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N-{1-[1-(2,1,3-benzoxadiazol-4-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-phenylbutanamide
N-(1-ethyl-1H-pyrazol-5-yl)-2-[4-(5-ethylpyrimidin-2-yl)-1H-pyrazol-1-yl]acetamide
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-4-(dimethylamino)butanamide
N-({5-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
N-methyl-5-[1-(piperidin-1-yl)ethyl]-N-(thiophen-3-ylmethyl)furan-2-carboxamide
2-(acetamidomethyl)-N-(2-methoxy-5-methylphenyl)-1-oxa-8-azaspiro[4.5]decane-8-carboxamide
2-{6-oxa-9-azaspiro[4.5]decan-9-ylmethyl}benzoic acid
3-({2-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidin-1-yl}methyl)-1,2-dihydroquinolin-2-one
1-[3-(2-fluorophenyl)benzoyl]-4-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1,4-diazepan-5-one
methyl 1-[(3S,5S)-5-(azepane-1-carbonyl)-1-(3-methylbut-2-en-1-yl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
8-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)-1-oxa-8-azaspiro[4.6]undecane
{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}(methyl){[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-{3-[(4-chlorophenyl)sulfanyl]propyl}-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
4-[4-(4-ethoxyphenyl)-1H-imidazol-2-yl]piperidine
2-[2-(dimethylamino)ethyl]-9-(4-fluoro-3-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-3-[1-(2-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)piperidin-3-yl]-N-[2-(pyridin-2-yl)ethyl]propanamide
(4aS,8aS)-4a-hydroxy-N-(5-methyl-1,3,4-thiadiazol-2-yl)-decahydroisoquinoline-2-carboxamide
2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]-N-(2-hydroxyethyl)-N-methylacetamide
7-(2-methylphenyl)-4-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-(2-chlorophenyl)-1-(2-methoxyethyl)-3-{2-oxo-2-[4-(thiomorpholin-4-yl)piperidin-1-yl]ethyl}pyrrolidine-2,5-dione
2-({5-[(N-methylmethanesulfonamido)methyl]-4-phenyl-4H-1,2,4-triazol-3-yl}sulfanyl)acetic acid
4-(2-fluorophenoxy)-1-{2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidine
N-[(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-3-yl)methyl]-2H-1,3-benzodioxole-5-carboxamide
N-[4-(2-hydroxyethyl)phenyl]-4-[(3-oxopiperazin-1-yl)methyl]benzamide
8-[2-(2-phenyl-1,3-thiazol-4-yl)acetyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
2-{2-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-1-yl]-2-oxoethyl}-1,2-dihydrophthalazin-1-one
3-{3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]propyl}-1H-indole
(2S)-N-[3-fluoro-5-(trifluoromethyl)phenyl]-2-(methoxymethyl)pyrrolidine-1-carboxamide
N-[4-(3-methoxyphenyl)phenyl]-1-(1-methylpiperidin-4-yl)pyrrolidine-2-carboxamide
1-(2,4-dimethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)-3-methyl-3-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)urea
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}acetamide
(2S,4S)-N-ethyl-4-[3-(1-methyl-1H-pyrazol-4-yl)propanamido]-1-(oxan-4-yl)pyrrolidine-2-carboxamide
3-{[1-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-4-yl]oxy}-N-cyclopropyl-4-methoxybenzamide
2-(1-ethylpiperidin-4-yl)-N-[phenyl(pyridin-4-yl)methyl]acetamide
1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperidine-3-carboxamide
5-methyl-N-{4-[2-methyl-3-(1H-pyrazol-1-yl)propanamido]phenyl}furan-3-carboxamide
2,6-dimethyl-8-{[(1-phenylpyrrolidin-3-yl)methyl]amino}octan-2-ol
4-({[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}(oxolan-2-ylmethyl)carbamoyl)pyridin-1-ium-1-olate
N-(2-hydroxyethyl)-N-{[4-(methylsulfanyl)phenyl]methyl}-6-oxo-1,6-dihydropyridine-3-carboxamide
1-(2,1,3-benzothiadiazol-5-ylmethyl)-4-[(2-fluorophenyl)methyl]-1,4-diazepan-5-one
2-(4-chlorophenyl)-4-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]morpholine
2-{1-[4-(5-methylfuran-2-yl)benzoyl]piperidin-2-yl}pyridine
N-(2,1,3-benzothiadiazol-5-ylmethyl)-7-fluoro-N,2-dimethylquinoline-4-carboxamide
{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amine
N-(2,4-dimethoxyphenyl)-3-[1-(thiophene-3-carbonyl)piperidin-4-yl]propanamide
N-[2-(1,3-benzothiazol-2-yl)ethyl]-2-(2,5-dioxoimidazolidin-1-yl)acetamide
1-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}piperidin-4-ol
N-[1-methyl-4-(pyridin-3-yloxy)-1H-indazol-3-yl]-2-(methylsulfanyl)acetamide
1-(3-chlorophenyl)-4-[3-(3-hydroxy-1,2-oxazol-5-yl)propanoyl]-5-methylpiperazin-2-one
1-(pyridin-2-ylmethyl)-N-[4-(pyridin-3-yloxy)phenyl]piperidine-4-carboxamide