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2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-(3-hydroxypropyl)-N-methyl-1,3-oxazole-4-carboxamide
3-(1H-indol-6-yl)-5-[(propan-2-yl)sulfamoyl]benzoic acid
{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
N3-[3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propyl]piperidine-1,3-dicarboxamide
methyl 8-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-1-(naphthalen-2-ylmethoxy)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
1-cycloheptyl-6-oxo-N-[2-(1,3-thiazol-2-yl)ethyl]piperidine-3-carboxamide
1-{3-[2-(4-chlorophenyl)morpholin-4-yl]-3-oxopropyl}piperidin-2-one
5-{1-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}pyrimidin-2-amine
5-ethyl-6-methyl-N4-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)pyrimidine-2,4-diamine
1-[(1S,5R)-3-acetyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(pyridin-3-yl)ethan-1-one
N'-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}pentanediamide
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-7-methylpyrazolo[1,5-a]pyrimidine-6-carboxamide
2-(dimethyl-1,3-thiazol-5-yl)-1-[4-(furan-2-carbonyl)-1,4-diazepan-1-yl]ethan-1-one
4-[3-(2-methoxyethyl)-5-(5-phenyl-1,2-oxazol-3-yl)-1H-1,2,4-triazol-1-yl]-1-methylpiperidine
3-(azepane-1-sulfonyl)-5-(1H-1,2,4-triazol-1-yl)benzoic acid
8-(6-aminopyridine-3-carbonyl)-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
4-(5-{6-[(dimethylamino)methyl]-1,4-oxazepane-4-carbonyl}furan-2-yl)-2-methylbut-3-yn-2-ol
1-(1-methyl-1H-pyrrole-2-carbonyl)-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
7-(2-methoxyethyl)-2-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-2,7-diazaspiro[4.5]decane
(1S,5R)-6-benzyl-3-(quinolin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-cyclohexyl-N-cyclopropyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,3-benzoxazole-6-carboxamide
(3R)-3,4,4-trimethyl-1-(1,3-thiazol-2-ylmethyl)pyrrolidin-3-ol
2,2-dimethyl-5-[3-(pyridin-2-yl)azetidine-1-carbonyl]thiomorpholin-3-one
4-{[7-methoxy-2-(thiophen-2-yl)quinolin-3-yl]methyl}-1-methylpiperazin-2-one
4-{4-[(4-phenyl-4H-1,2,4-triazol-3-yl)methyl]piperidine-1-carbonyl}-1-(prop-2-en-1-yl)pyrrolidin-2-one
1-[(4-fluorophenyl)methyl]-4-(5-methoxypyrimidin-2-yl)-1,4-diazepane
6-cyclopropyl-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methylpyrimidin-4-amine
N-{2-[4-(4-fluorophenyl)-5-{[(2-methylphenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl]ethyl}-4-(1H-pyrazol-1-yl)benzamide
1-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine
3-[1-(2-methoxyethyl)-2-methyl-1H-indol-5-yl]-1-methyl-1-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]urea
N-[1-(4-methoxyphenyl)ethyl]-N,3-dimethylbut-2-enamide
2-[(1-benzyl-1H-imidazol-5-yl)methyl]-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
(3S,9aR)-8-(cyclopropylmethyl)-3-[(4-hydroxyphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-[2-(3-fluoropyridin-4-yl)-4-methylphenoxy]acetamide
2-[2-(2,3-dimethylphenoxy)acetyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
4-(4-{[(1H-imidazol-2-ylmethyl)(methyl)amino]methyl}phenyl)-2-methylbutan-2-ol
(3S)-1-[(1-{[1-(1-methylcyclohexanecarbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]pyrrolidin-3-ol
4-[3-(propan-2-yl)-1H-pyrazol-5-yl]-1-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}piperidine
(3R,4S)-4-cyclopropyl-1-(2-phenoxybenzoyl)pyrrolidin-3-amine
1-(4-methoxyphenyl)-3-methyl-4-(thiophene-3-carbonyl)piperazin-2-one
N-(2-oxo-2,3-dihydro-1H-indol-3-yl)-6-phenylimidazo[2,1-b][1,3]thiazole-3-carboxamide
2-(4-hydroxyphenyl)-2-[4-(thiomorpholin-4-yl)piperidin-1-yl]acetic acid
N-(5-chloro-2-methylphenyl)-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
(3S,5R)-1-[(4,5-dimethylfuran-2-yl)methyl]-5-[(pyridin-3-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
N-[1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-4-methyl-1,2,3-thiadiazole-5-carboxamide
2-amino-N-methyl-6-(2-methylpropyl)-N-[(3-methylthiophen-2-yl)methyl]pyrimidine-4-carboxamide
(3aR,6aR)-2-cyclopropanecarbonyl-5-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-N-(quinolin-2-ylmethyl)propanamide
(3aR,5S,6S,7aS)-2-[4-(4-fluorophenyl)oxane-4-carbonyl]-octahydro-1H-isoindole-5,6-diol
(furan-3-ylmethyl)(methyl)[(3-{[1-(4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)piperidin-4-yl]oxy}phenyl)methyl]amine