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3-methyl-1-(2-methylphenyl)-5-({[1,2,4]triazolo[4,3-b]pyridazin-6-yloxy}methyl)-1H-1,2,4-triazole
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-(1,3-thiazol-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-{imidazo[1,2-a]pyrimidine-2-carbonyl}-2-(3-methoxyphenyl)azetidine
(1S,5S)-3-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonane
3-(4-fluorophenyl)-N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-N-methyl-1H-pyrazole-5-carboxamide
6-[(diethylamino)methyl]-N-(3-oxo-1,3-dihydro-2-benzofuran-5-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-[1-(cyclohex-1-en-1-yl)ethyl]-4-(4H-1,2,4-triazol-4-yl)benzamide
2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]acetamide
7-{2-[(1S,4R)-2-azabicyclo[2.2.1]heptan-2-yl]acetyl}-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-methoxypropan-1-one
N-cycloheptyl-1-ethyl-3-(4-methyl-1,4-diazepane-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
9-[(2S)-2-hydroxy-2-phenylacetyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-(thiophen-2-ylmethyl)acetamide
2-{1'-[(2-ethylpyrimidin-5-yl)methyl]-2-oxo-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-1-yl}acetamide
2,6-dihydroxy-N-[2-(N-methylmethanesulfonamido)ethyl]benzamide
8-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-[4-(cyclopropylamino)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]-4-(1H-pyrazol-4-yl)butan-1-one
N-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-2-(thiophen-3-yl)acetamide
N2,N2-dimethyl-N4-[1-(oxolan-2-ylmethyl)piperidin-4-yl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
N-[(5-chloro-2-methoxyphenyl)methyl]-N-methyl-2-(2-methyl-5-oxopyrrolidin-1-yl)acetamide
1-cyclopentyl-4-[2-(2,4,6-trifluorophenyl)ethyl]piperazine
(2S,4R)-4-amino-1-{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}-N-(propan-2-yl)pyrrolidine-2-carboxamide
3-(2-fluorophenyl)-N-(2-methoxyethyl)-N-(pyridin-4-ylmethyl)-1H-pyrazole-4-carboxamide
5-benzyl-3-cyclopentyl-5-(piperidin-4-yl)imidazolidine-2,4-dione
3-methoxy-1-(4-{4-methyl-5-[(4-methylpiperazin-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)propan-1-one
N-[2-(dimethylamino)-2-(3-methylphenyl)ethyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
5-(3-acetylphenoxymethyl)-N-[furan-2-yl(phenyl)methyl]-1,2-oxazole-3-carboxamide
3-[5-(oxolan-3-yl)-1H-1,2,4-triazol-3-yl]pyridine
1-{4-[3-(4-ethylpiperazin-1-yl)-3-oxopropyl]piperidin-1-yl}-2-(2-methyl-1H-imidazol-1-yl)propan-1-one
2-ethoxy-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]pyridine-3-carboxamide
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(methylsulfanyl)benzamide
2-({5-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-phenyl-4H-1,2,4-triazol-3-yl}sulfanyl)acetic acid
N-benzyl-2-methanesulfonyl-N-methyl-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
N-{[4-(methylsulfanyl)phenyl]methyl}-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
4-({[1-(2H-1,3-benzodioxol-5-yl)-3-cyclopropyl-1H-1,2,4-triazol-5-yl]methyl}sulfanyl)pyridine
2-[5-(4-chloro-1-methyl-1H-pyrazol-3-yl)-3-[(3,4-dimethoxyphenyl)methyl]-1H-1,2,4-triazol-1-yl]ethan-1-ol
N-[2-(7-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]cyclohexanecarboxamide
1-{[4-(2,5-dimethoxyphenyl)-4H-1,2,4-triazol-3-yl]methyl}-4-(4-fluorophenyl)piperazine
4-{[3-(difluoromethoxy)phenyl]methyl}-9-ethyl-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
(3R,4S)-4-cyclopropyl-1-[1-(4-methylbenzoyl)piperidine-4-carbonyl]pyrrolidin-3-amine
1-[(2E)-3-(3-fluorophenyl)prop-2-enoyl]-4-(2-phenoxyethyl)-1,4-diazepan-5-one
1-[1-(2-methoxyethyl)piperidin-4-yl]-N-(2-phenylethyl)piperidine-3-carboxamide
3-[1-(6-chloropyridazin-3-yl)piperidin-4-yl]-1-methyl-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[(5-chlorofuran-2-yl)methyl]-4-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine
(2R,3R)-3-amino-1'-{[1-(propan-2-yl)piperidin-4-yl]methyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-(1,3-benzothiazol-2-ylmethyl)-N-methyl-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
5-({5-cyclobutanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)pyridin-2-amine
6,8-dimethyl-2-{[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]methyl}quinolin-4-ol
(1S,5R)-6-(2,5-dimethoxybenzenesulfonyl)-3-methyl-3,6-diazabicyclo[3.2.2]nonane
2-({methyl[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]amino}methyl)pyridine-3-carboxylic acid