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1-cyclohexyl-3-(cyclopropylmethyl)-5-(piperazine-1-carbonyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N-(prop-2-yn-1-yl)cyclohexanamine
4-{[2-(2-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-{4-[2-(ethylamino)pyrimidine-5-carbonyl]piperazin-1-yl}-1-(morpholin-4-yl)ethan-1-one
2-(butan-2-ylsulfanyl)-5-({4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazin-1-yl}methyl)pyrimidine
2-(1-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-2-yl)ethan-1-ol
N-(3-methoxyphenyl)-3-{1-[1-(methylsulfanyl)propan-2-yl]piperidin-4-yl}propanamide
2-(4-{[3-(2-phenylacetyl)piperidin-1-yl]methyl}phenyl)acetic acid
2-[methyl(phenyl)amino]-1-{3-[2-(1,4-oxazepan-4-yl)-2-oxoethyl]morpholin-4-yl}ethan-1-one
7-methoxy-N-{2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethyl}-1,2,3,4-tetrahydronaphthalen-2-amine
3-({methyl[(trimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)-7-(methylsulfanyl)-1,2-dihydroquinolin-2-one
2-(1,2,3,6-tetrahydropyridin-1-yl)-4-(trimethyl-1H-pyrazol-4-yl)pyrimidine
3-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]-3,9-diazaspiro[5.6]dodecan-10-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-(2-methoxy-4-methylphenoxymethyl)-1,3-oxazole-4-carboxamide
{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}(2,1,3-benzoxadiazol-5-ylmethyl)methylamine
5-fluoro-1-methyl-2-{[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]methyl}-1H-indole
8-[(3-methoxyphenyl)methyl]-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
2-methyl-6-[2-(piperidin-1-ylmethyl)phenoxy]-4-(trifluoromethyl)pyridine
3-({4-[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)pyridine
2-(3-{[3-(methoxymethyl)piperidin-1-yl]methyl}phenyl)-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
1-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-3-(1H-pyrazol-1-yl)propan-1-one
N-[2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)ethyl]-1-benzothiophene-2-carboxamide
(2R,3R,6R)-3-(3-methoxyphenyl)-N,N-dimethyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxamide
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}imidazo[1,2-a]pyrimidine-2-carboxamide
2-{1-benzyl-3-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-6-ethoxyphenol
4-methyl-N-{[1-(morpholin-4-yl)cyclopentyl]methyl}pyrimidin-2-amine
N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-4,5,6,7-tetrahydro-1,2-benzoxazole-3-carboxamide
2-(4-acetylphenoxy)-1-{1-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-6-azaspiro[2.5]octan-6-yl}ethan-1-one
N-(propan-2-yl)-6-(1H-pyrazol-3-yl)pyrimidin-4-amine
5-[(3S,4R)-4-amino-3-methoxypiperidine-1-carbonyl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
5-(3-{[(diethylsulfamoyl)amino]methyl}pyrrolidin-1-yl)-2-methyl-2,3-dihydropyridazin-3-one
N-(1,3-dihydro-2-benzofuran-5-yl)-3-({[2-(furan-2-yl)phenyl]methyl}amino)-5-[(propan-2-yl)sulfamoyl]benzamide
6-[4-(1-ethoxyethyl)phenyl]pyridine-2-carboxamide
4-methyl-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperazine-1-sulfonamide
N-ethyl-5-{1-[2-(propan-2-yloxy)ethyl]-1H-1,2,3-triazol-4-yl}pyrimidin-2-amine
N-(4-chloro-3-methoxyphenyl)-2-{cyclopropyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}acetamide
3-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]propanamide
1-(2-{1,8-dioxa-4,11-diazaspiro[5.6]dodecan-4-yl}-2-oxoethyl)-1,2,3,6-tetrahydropyridazine-3,6-dione
N-{5H,6H,7H-cyclopenta[b]pyridin-3-ylmethyl}-6-methyl-4-(3-methylphenyl)-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)[(5-methylfuran-2-yl)methyl]amine
(4aR,8aS)-6-benzyl-1-[4-(2,5-dimethoxybenzoyl)benzoyl]-decahydro-1,6-naphthyridine
2-({3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}methyl)-4,5,6,7-tetrahydro-1,3-benzothiazole
1-(4-aminoazepan-1-yl)-2-(7-fluoro-2-methyl-1H-indol-3-yl)ethan-1-one
1-(4-{[2-(1,3-benzothiazol-2-yl)ethyl]amino}-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
1-[4-(3-hydroxypyrrolidin-1-yl)pyrimidin-2-yl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
3-{[4-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}-3-hydroxy-1-(2-methoxyethyl)piperidin-2-one
1-methyl-4-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine-1-carbonyl}-1,2-dihydroquinolin-2-one
6-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-2,3,4,5-tetrahydropyridazin-3-one
6-fluoro-2-oxo-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1,2,3,4-tetrahydroquinoline-4-carboxamide
butyl (2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxylate