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(3R,4R)-1-[(3-cyclohexyl-1,2-oxazol-5-yl)methyl]-4-ethylpiperidine-3,4-diol
(3S)-3-benzyl-4-(4-hydroxy-2-phenylpyrimidine-5-carbonyl)piperazin-2-one
9-[(2-chlorophenyl)methanesulfonyl]-1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-2-(1H-imidazol-4-yl)-N-methylacetamide
1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-hydroxy-4-(methylsulfanyl)butan-1-one
[2-(azepan-1-yl)ethyl][(5-tert-butyl-1H-pyrazol-3-yl)methyl]ethylamine
3-propyl-4-{[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}morpholine
(1R,5S,8R)-3-[(2-ethylpyrimidin-4-yl)methyl]-8-methoxy-3-azabicyclo[3.2.1]octane
2-[(dimethylamino)methyl]-4-[1-(propan-2-yl)-1H-imidazol-2-yl]phenol
(3R,4S)-3,4-dimethyl-1-[3-(1H-pyrazol-1-yl)propyl]piperidin-4-ol
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-1-[(3-methoxyphenyl)methyl]-N-methyl-6-oxopiperidine-3-carboxamide
N-ethyl-N-methyl-2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]acetamide
2-{[1-ethyl-3-(hydroxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-8-fluoroquinolin-4-ol
2-methyl-4-{3-[2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane-4-carbonyl]phenyl}but-3-yn-2-ol
4-(1-{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-3-carbonyl)morpholine
1-[2-hydroxy-3-(3-{[methyl(thian-4-yl)amino]methyl}phenoxy)propyl]piperidin-4-ol
7-[2-(1H-pyrazol-1-yl)butanoyl]-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
methyl[(4-methyl-1H-imidazol-2-yl)methyl][(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]amine
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2,5-dimethylbenzamide
N-[1-(cyclohexylmethyl)piperidin-3-yl]-2-(quinazolin-4-yloxy)acetamide
1-methyl-4-[1-(1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-4-yl)ethyl]piperazine
N-[3-(4-hydroxypiperidin-1-yl)propyl]-4-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl)methyl]benzamide
(4aR,7aS)-1-cyclopropanecarbonyl-4-[2-(6-methylpyridin-2-yl)ethyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-(1,5-dimethyl-1H-pyrazol-4-yl)-N-[(1-methylpiperidin-3-yl)methyl]-1,2-oxazole-3-carboxamide
1-[4-(thiomorpholine-4-carbonyl)phenyl]imidazolidine-2,4-dione
3-{[methyl({3-[(4-methylphenyl)sulfanyl]propyl})amino]methyl}piperidin-3-ol
N-benzyl-1-[2-(3-fluorophenyl)ethyl]-N-(2-hydroxyethyl)-6-oxopiperidine-3-carboxamide
2-(4-methoxyphenyl)-N-{[4-(morpholin-4-yl)phenyl]methyl}acetamide
3-{[(4-fluorophenyl)methyl]sulfanyl}-N-[(3-propyl-1,2-oxazol-5-yl)methyl]propanamide
1-(morpholin-4-yl)-2-{3-oxa-9-azaspiro[5.5]undecan-9-yl}ethane-1,2-dione
1-[(2-methylphenyl)methyl]-N-[2-(2-oxoimidazolidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3,3-dimethyl-1-(1-methyl-1H-pyrrole-2-carbonyl)-4-(morpholin-4-ylmethyl)piperidin-4-ol
1-{2-methoxy-4-[(4-methylpiperidin-1-yl)methyl]phenoxy}-3-(thiomorpholin-4-yl)propan-2-ol
ethyl 1-(3-fluoro-4-methoxybenzoyl)-4-(2-phenylethyl)piperidine-4-carboxylate
3-chloro-5-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
4-(5-{[(1H-imidazol-2-ylmethyl)(methyl)amino]methyl}thiophen-2-yl)-2-methylbut-3-yn-2-ol
4-(5-{[(3-fluorophenyl)carbamoyl]amino}-1H-pyrazol-1-yl)-N-(propan-2-yl)piperidine-1-carboxamide
2-(2-amino-6-oxo-1,6-dihydropyrimidin-4-yl)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}acetamide
3-{4-[4-(azetidine-1-carbonyl)phenoxy]piperidine-1-carbonyl}pyridine
5-{1-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-1H-imidazol-2-yl}-2-(pyrrolidin-1-yl)pyrimidine
2-(4-fluorophenyl)-4-[3-(1,3-thiazole-2-carbonyl)pyridin-2-yl]morpholine
3-{[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]methyl}-N-methyl-1,2,4-oxadiazole-5-carboxamide
1-[(2-chlorophenyl)methyl]-N-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-1H-1,2,3-triazole-4-carboxamide
{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}({[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl})amine
(1R,2R,6S,7S)-4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-4-azatricyclo[5.2.1.02,6]decane
2-{4-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]piperazin-1-yl}pyrazine
2-amino-6-(furan-2-yl)-4-[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]pyridine-3-carbonitrile
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[1-(1,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1,3-oxazole-4-carboxamide
3-(propan-2-yl)-5-{1-[2-(propan-2-yl)-1H-imidazol-1-yl]ethyl}-1,2,4-oxadiazole
2-(benzylsulfanyl)-5-{[3-(4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}pyrimidine