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N,N-dimethyl-3-({1-oxa-8-azaspiro[4.5]decan-3-yl}sulfamoyl)benzamide
N-[4-(3-fluorophenyl)phenyl]-1-(1-methylpiperidin-4-yl)pyrrolidine-2-carboxamide
N-({6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[2,1-b][1,3]thiazol-5-yl}methyl)-1-phenylcyclopropan-1-amine
2-amino-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-6-(thiophen-2-yl)pyridine-3-carbonitrile
4-(1-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-4-phenyl-1H-imidazol-5-yl)benzonitrile
5-{2-[(prop-2-en-1-yl)amino]ethyl}-1-(thiophen-2-ylmethyl)pyrrolidin-2-one
N-(3-chloro-4-fluorophenyl)-3-[1-(pyridine-3-carbonyl)piperidin-4-yl]propanamide
1-(2H-1,3-benzodioxol-5-yl)-N-[1-(3-methylpyridin-2-yl)propan-2-yl]piperidin-4-amine
5-(morpholin-4-ylmethyl)-N-[1-(pyrimidin-2-yl)piperidin-3-yl]furan-3-carboxamide
5-cyclopropyl-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-N-(1-methoxypropan-2-yl)-1H-pyrazole-4-carboxamide
(2E)-1-[4-(hydroxymethyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidin-1-yl]-4-methylpent-2-en-1-one
4-{[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]sulfamoyl}-N-(propan-2-yl)benzamide
7-(propan-2-yl)-N-[1-(pyrimidin-2-yl)piperidin-3-yl]-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
5-[3-(methoxymethyl)piperidine-1-carbonyl]-N-(2-methylprop-2-en-1-yl)pyridin-2-amine
5-methoxy-9-(quinoxaline-6-carbonyl)-1-oxa-9-azaspiro[5.5]undecane
6-methoxy-3-methyl-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-1-benzofuran-2-carboxamide
[(4-chloro-1-methyl-1H-indazol-3-yl)methyl](methyl)[2-(2-methyl-1H-imidazol-1-yl)ethyl]amine
N4-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-N2,N2-dimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
(3aS,6aR)-5-[(3,4-difluorophenyl)methyl]-3-[2-(4-methoxyphenyl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
3-[4-(piperidin-4-yl)piperazin-1-yl]-1,2-benzothiazole
(2,1,3-benzoxadiazol-5-ylmethyl)(methyl){[5-(oxolan-2-yl)thiophen-2-yl]methyl}amine
methyl 5-[2-oxo-2-(pyridin-3-yl)acetyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
6-({[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}amino)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
N-methyl-4-oxo-1-(2-phenylethyl)-5-(4-phenylpiperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
7-(cyclobutylmethyl)-2-(1-methyl-1H-pyrrole-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-phenyl-2-({[2-(1H-1,2,4-triazol-1-yl)pyridin-3-yl]methyl}amino)butanamide
N-(3,4-diethyl-1-methyl-1H-pyrazol-5-yl)-3-[(2-methylpyrrolidin-1-yl)methyl]benzamide
N-[(3-methoxyphenyl)methyl]-N-propyloxan-4-amine
1-[3-(2-methyl-1,3-thiazol-4-yl)phenyl]-4-(pyrrolidin-1-yl)piperidine
N-[(3S,4R)-4-(4-methoxyphenyl)-1-(1-methyl-1H-pyrrole-2-carbonyl)pyrrolidin-3-yl]acetamide
3-[2-(dimethylamino)ethyl]-3,4-dihydroquinazolin-4-one
N,2-dimethyl-N-[1-(1,2-oxazol-3-yl)ethyl]-1-phenyl-1H-1,3-benzodiazole-5-carboxamide
2-(5-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}-1H-pyrazol-3-yl)phenol
1-[3-({[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)phenyl]ethan-1-one
ethyl 3-{[7-(pyridine-2-amido)-1,2,3,4-tetrahydroisoquinoline-2-carbonyl]amino}propanoate
N-{[2-(dimethylamino)-7-methylquinolin-3-yl]methyl}-N-[2-(4-fluorophenyl)ethyl]-2,2-dimethyloxane-4-carboxamide
N-(1-benzylpyrrolidin-3-yl)-1-(6-chloropyridazin-3-yl)piperidin-4-amine
N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-(pyridin-2-yl)acetamide
(3aR,6aR)-2-cyclopentyl-5-[3-(dimethylamino)pyrazin-2-yl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(furan-2-ylmethyl)-2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)-N-(prop-2-en-1-yl)acetamide
(1S,5R)-6-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
N-{[4-hydroxy-1-(thiophene-2-carbonyl)azepan-4-yl]methyl}-2,5-dimethylfuran-3-carboxamide
4-fluoro-N-{2-[2-(3-hydroxy-4-methoxyphenyl)-1H-imidazol-1-yl]ethyl}benzamide
N-phenyl-3-({[3-(piperidin-1-ylmethyl)phenyl]carbamoyl}amino)propanamide
N-{[4-fluoro-7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,2-diphenylacetamide
2-{[({5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl}methyl)(methyl)amino]methyl}-6-methoxyphenol
1-ethyl-4-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,2-dihydropyridin-2-one
3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)propanamide
2-[(1S,5R)-3-[4-(dimethylamino)-5-methylpyrimidin-2-yl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
3-[3-cyclopropyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]-4-methylbenzene-1-sulfonamide