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4-(4-butyl-1H-1,2,3-triazol-1-yl)-1-(2-methylbutyl)piperidine
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide
N-[(2,5-dimethylphenyl)(pyridin-3-yl)methyl]-4-(4H-1,2,4-triazol-4-yl)benzamide
methyl({5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)(quinoxalin-6-ylmethyl)amine
(4aR,6R,8aS)-2-(1H-imidazol-2-ylmethyl)-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinoline
5-(cyclopropylamino)-1-methyl-N-[(5-methylfuran-2-yl)methyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[(5-chloro-3-methyl-2-phenyl-1H-indol-7-yl)methyl]-2,4-dimethyl-1,3-oxazole-5-carboxamide
4-[(4-methoxy-2,3-dimethylphenyl)methyl]-7-(pyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}-2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetamide
2-{[(3R,4R)-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1-methylpyrrolidin-3-yl]formamido}acetamide
N-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
(2S,4R)-N-ethyl-4-(2-hydroxy-3-methylbenzamido)-1-(1H-imidazol-2-ylmethyl)pyrrolidine-2-carboxamide
1-(1-methyl-1H-pyrazole-5-carbonyl)-3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine
3-[(4,6-dimethylpyrimidin-2-yl)methyl]-1-[4-(2-methylpropoxy)phenyl]urea
1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-(1,3-thiazol-2-yl)piperazine
3-[(3S,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-(pyridin-2-ylmethyl)piperidin-3-yl]-N-(2-methylpropyl)propanamide
2-{[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]amino}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
3-[6-amino-5-cyano-4-(1-methyl-1H-pyrazol-4-yl)pyridin-2-yl]benzoic acid
1-(2,3-dihydro-1H-inden-2-yl)-4-[(2,4-dimethoxyphenyl)methyl]piperazine
8-(2-ethoxyphenyl)quinolin-4-amine
2-(1-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)-1,3-benzoxazole
9-{3-[4-(dimethylamino)phenyl]propanoyl}-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
N-[3-(difluoromethoxy)phenyl]-3-(morpholine-4-carbonyl)piperidine-1-carboxamide
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-7-methyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carboxamide
N-(2,2-difluoro-2H-1,3-benzodioxol-5-yl)-2-(3-methyl-1H-1,2,4-triazol-5-yl)pyrrolidine-1-carboxamide
1-[(2,2-diphenylcyclopropyl)methyl]-4-(2-methoxyethoxy)piperidine
1-[1-(3-methoxy-5-methylthiophene-2-carbonyl)piperidin-4-yl]-2-phenylethan-1-ol
5-chloro-4,6-dimethyl-3-[(1R,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1,2-dihydropyridin-2-one
1,4-dimethyl-9-{[4-(2-methylpropyl)phenyl]methyl}-1,4,9-triazaspiro[5.5]undecane
4-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)thiomorpholine
5-chloro-2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-(1,4-dioxan-2-ylmethyl)benzamide
2-(morpholin-4-yl)-1-(4-{1H-pyrazolo[3,4-b]pyridin-1-yl}phenyl)ethan-1-ol
{4-[(2-chlorophenyl)methyl]-1-[(2-methylphenyl)methyl]piperidin-4-yl}methanol
1-(5-methoxy-2-{1-oxa-7-azaspiro[3.5]nonan-7-ylmethyl}phenoxy)-3-(pyrrolidin-1-yl)propan-2-ol
1-(4-methoxyphenyl)-2,2-dimethyl-4-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}piperazine
(4aS,7aR)-1-(2-chlorobenzoyl)-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(3R,4S)-3-amino-4-propylpyrrolidin-1-yl]-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]ethan-1-one
3,5-difluoro-N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methylpyridine-2-carboxamide
N-ethyl-2-[(8-hydroxyquinolin-7-yl)formamido]propanamide
2-{[(1-{6-methylpyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidin-3-yl)oxy]methyl}pyridine
4-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}({[2-(methylsulfanyl)pyrimidin-5-yl]methyl})amine
N-({1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-3-yl}methyl)quinoline-8-sulfonamide
2,4-dioxo-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}-1,2,3,4-tetrahydropyrimidine-5-carboxamide
4-{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}-1,2-dimethylpiperazine
2-(5-ethoxyfuran-2-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
(4aR,7aS)-1-(2-phenylethyl)-4-(pyridine-4-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-chloro-N-[(2,6-difluorophenyl)methyl]-5-acetamidobenzamide
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]imidazo[1,2-a]pyridine-6-carboxamide
5-(2-chloroprop-2-en-1-yl)-7-{[(naphthalen-1-ylmethyl)amino]methyl}-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one