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1-benzyl-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-1H-pyrazole-4-carboxamide
ethyl({[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl})(pyridin-4-ylmethyl)amine
N-methyl-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propanamide
N-{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-N-methyloxolan-3-amine
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepine-3-carboxamide
3-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1-(1H-indazol-4-yl)urea
1'-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-methyl-6-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridazine
3-(3-hydroxyquinoxalin-2-yl)-N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]propanamide
1-[4-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)piperidin-1-yl]-2-(1,3-thiazol-4-yl)ethan-1-one
1-(2-{4-[1-(4-methylpiperazin-1-yl)ethyl]piperidin-1-yl}-2-oxoethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
(2S,4S)-4-[(4-methylpyrimidin-2-yl)sulfanyl]-N-(propan-2-yl)-1-{[3-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxamide
7-{imidazo[1,2-b]pyridazine-3-carbonyl}-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
(2S,6S)-1-(furan-2-carbonyl)-4-methyl-2,6-bis(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
3-[3-(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)-1,2,4-oxadiazol-5-yl]benzonitrile
N-[(5-ethylpyridin-2-yl)methyl]-N-methyl-1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
3-[1-(oxolane-3-carbonyl)piperidin-4-yl]-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
1-(2,2-diphenylethyl)-3-(pyrrolidin-1-yl)piperidine
3-{[1-(4-ethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1H-pyrazole
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-(pyrrolidin-1-ylmethyl)piperidin-2-one
1-[3-({4-[1-(2-methylphenyl)-1H-pyrazol-4-yl]pyrimidin-2-yl}amino)propyl]pyrrolidin-2-one
3-(4-fluorophenyl)-N-[3-(methylsulfanyl)propyl]-1H-pyrazole-5-carboxamide
2-[2-oxo-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]-5-(piperidin-1-yl)-2,3-dihydropyridazin-3-one
1-methyl-4-[1-(4-methylphenyl)piperidin-4-yl]-1,4,9-triazaspiro[5.6]dodecan-10-one
2-[6-(4,4-diphenylpiperidin-1-yl)pyrimidin-4-yl]ethan-1-amine
3-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)-1-(1,3-thiazol-2-ylmethyl)urea
1-(1,3-thiazol-4-ylmethyl)-4-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]piperazine
2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(morpholin-4-yl)propyl]acetamide
3-{3-[methyl(2-methylpropyl)amino]propyl}-8-(1-methylpiperidine-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-methyl-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
(2S,4R)-1-benzyl-4-[(1-benzylpiperidin-4-yl)amino]-N-methylpyrrolidine-2-carboxamide
N,1-dimethyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
2-oxo-N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-1H,2H,5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
3-{1-[(5-chlorofuran-2-yl)methyl]piperidin-4-yl}-N-(3-methoxyphenyl)propanamide
N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-4,6-dihydroxypyridine-3-carboxamide
(2S,4R)-4-amino-N-ethyl-1-(5-methylpyridine-3-carbonyl)pyrrolidine-2-carboxamide
ethyl (4aS,8aR)-6-(5-chloro-6-oxo-1,6-dihydropyridine-3-carbonyl)-decahydro-1,6-naphthyridine-4a-carboxylate
2-(5-{1-[(3E)-4-phenylbut-3-enoyl]piperidin-4-yl}-1H-pyrazol-3-yl)acetic acid
1,3-dimethyl-6-{3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
ethyl 2-(1-{2-[3-(3-fluorophenyl)-1-methyl-2,5-dioxopyrrolidin-3-yl]acetyl}piperidin-2-yl)acetate
1-(furan-3-carbonyl)-4-(4-methoxyphenoxy)piperidine
(4aS,7aR)-1-{5-[(diethylamino)methyl]-2-methylfuran-3-carbonyl}-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-methyl-2-(4-{1H-pyrazolo[3,4-b]pyridin-1-yl}phenyl)pyrimidine
1-{4-[2-(2H-1,3-benzodioxol-5-yl)-5-fluoro-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}-2-(2-methylphenyl)ethan-1-one
N-(2-fluoro-4-methylphenyl)-2-{2-[5-(oxan-2-yl)furan-2-yl]-1H-imidazol-1-yl}acetamide
2-amino-7-[3-(4-methoxyphenyl)propanoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-(carbamoylmethyl)-N-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}piperidine-4-carboxamide
({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)[(5-methyl-1,2,4-oxadiazol-3-yl)methyl](oxolan-2-ylmethyl)amine