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4-(1H-pyrazol-1-yl)-1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)piperidine-4-carboxylic acid
1-(2,3-dihydro-1H-inden-2-yl)-4-{imidazo[1,2-a]pyridine-6-carbonyl}-1,4-diazepane
4-(4-hydroxybutyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(3-{[4-(aminomethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-2-(cyclohex-1-en-1-yl)ethan-1-one
5-(2-fluorophenoxymethyl)-N-[1-(2-hydroxyphenyl)ethyl]-1H-pyrazole-3-carboxamide
(3aS,6aS)-2-(dimethylcarbamoyl)-5-[(4-ethylphenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(4aS,8aR)-1-(2-aminoethyl)-6-[2-(thiophen-2-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
2-(2-{[2-(1,3-thiazol-4-yl)ethyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
(1R,5R)-3-[3-(1H-imidazol-2-yl)benzoyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonane
2-({[(6-hydroxy-1,4-oxazepan-6-yl)methyl](methyl)amino}methyl)-3,4-dihydroquinazolin-4-one
N-methyl-2-{5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-5H,6H,7H-cyclopenta[d]pyrimidin-4-amine
(3S,4S)-4-({[(9-ethyl-9H-carbazol-3-yl)methyl]amino}methyl)piperidin-3-ol
4-[1-(4-methoxyphenyl)piperidin-4-yl]-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
N-(1-carbamoylcyclopentyl)-4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzamide
2-cyclopropyl-4-hydroxy-N-{[2-(3-methoxyphenyl)-1,3-thiazol-5-yl]methyl}pyrimidine-5-carboxamide
3-(2-fluorophenyl)-6-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}-1-(pyridin-4-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-{2-[4-(1-methyl-1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]ethyl}aniline
N-(2-fluoroethyl)-3-{[2-(pyrazin-2-yl)ethyl]sulfamoyl}benzamide
2-(dimethylamino)-N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}-2-(3-methylphenyl)acetamide
2-ethyl-4-({4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyrimidine
(3S,4R)-4-(3-methylthiophen-2-yl)-1-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-3-ol
2-methoxy-6-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]phenol
N-[(2-ethyl-4-methyl-1,3-thiazol-5-yl)methyl]-1-(propan-2-yl)piperidine-4-carboxamide
3-({5-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]-1H,4H-pyrazolo[3,4-d]imidazol-1-yl}methyl)pyridine
{[1-(3-fluorophenyl)-3-(5-methylfuran-2-yl)-1H-pyrazol-4-yl]methyl}(pyridin-3-ylmethyl)amine
2-(1,5-dimethyl-1H-pyrazol-4-yl)-1-methyl-5-(pyrrolidine-1-sulfonyl)-1H-1,3-benzodiazole
1-cyclopropyl-5-[4-(morpholin-4-ylmethyl)piperidine-1-carbonyl]piperidin-2-one
N-[2-(5-chloro-4-methyl-1,3-thiazol-2-yl)ethyl]-2-(1-ethylpiperidin-4-yl)acetamide
5-[2-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-2-oxoethyl]-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(2-{2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidine-1-carbonyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl)ethan-1-one
methyl (2S,4R)-4-(2,3-dimethyl-1H-indole-7-amido)-1-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}pyrrolidine-2-carboxylate
1,3-dimethyl-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
(3S,4S)-1-[6-(2-chlorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-4-(propan-2-yloxy)pyrrolidin-3-ol
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-3,6,7-trimethyl-1-benzofuran-2-carboxamide
(4aR,7aS)-1-(pyrimidin-2-yl)-4-(1,3-thiazol-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(5-{[3-(4-chlorophenyl)piperidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)pyridine
N,N,6-trimethyl-2-[2-(pyridin-2-yl)pyrimidin-5-yl]quinoline-4-carboxamide
{[2-(adamantan-1-yl)-1,3-thiazol-4-yl]methyl}({5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl})amine
3-[(1-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-4-yl)oxy]pyridine
N,N-diethyl-1-{[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)carbamoyl]methyl}piperidine-3-carboxamide
2-(2-aminoethyl)-N-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]quinazolin-4-amine
3-(1H-imidazol-2-yl)-N-methyl-N-{[3-(trifluoromethyl)phenyl]methyl}benzamide
methyl 3-[({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(oxolan-2-ylmethyl)carbamoyl]propanoate
4-{1-[3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]cyclohexyl}morpholine
3-(2-{[1-(6-ethyl-2-methylpyrimidin-4-yl)piperidin-4-yl]amino}-1-hydroxyethyl)phenol
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N,1-dimethyl-6-oxo-1,6-dihydropyridazine-3-carboxamide
1-(5-ethylthiophene-3-carbonyl)-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
2-(4-cyclohexyl-3-oxopiperazin-1-yl)-2-(3-hydroxyphenyl)acetic acid
(2S,4S)-4-amino-N-(propan-2-yl)-1-[3-(thiophen-2-yl)-1H-pyrazole-4-carbonyl]pyrrolidine-2-carboxamide
3-[6-amino-2-(morpholin-4-yl)pyrimidin-4-yl]-5-[2-(piperidin-2-yl)ethyl]phenol