
N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2-methyl-1-benzofuran-5-carboxamide
N-(1-{[4-(2-phenylethoxy)phenyl]methyl}pyrrolidin-3-yl)acetamide
N-[(1-{5-[(methylsulfanyl)methyl]pyridin-2-yl}piperidin-4-yl)methyl]acetamide
(4aR,8aS)-1-[(3,4-dimethoxyphenyl)methyl]-6-(thiophen-3-ylmethyl)-decahydro-1,6-naphthyridin-2-one
3-benzyl-4-[(2-methyl-1,3-oxazol-4-yl)methyl]piperazin-2-one
8-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-2-(dimethylamino)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
N-[2-(3-methoxyphenyl)phenyl]-1-(3-methylbutyl)piperidine-4-carboxamide
2-ethyl-1-[(4-methoxyphenyl)methyl]-6-methyl-3-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]-1,4-dihydropyridin-4-one
3-({1-[3-(3-methoxyphenyl)phenyl]piperidin-4-yl}amino)-1-methylpyrrolidin-2-one
N,N-dimethyl-5-({[3-(pyrrolidin-1-yl)propyl]carbamoyl}amino)-1-benzothiophene-2-carboxamide
(1S,6R)-9-[2-(2-hydroxyphenyl)-6-methylpyrimidin-4-yl]-3-methyl-3,9-diazabicyclo[4.2.1]nonan-4-one
N-[(3S,4R)-1-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
N-(1-{1-[(4,5-dimethylfuran-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methoxy-2-phenylacetamide
2-(3,4-dichlorophenyl)-4-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]morpholine
2-(methylsulfanyl)-5-({2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}methyl)pyrimidine
4-(2-methoxyphenoxy)-1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperidine-4-carboxylic acid
N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-1-(2-methyl-6-propylpyrimidin-4-yl)piperidin-4-amine
[(3R,4S)-1-[(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
4-ethyl-6-[4-(5-phenyl-1,2-oxazole-3-carbonyl)piperazin-1-yl]pyrimidine
(2S,4R)-4-amino-N-ethyl-N-{[2-(prop-2-en-1-yloxy)phenyl]methyl}pyrrolidine-2-carboxamide
3-(2-methoxyethyl)-5-{6-methylimidazo[1,2-a]pyridin-2-yl}-1,2,4-oxadiazole
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}acetamide
5-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazol-4-yl}-3-propyl-1,2,4-oxadiazole
4-[2-(1-{imidazo[1,2-a]pyridine-6-carbonyl}piperidin-2-yl)ethyl]phenol
1-tert-butyl-4-{[methyl({1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl})amino]methyl}pyrrolidin-2-one
N-(2,3-dihydro-1H-inden-2-yl)-2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}acetamide
6-[(3R,5S)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
6-[ethyl(methyl)amino]-N-[(3-propyl-1,2-oxazol-5-yl)methyl]pyridine-3-carboxamide
1-methyl-1-(2-oxo-2-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethyl)urea
1-cyclopropanecarbonyl-N-{6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidin-3-amine
1-cyclopentyl-N-[2-(quinolin-8-yloxy)ethyl]piperidine-3-carboxamide
4-(benzyloxy)-1-(1-methanesulfonylpyrrolidine-2-carbonyl)piperidine
2-(quinolin-3-yl)pyridine-4-carbonitrile
N-(2-methylpropyl)-1-[(1s,4s)-4-(4-methoxybenzamido)cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N,8-dimethyl-3-[(2-methylpyrrolidin-1-yl)methyl]-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
N-[2-(3-methoxyphenyl)-1-[1-(6-methylpyridine-2-carbonyl)piperidin-4-yl]ethyl]-N,1-dimethyl-1H-pyrazole-3-carboxamide
2-[3-(trifluoromethoxy)phenyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
(3S,4R)-3-ethyl-4-methyl-1-(9-methyl-9H-carbazole-3-carbonyl)piperidin-4-ol
N-[(3S,4R)-1-{3-[4-(dimethylamino)phenyl]propanoyl}-4-propylpyrrolidin-3-yl]acetamide
(2S,4R)-N-[2-(2-fluorophenyl)ethyl]-1-(propan-2-yl)-4-[(1-propylpiperidin-4-yl)amino]pyrrolidine-2-carboxamide
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-3-yl}propanamide
3-(1-cycloheptylpiperidin-3-yl)-1-methyl-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[3-(1H-imidazol-1-yl)propyl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
3-[2-(1H-pyrazol-1-yl)ethyl]-7-thia-2,4,5-triazatricyclo[6.4.0.02,6]dodeca-1(12),3,5,8,10-pentaene