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N-methyl-N-[2-(2-methylphenyl)-1-{1-[3-(4-methylphenyl)propanoyl]piperidin-4-yl}ethyl]cyclobutanecarboxamide
N-[3-(furan-2-yl)phenyl]-1-(morpholine-4-carbonyl)piperidine-4-carboxamide
(2S,4R)-4-[2-(2,4-difluorophenoxy)acetamido]-N,N-diethyl-1-methylpyrrolidine-2-carboxamide
[(3R,4S)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-[(4-methoxy-3-methylphenyl)methyl]pyrrolidin-3-yl]methanol
1-ethyl-4-[2-(2-methoxy-4-methylphenoxymethyl)-1,3-oxazole-4-carbonyl]piperazin-2-one
6-{4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-9H-purine
N-methyl-3-(1-methyl-1H-pyrazol-4-yl)-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}propanamide
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-4-hydroxybenzamide
4-(5-{[({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl)amino]methyl}thiophen-2-yl)-2-methylbut-3-yn-2-ol
2-[4-(2,2-diphenylethyl)morpholin-2-yl]ethan-1-amine
N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-4-(2-oxopyrrolidin-1-yl)butanamide
1-[(4aS,8aS)-4a-hydroxy-7-(1H-imidazol-4-ylmethyl)-decahydro-2,7-naphthyridin-2-yl]-2-propoxyethan-1-one
1-{1-[(2-methyl-1,3-thiazol-4-yl)methyl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-N,3,6-trimethyl-1-benzofuran-2-carboxamide
5-fluoro-N,3-dimethyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1H-indole-2-carboxamide
[(3R,4R)-1-(3,4-difluorobenzenesulfonyl)-4-[(dimethylamino)methyl]pyrrolidin-3-yl]methanol
methyl 9-(2,3-dihydro-1H-inden-2-yloxy)-3-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
[1-(2-{[2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}ethyl)piperidin-2-yl]methanol
2-{1-cyclohexyl-4-[4-(methylamino)-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl]piperazin-2-yl}ethan-1-ol
4-{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}morpholine
methyl 6-benzyl-2-[(1-methoxypropan-2-yl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-(4-{[4-(difluoromethoxy)phenyl]methyl}-1-(2-methylpropyl)piperazin-2-yl)ethan-1-ol
5-(3-methoxyphenyl)-N-[(5-methylpyrazin-2-yl)methyl]-1,2,4-triazin-3-amine
N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
5-{2-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-2-oxoethyl}-2-methyl-3,4-dihydropyrimidin-4-one
N-[(2-methoxyphenyl)methyl]-5-methyl-N-(prop-2-en-1-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
[1-(1-benzoylpiperidin-4-yl)-3-(prop-2-en-1-yl)piperidin-3-yl]methanol
(1S,6R)-9-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
1-(3-chloro-2-fluorophenyl)-3-{[1-(hydroxymethyl)cyclopentyl]methyl}-3-methylurea
3-ethoxy-N-[1-(4-fluorophenyl)-4-(morpholin-4-yl)-1H-indazol-3-yl]propanamide
3-(3-{1-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyridine
N-ethyl-2,5-dimethyl-N-(pyridin-4-ylmethyl)-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
1-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-3-(4-ethyl-1,3-dimethyl-1H-pyrazol-5-yl)-1-methylurea
9-(4-methoxy-2-methylbenzoyl)-1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane
4-{4-[5-(pyrrolidin-2-yl)thiophene-2-carbonyl]piperazin-1-yl}quinazoline
9-(furan-3-carbonyl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
5-acetyl-N-[(1R,3S)-3-{[(2-methylphenyl)methyl]carbamoyl}cyclopentyl]thiophene-2-carboxamide
14-(1-benzofuran-2-yl)-5-methyl-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
2-(3-chlorophenyl)-5-methyl-4-(pyrrolidin-1-ylmethyl)-1,3-oxazole
2-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
N-(3-chloro-4-propanamidophenyl)-4-(pyrrolidin-1-yl)butanamide
4-[6-(2-fluoro-5-methoxyphenyl)pyrazine-2-carbonyl]morpholine
2-[2-methyl-3-({[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]amino}methyl)-1H-indol-1-yl]acetamide
1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-4-(naphthalen-2-yl)piperazine
2-{2-[1-(3-methylbutan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1H-pyrrol-1-yl}-1,3-thiazole
2-methyl-9-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}acetyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(3-{4-[(1,4-dioxan-2-ylmethyl)(methyl)amino]piperidin-1-yl}phenyl)-3-(trifluoromethyl)benzamide
6-[4-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
(1S,5R)-3-(1,3-dihydroxypropan-2-yl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
[(3R,4R)-1-{6-chloro-3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol