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4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-[(2,3-dimethoxyphenyl)methyl]piperidine
1-{5-[(2-chlorophenyl)methyl]-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperidin-3-ol
8-(1,4-dioxan-2-ylmethyl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
dimethyl(3-{2-[1-(3-methylpyridin-4-yl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)amine
(2R,6S)-4-{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}-2,6-dimethylmorpholine
4-{[(1R,3S,5S)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl]methyl}-N-(3-methoxyphenyl)benzamide
2-benzyl-N-(1H-indol-2-ylmethyl)-1,3-benzoxazole-5-carboxamide
9-(but-3-yn-1-yloxy)-7-(5-methylthiophen-2-yl)-4-(propan-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-[1-(2,5-difluorophenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]cyclopropane-1-carboxamide
6-[4-(hydroxymethyl)-4-(3-phenylpropyl)piperidin-1-yl]pyridine-2-carbonitrile
1-(1-{[2-(difluoromethoxy)phenyl]methyl}piperidin-3-yl)-4-(4-methoxyphenyl)piperazine
2-[3-(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]pyridine-3-carboxamide
N-(carbamoylmethyl)-2-{4-[(2-methoxyquinolin-3-yl)methyl]morpholin-3-yl}acetamide
2-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}acetamide
3-[5-(6-phenylpyridine-2-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
2-(ethoxymethyl)-N-[1-(thiophen-2-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
9-[(2S)-2-amino-3-hydroxypropanoyl]-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-(4-{[3-(2-hydroxyethyl)-4-(2-methylpropyl)piperazin-1-yl]methyl}phenoxy)ethan-1-ol
2-methyl-6-({[4-(pyridin-2-yl)pyrimidin-2-yl]amino}methyl)pyrimidin-4-ol
[(3R,4S)-1-[(2,4-difluorophenyl)methyl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
(3S,4S)-1-(1-ethylpiperidine-4-carbonyl)-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
2-(4-{[3-(pyridin-3-ylmethoxy)piperidin-1-yl]methyl}phenyl)pyridine
1-[1-(3-cyanophenyl)-3-(1-hydroxycyclopentyl)prop-2-yn-1-yl]piperidine-4-carboxamide
2-[(isoquinolin-5-yloxy)methyl]-N-[2-(3-methylpyridin-2-yl)ethyl]-1,3-oxazole-4-carboxamide
1-({1-[(4-chlorophenyl)methyl]-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl}methyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N-methyl-3-(4-methyl-1,3-thiazol-5-yl)propanamide
2-{3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}acetamide
2-[(1-acetylpiperidin-4-yl)oxy]-5-methoxy-N-(1-phenylbutyl)benzamide
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-1-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]ethan-1-one
2-{[(3S,4R)-4-amino-3-methoxypiperidin-1-yl]methyl}-3,5-dimethoxybenzoic acid
6-methyl-1-(oxan-2-ylmethyl)-4-(trifluoromethyl)-1,2-dihydropyridin-2-one
2-{9-[2-(3-methoxyphenyl)acetyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetamide
(3S)-N-tert-butyl-2-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
1-(2-{1-[2-(benzyloxy)acetyl]piperidin-2-yl}ethyl)pyrrolidin-2-one
3-[2-(3-acetyl-4-hydroxyphenyl)ethyl]-1λ6-thiolane-1,1-dione
N-(1-ethyl-1H-1,2,3-triazol-4-yl)-2-[4-(6-methoxypyridazin-3-yl)-1H-pyrazol-1-yl]acetamide
5-{[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
2-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1-methyl-1H-indole
4-(benzyloxy)-N-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]butanamide
N-[3-(4-chloro-3-methylphenoxy)-2-hydroxypropyl]-3-ethyl-1H-pyrazole-4-carboxamide
3-hydroxy-1-[(3-methoxyphenyl)methyl]-3-({[2-(3-methyl-1H-pyrazol-1-yl)ethyl]amino}methyl)piperidin-2-one
5-[2-(5-methyl-1,2-oxazol-3-yl)piperidine-1-carbonyl]-N-phenylpyrimidin-2-amine
5-[4-(pyridin-2-ylmethyl)-1,4-diazepane-1-carbonyl]pyridin-2-amine
N-[(3R,5S)-5-(4,4-difluoropiperidine-1-carbonyl)pyrrolidin-3-yl]-2-phenylacetamide
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-5-hydroxypyrazine-2-carboxamide
2-(benzyloxy)-1-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-9-yl]ethan-1-one
4-(3-hydroxy-3,4,4-trimethylpyrrolidine-1-carbonyl)oxane-4-carbonitrile
2-{3-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidine-1-carbonyl]phenoxy}acetamide
3-[(3R,4S)-1-[(2-fluorophenyl)carbamoyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-1-{2-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-amine