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4-ethyl-3-{[1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
3-[2-(4-fluorophenyl)-2-hydroxyacetyl]-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
1-({3-[3-(methoxymethyl)piperidine-1-carbonyl]-1H-pyrazol-5-yl}methyl)-1H-indole
1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-4-(2-phenylethyl)piperazine
3-[5-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]-N-(propan-2-yl)propanamide
1-{1-[(5-chloro-2-hydroxyphenyl)methyl]piperidin-3-yl}-N,N-diethyl-1H-1,2,3-triazole-4-carboxamide
1-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
4-(6-ethylpyrimidin-4-yl)-1-(2-phenylethyl)piperazin-2-one
(2S,4R)-4-amino-N,N-diethyl-1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)pyrrolidine-2-carboxamide
1-(2-chlorophenyl)-4-(2-hydroxypropanoyl)piperazin-2-one
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-[2-(N-methylmethanesulfonamido)ethyl]acetamide
4-[(2-methoxypyridin-3-yl)methyl]-1-methyl-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine-2,5-dione
3-(1-{1-[(4-phenylphenyl)methyl]-1H-1,2,3,4-tetrazol-5-yl}piperidin-3-yl)propanamide
2-(2H-1,3-benzodioxol-5-yl)-1-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]ethan-1-one
1-(4-{1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-1H-pyrazol-3-yl)-1H-1,2,3,4-tetrazole
1-{imidazo[1,2-b]pyridazin-6-yl}-4-[(4-methoxy-2,5-dimethylphenyl)methyl]piperazine
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-6-yl}acetamide
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-ylmethyl}-3-(5-methylfuran-2-yl)-1-phenyl-1H-pyrazole
(3S,4S)-1-[(3-phenoxyphenyl)methyl]-4-(piperidin-1-yl)pyrrolidin-3-ol
5-benzyl-1-(3-methoxyphenyl)-4-propylpiperazin-2-one
N-[1-benzyl-6-(propan-2-yloxy)-1H-indazol-3-yl]-1,2-oxazole-3-carboxamide
5-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-3-cyclopropyl-1-phenyl-1H-1,2,4-triazole
3-[1-(propan-2-yl)-1H-1,2,3-triazol-4-yl]-1-{1-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}urea
1'-(2,4-difluoro-3-methoxybenzoyl)-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
2-(2,5-dioxoimidazolidin-4-yl)-N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
3-(2-oxo-2-{spiro[azepane-4,2'-chromene]-1-yl}ethyl)imidazolidine-2,4-dione
7-(3-chlorophenyl)-4-[(1-methyl-1H-imidazol-5-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-{4H,5H,6H,7H,8H-cyclohepta[b]thiophene-2-carbonyl}-4-(1-ethyl-1H-imidazol-2-yl)piperidine
2-[2-(1H-imidazol-4-yl)ethyl]-8-(pyrazine-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
1-(2-butoxyacetyl)-N-(4-fluorophenyl)piperazine-2-carboxamide
5-({[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl](methyl)amino}methyl)-N-ethylpyrimidin-2-amine
5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]-N-[2-(pyrazin-2-yl)ethyl]pyridin-2-amine
[(2S,6S)-11-methoxy-4-(pyridin-3-ylmethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
N-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}-1-[4-(morpholine-4-carbonyl)phenyl]piperidin-4-amine
N-[(3,5-dimethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-3-(4,5,6,7-tetrahydro-2H-indazol-3-yl)propanamide
N-cyclopropyl-5-phenyl-N-(1,3-thiazol-2-ylmethyl)-1H-pyrazole-3-carboxamide
N-(carbamoylmethyl)-2-[2-methyl-4-oxo-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
1-cyclohexyl-N-methyl-N-[(2-phenyl-1,3-thiazol-5-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
N-[1-(5,6,7,8-tetrahydronaphthalen-2-yl)ethyl]thian-4-amine
[3-(2-phenylethyl)-1-[6-(propan-2-yl)pyridazin-3-yl]piperidin-3-yl]methanol
4-[(1E)-3-[4-benzyl-3-(2-hydroxyethyl)piperazin-1-yl]prop-1-en-1-yl]-2-methoxyphenol
8-methoxy-2-(2-methoxyphenyl)-5-[(6-methylpyridin-2-yl)methyl]-2,3,4,5-tetrahydro-1,5-benzothiazepine
5-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]pyrimidine
2-{1-[(4-ethoxyphenyl)methyl]-4-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
8-{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-(ethoxymethyl)-N-(5-fluoro-2-methoxyphenyl)pyrrolidine-1-carboxamide
N-{[7-(5-acetyl-2-fluorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(dimethylamino)acetamide
2-[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]-6-(propan-2-yl)pyridine-3-carbonitrile
5-fluoro-2-[1-(5-methyl-1,3-oxazole-4-carbonyl)piperidin-2-yl]-1H-1,3-benzodiazole
4-benzyl-3-[1-(2,5-dimethylfuran-3-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one