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N-{[6,7-dimethoxy-2-(3-methoxyphenyl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)cyclohexanecarboxamide
3-{2-[7-(hydroxymethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-oxoethyl}-3,4-dihydroquinazolin-4-one
2-[(3-fluorophenyl)methyl]-4-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}morpholine
(1R,5R)-6-(3-methylbut-2-en-1-yl)-3-(pyridine-3-sulfonyl)-3,6-diazabicyclo[3.2.2]nonane
4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidine
1-[(1R,3S,5S)-3-(4-fluoro-3-methylphenyl)-8-azabicyclo[3.2.1]octan-8-yl]-3-(4-methylpiperazin-1-yl)propan-1-one
(1R,5R)-6-[6-(methoxymethyl)pyridine-2-carbonyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(2-propyl-1,3-thiazole-4-carbonyl)piperidine
1-({3-[3-(4-ethylpiperazin-1-yl)-2-hydroxypropoxy]phenyl}methyl)piperidine-4-carbonitrile
[(2-chlorophenyl)methyl](2-methoxyethyl){[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amine
1-(3-{[2-(2-methoxyethyl)piperidin-1-yl]methyl}phenyl)ethan-1-one
N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
4-{4-[methyl(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)amino]piperidin-1-yl}-N-[(3S)-2-oxoazepan-3-yl]benzamide
(5S)-5-{[benzyl({4-[(thiophen-2-ylmethyl)amino]quinazolin-2-yl}methyl)amino]methyl}pyrrolidin-2-one
N-[(3S)-2-oxoazepan-3-yl]-N-{[4-(propan-2-yloxy)phenyl]methyl}pyridine-2-carboxamide
1-[2-hydroxy-5-(2-methylbutan-2-yl)phenyl]-5-oxopyrrolidine-3-carboxylic acid
5-chloro-6-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carboxylic acid
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-(6-methoxypyrimidin-4-yl)-2,8-diazaspiro[4.5]decan-3-one
1-(naphthalen-1-ylmethyl)-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-1H-1,2,3-triazole-4-carboxamide
1-(4-chlorophenyl)-N-({1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperidin-3-yl}methyl)cyclopropane-1-carboxamide
N-(3-sulfamoylphenyl)-2-(1,3-thiazol-2-yl)piperidine-1-carboxamide
1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-4-(4-methoxybenzoyl)piperazine
(3S)-3-[(5-{3-[(4-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)amino]azepan-2-one
3-(5-{1-[2-(1H-indol-3-yl)ethyl]-1H-imidazol-2-yl}thiophen-2-yl)prop-2-yn-1-ol
(3S,4R)-1-(2,3-dihydro-1-benzofuran-7-carbonyl)-3-methoxypiperidin-4-amine
3-{[4-(5-tert-butyl-1H-pyrazol-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}pyridine
3-[(dimethylamino)methyl]-1-{1,3,6-trimethyl-1H-pyrazolo[3,4-b]pyridine-4-carbonyl}piperidin-3-ol
methyl 1-[3-(2-{[4-(methylsulfanyl)phenyl]methyl}-5-oxopyrrolidin-2-yl)propanoyl]piperidine-4-carboxylate
2-[4-(2,5-dimethylbenzoyl)-2-oxopiperazin-1-yl]benzonitrile
3-(benzyloxy)-1-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}piperidine
N-(isoquinolin-5-ylmethyl)-N-methyl-1,2,3,4-tetrahydronaphthalene-2-carboxamide
1-(1-benzofuran-5-carbonyl)-3-(2,5-dimethoxyphenyl)pyrrolidine
1-[(5-{[3-(2-fluorophenyl)pyrrolidin-1-yl]methyl}-2-methoxyphenyl)methyl]-1H-1,2,4-triazole
(2S,4R)-4-amino-N,N-diethyl-1-(2-methoxy-5-methylbenzenesulfonyl)pyrrolidine-2-carboxamide
methyl 2-(2-butyl-1H-imidazol-4-yl)-1H-1,3-benzodiazole-6-carboxylate
(3S,4R)-1-(6-aminopyridine-3-carbonyl)-4-(2H-1,3-benzodioxol-5-yl)pyrrolidine-3-carboxylic acid
N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-4-methyl-1H-imidazole-2-carboxamide
2-(2,6-dioxo-1,3-diazinan-1-yl)-N-methyl-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)acetamide
2-[3-(2-fluorophenyl)pyrrolidin-1-yl]-5-(1H-imidazol-1-ylmethyl)pyridine
N-[(3S)-piperidin-3-yl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
(1R,3S)-N1,N1,2,2,3-pentamethyl-N3-[3-(pyridin-3-yloxy)propyl]cyclopentane-1,3-dicarboxamide
N-{[8-(3-methylbut-2-en-1-yl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}-2-(2-oxo-1,2-dihydropyridin-1-yl)acetamide
(3R,9R)-11-(4-phenylbenzoyl)-5-thia-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
1-[2-(1,3-benzothiazol-2-yl)pyrrolidin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
N-(1-{1-[(2,6-dioxo-1,2,3,6-tetrahydropyrimidin-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-methylbutanamide
N-ethyl-N-methyl-2-{[1-(1,4-oxazepan-4-yl)hex-5-en-2-yl]oxy}pyrimidin-4-amine
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]acetamide
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}(1H-imidazol-2-ylmethyl)(oxolan-2-ylmethyl)amine
N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carboxamide