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N-{[7-chloro-2-(2-methoxyphenyl)quinolin-3-yl]methyl}-N-(2-methoxyethyl)-1,3-dimethyl-1H-pyrazole-5-carboxamide
1-[3-(1H-pyrazol-1-yl)benzoyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-(6-fluoro-2-oxo-1,2,3,4-tetrahydroquinolin-8-yl)thiomorpholine-4-carboxamide
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-1-cyclobutanecarbonylpiperidine-4-carboxamide
1-methyl-3-phenyl-8-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-1,8-diazaspiro[4.5]decane
2-[2-(pyridin-4-yl)ethyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-[(2E)-3,7-dimethylocta-2,6-dien-1-yl]-1-propylpiperidin-4-amine
(3S,4R)-1-(1-ethyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid
3-(5-{[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]methyl}thiophen-2-yl)prop-2-yn-1-ol
1-(4-chloro-3-fluorophenyl)-3-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}urea
(2-methoxyethyl)[(4-methylphenyl)methyl]{[3-(1H-pyrazol-1-yl)phenyl]methyl}amine
N-[(3S,7S,8aS)-3-(4-aminobutyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,6-dichlorobenzamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}pyrimidine-4-carboxamide
N-({1-[(2-fluorophenyl)methyl]pyrrolidin-3-yl}methyl)-2-hydroxyacetamide
methyl 4-(5-{[(1,3-benzothiazol-2-ylmethyl)(methyl)amino]methyl}-1,2,4-oxadiazol-3-yl)benzoate
N-(propan-2-yl)-1-(1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)piperidine-4-carboxamide
9-[6-methyl-2-(methylamino)pyrimidin-4-yl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[3-(1H-imidazol-1-yl)propyl]-2-(3-methyl-5-oxo-1-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl)acetamide
1-(2,3-dihydro-1H-inden-4-yl)-3-(2-methoxyethyl)-5-(2H-1,2,3-triazol-2-ylmethyl)-1H-1,2,4-triazole
2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]acetamide
2-cyclopropyl-4-methyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}pyrimidine-5-carboxamide
1-tert-butyl-N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-5-oxopyrrolidine-3-carboxamide
(1R,5R)-6-(cyclopropylmethyl)-3-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
N-cyclopropyl-N-[(3-methylthiophen-2-yl)methyl]quinoline-3-carboxamide
3-[(dimethylamino)methyl]-1-{[2-(3-methoxyphenyl)-1,3-thiazol-5-yl]methyl}pyrrolidin-3-ol
N-(2,1,3-benzoxadiazol-4-ylmethyl)-1-[(3-methoxyphenyl)methyl]piperidin-3-amine
1-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(methylsulfanyl)ethan-1-one
4-(3-hydroxybenzoyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
{[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)[(5-phenyl-1H-pyrazol-3-yl)methyl]amine
2-(pyridin-2-ylmethyl)-8-(4,4,4-trifluorobutyl)-2,8-diazaspiro[5.5]undecan-3-one
6-{[4-(azetidine-1-carbonyl)-1,3-oxazol-2-yl]methoxy}quinoline
7-(1-benzothiophen-3-yl)-4-(2,2-difluorocyclopropanecarbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-(furan-3-ylmethyl)-5-[1-(5-methyl-1,3-oxazole-4-carbonyl)pyrrolidin-2-yl]thiophene-2-carboxamide
(2R)-N-methyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}oxolane-2-carboxamide
N-{[2-(dimethylamino)-7-methoxyquinolin-3-yl]methyl}-3-methoxy-N-(2-methoxyethyl)benzamide
4-({methyl[(1-methyl-5-oxopyrrolidin-3-yl)methyl]amino}methyl)benzonitrile
6-methyl-2-{6-oxo-7-propyl-2,7-diazaspiro[4.5]decan-2-yl}pyridine-3-carbonitrile
6-[1-(1-benzothiophen-2-ylmethyl)piperidin-4-yl]-2-methylpyrimidin-4-ol
5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-(pyrazin-2-ylmethyl)pyridin-2-amine
4-(1-methyl-1H-imidazol-2-yl)-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidine
1-[4-(adamantan-1-yl)piperazin-1-yl]-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
(1S,5R)-6-(2,4-dimethylpyrimidine-5-carbonyl)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
4-{5-[2-(cyclopentyloxy)phenyl]-1H,4H-pyrazolo[3,4-d]imidazol-1-yl}-1-methylpiperidine
1-{[5,8-dimethoxy-2-(2-methoxyphenyl)quinolin-3-yl]methyl}azetidin-3-ol
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2,2-diphenylacetamide
4-(4-chlorophenyl)-N-methyl-N-[1-(pyrimidin-4-yl)ethyl]butanamide
1-(pyridin-4-yl)-4-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperazine
2-[(1-ethylpyrrolidin-2-yl)methyl]-2-azatricyclo[6.3.1.04,12]dodeca-1(12),4,6,8,10-pentaen-3-one
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-5-(propan-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
(2S,4R)-N-ethyl-4-{4-[4-(morpholin-4-ylmethyl)phenyl]-1H-1,2,3-triazol-1-yl}pyrrolidine-2-carboxamide