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[(1-benzyl-1H-imidazol-2-yl)methyl](benzylsulfamoyl)methylamine
5-{[2-(4-fluorophenyl)morpholin-4-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
N4-ethyl-N2-(furan-3-ylmethyl)-N2,N4-dimethylpyrimidine-2,4-diamine
N4-[1-(3-methylpyridin-2-yl)propan-2-yl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
6-methoxy-2-({2-[2-(pyrrolidin-1-yl)pyrimidin-5-yl]-1H-imidazol-1-yl}methyl)-1H-1,3-benzodiazole
3-[2-(benzenesulfonyl)ethyl]-4,5-dimethyl-2,3-dihydro-1,3-oxazol-2-one
1-{4-methyl-2-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonan-3-yl]pyrimidin-5-yl}ethan-1-one
8-methoxy-5-[2-(morpholin-4-ylmethyl)phenyl]quinoline
1-methyl-N-(morpholin-2-ylmethyl)-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
8-[3-oxo-3-(pyrrolidin-1-yl)propyl]-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-{1-[1-(furan-2-ylmethyl)piperidine-3-amido]cyclohexyl}acetic acid
{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)(oxan-2-ylmethyl)amine
1-benzyl-8-(1H-indol-3-ylmethyl)-3-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3aS,6aS)-2-methyl-5-{[5-(3-methyl-1,2-oxazol-5-yl)furan-2-yl]sulfonyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-N-(3-methoxypropyl)-5-methyl-1H-pyrazole-4-carboxamide
(2S)-1-{9-oxo-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraene-10-carbonyl}pyrrolidine-2-carboxylic acid
2-{5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1H-pyrazole-3-carbonyl}-1,2-oxazinane
4-(4-tert-butylbenzoyl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
4-{3-[2-(morpholin-4-ylmethyl)piperidin-1-yl]propoxy}benzamide
N-[(2S,4R,6R)-2-(2-aminopyrimidin-5-yl)-6-cyclohexyloxan-4-yl]benzamide
(3S,4R)-4-(3-methoxyphenyl)-1-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)pyrrolidine-3-carboxylic acid
4-({[3-hydroxy-1-(4-methylphenyl)propyl]carbamoyl}amino)-N,3-dimethylbenzamide
5-acetyl-N-[1-(3-propyl-1,2,4-oxadiazol-5-yl)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-[methyl(oxan-4-ylmethyl)amino]-2-[2-(methylsulfanyl)phenyl]acetic acid
N-[2-(2-chlorophenoxy)ethyl]-1-methyl-1H-imidazole-2-carboxamide
5-{[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-3-(3-hydroxy-3-methylbutyl)benzamide
3-phenyl-6-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]pyridazine
N-[1-(2-phenylethyl)piperidin-3-yl]-1-(1H-pyrazol-1-ylmethyl)cyclopropane-1-carboxamide
N-{[7-(2-methylbutyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}-2-phenoxyacetamide
2-[2-(ethylcarbamoyl)phenyl]-6-methylpyridine-3-carboxamide
1-(2-methoxyacetyl)-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-3-carboxamide
1-(furan-2-carbonyl)-4-[3-(trifluoromethyl)phenoxy]piperidine
4-{3-[4-(3-methoxyphenyl)piperazine-1-carbonyl]piperidin-1-yl}-2-[1-(thiophen-2-yl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}pyrazolo[1,5-a]pyridine-3-carboxamide
2-methyl-1-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)propan-1-one
3-(5-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl)-5-methyl-1,2-oxazole
4-oxo-N,N-bis(propan-2-yl)-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carboxamide
3-[({1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}oxy)methyl]pyridine
3-(1H-indol-3-yl)-1-{5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}propan-1-one
1-ethyl-3,5-dimethyl-4-({2-[5-(1H-pyrazol-3-yl)furan-2-yl]-1H-imidazol-1-yl}methyl)-1H-pyrazole
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-6-(piperidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
2-methyl-5-{[4-(pyrrolidine-1-carbonyl)-1,3-oxazol-2-yl]methoxy}-1,3-benzothiazole
N-(1,4-dioxan-2-ylmethyl)-5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-methylpyridin-2-amine
(4aS,7aR)-1-(1-ethyl-1H-pyrazole-3-carbonyl)-4-methanesulfonyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-N,4-dimethyl-1,3-thiazol-2-amine
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-1,3-oxazole-4-carboxamide
2-(4-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1H-1,2,3-triazol-1-yl)ethan-1-amine
6-chloro-3-fluoro-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}imidazo[1,2-a]pyridine-2-carboxamide
methyl 2-(4-{6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-3-methyl-2-oxopiperazin-1-yl)acetate