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3-(5-chloro-2-methoxybenzoyl)-1-(oxan-4-yl)piperidine
methyl (2R,4S)-4-hydroxy-1-{[3-hydroxy-5-(hydroxymethyl)-2-methylpyridin-4-yl]methyl}piperidine-2-carboxylate
3-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1H-pyrazol-5-amine
methyl 4-[(4-{3-[(2-methoxyethyl)carbamoyl]phenoxy}piperidin-1-yl)methyl]benzoate
1-{3-[(3-fluorophenyl)amino]piperidin-1-yl}-4-(4-methoxyphenyl)butane-1,4-dione
(4aR,7aS)-1-(2-methylpropyl)-4-({7-oxo-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl}methyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[3-(4-methyl-1,3-thiazol-2-yl)propyl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
N-[(5-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)methyl]methanesulfonamide
1-[2-(3,3-diphenylpiperidin-1-yl)-2-oxoethyl]-1,2-dihydropyrimidin-2-one
5-[(3-benzyl-1H-1,2,4-triazol-5-yl)methyl]imidazolidine-2,4-dione
(1S,5R)-3-(thiophen-3-ylmethyl)-3,9-diazabicyclo[3.3.2]decan-10-one
2-(2-methoxyethyl)-8-[3-(thiophen-3-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
(butan-2-yl)({[5-(1H-pyrazol-5-yl)thiophen-2-yl]methyl})(pyridin-4-ylmethyl)amine
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-{2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperazine
4-{5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-1H-pyrazole-3-carbonyl}thiomorpholine
1-ethyl-3-methyl-N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]piperidine-3-carboxamide
2-{3-[4-(1,3-thiazol-2-yl)piperazine-1-carbonyl]piperidin-1-yl}acetamide
methyl 2-(2,3-dimethylphenyl)-1H-1,3-benzodiazole-6-carboxylate
3-{3-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl}benzoic acid
3-(1H-imidazol-4-yl)-2-[3-(4-methyl-1,3-thiazol-5-yl)propanamido]propanoic acid
1-(1-methyl-1H-imidazole-2-carbonyl)-4-{[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]methyl}piperidine
2-amino-4-(dimethyl-1,3-thiazol-5-yl)-6-(thiophen-3-yl)pyridine-3-carbonitrile
N-(1-phenylethyl)-7-(pyridin-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-(cyclohexylmethyl)-3-hydroxy-3-(piperidin-1-ylmethyl)piperidin-2-one
5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-(2,2,2-trifluoroethyl)-1,2-oxazole-3-carboxamide
2-methyl-4-propyl-6-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
5-[4-(azepane-1-carbonyl)-6-fluoroquinolin-2-yl]pyrimidin-2-amine
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}oxane-4-carbonitrile
1-(2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}-5-methylphenyl)-3,5-dimethyl-1H-pyrazole
{1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-4-(3-phenylpropyl)piperidin-4-yl}methanol
[(3R,4R)-4-[(dimethylamino)methyl]-1-[1-(4-fluoro-2-methylphenyl)piperidin-4-yl]pyrrolidin-3-yl]methanol
1'-(4,5-dimethylthiophene-2-carbonyl)-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-butyl-4-{[2-(3,4-dimethoxyphenyl)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
2-methoxy-4-[3-(3-methoxyphenoxymethyl)piperidine-1-carbonyl]pyridine
N-[(3R,4S)-1-acetyl-4-cyclopropylpyrrolidin-3-yl]-1-methylcyclopentane-1-carboxamide
(2E)-1-[3-(3-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-(1H-imidazol-4-yl)prop-2-en-1-one
4-{1-[1-(1H-1,2,4-triazole-5-carbonyl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
2-amino-1-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]ethan-1-one
N,N-dimethyl-5-(naphthalen-1-ylmethyl)-1-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-(3-propoxypiperidine-1-carbonyl)pyridazine
N-methyl-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-[1-(1,3-thiazol-2-yl)ethyl]-1,2-oxazole-3-carboxamide
7-[(6-ethoxypyridin-3-yl)methyl]-N-(2-methoxyethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-(cyclohex-1-en-1-yl)-7-(2-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N,2-dimethyl-2-{methyl[(7-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]amino}propanamide
(3S,4S)-4-(dimethylamino)-1-[5-(3-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]pyrrolidin-3-ol
3-methyl-N-[(2R,3R)-2-(pyridin-3-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]butanamide
5-(4-chlorophenyl)-N-methyl-N-[2-(4-methylphenoxy)ethyl]-1,2,4-triazin-3-amine
6-[3,5-difluoro-4-(pyrrolidin-1-ylmethyl)phenoxy]pyridine-2-carbonitrile
1-(cyclohexylmethyl)-3-hydroxy-3-{[methyl(pyridin-3-ylmethyl)amino]methyl}piperidin-2-one
2-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-6-methoxyphenol