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1-(3-chlorophenyl)-4-[(3-{2-[1-(pyridine-3-carbonyl)piperidin-2-yl]ethoxy}phenyl)methyl]piperazine
5-benzyl-4-(furan-2-ylmethyl)-1-(3-methoxyphenyl)piperazin-2-one
2-(5-methyl-3-oxo-2,3-dihydro-1H-pyrazol-4-yl)-N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)acetamide
1-methyl-1'-[3-(6-oxo-1,6-dihydropyridazin-3-yl)propanoyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
6-({1-[(2-chlorophenyl)methyl]-5-oxopyrrolidin-3-yl}amino)pyridine-2-carbonitrile
2-methyl-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-3-oxo-2H,3H,5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide
2-({3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}methyl)phenol
3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-[2-(methylsulfanyl)benzoyl]piperidine
(3S,5R)-1-benzyl-N3-cyclopropyl-N5-(2,3-dihydro-1H-inden-5-yl)piperidine-3,5-dicarboxamide
1-(4-{[2-(2-chlorophenoxy)ethyl]amino}piperidin-1-yl)-2-methylpropan-1-one
2-(phenylamino)-1-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}butan-1-one
3-(4-fluorophenoxymethyl)-1-(1-propyl-1H-pyrazole-5-carbonyl)piperidine
N-[(1S,2R)-2-aminocyclobutyl]-2-(1,1,2,2-tetrafluoroethoxy)benzamide
4,6-dimethyl-1-{2-oxo-2-[(1S,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethyl}-1,2-dihydropyrimidin-2-one
4-phenyl-1-(1,3-thiazol-4-ylmethyl)pyrrolidin-2-one
N-[2-(2-methylpropanesulfonyl)ethyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
2-({2-cyclopropyl-5-oxo-5H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl}methyl)-5-(dimethylamino)-2,3-dihydropyridazin-3-one
1-[2-(4-fluorophenyl)ethyl]-4-({[4-(1H-pyrazol-1-yl)phenyl]methyl}amino)pyrrolidin-2-one
3-(azepane-1-carbonyl)-1-ethyl-5-[4-(propan-2-yl)piperazin-1-yl]-4,5,6,7-tetrahydro-1H-indazole
methyl N-{2-[3-(4-fluorophenoxymethyl)piperidin-1-yl]-2-oxoethyl}carbamate
8-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
2-(1-{[2-fluoro-5-(trifluoromethyl)phenyl]methyl}pyrrolidin-2-yl)pyridine
4-benzyl-3-[1-(6-methylpyridazin-3-yl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
3-cyclopropaneamido-N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)propyl]-4-methylbenzamide
N-methyl-N-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}-2-(2,3,6-trimethylphenoxy)acetamide
2-chloro-N-[2-({4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl}amino)ethyl]benzamide
1-{3-[2-(3-fluorophenyl)piperidine-1-carbonyl]phenyl}pyrrolidin-2-one
2-[2-(2-chlorophenyl)phenoxy]propanamide
1-methyl-N-[1-(3-methylphenyl)piperidin-4-yl]azepane-2-carboxamide
N,N-diethyl-3-{[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]sulfamoyl}benzamide
N-[4-(1H-indol-2-yl)phenyl]-1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidine-4-carboxamide
(3aR,6aR)-2-(2-methoxyethyl)-5-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1'-(isoquinoline-1-carbonyl)-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(5-propyl-1,2,4-oxadiazol-3-yl)piperidine
N-(3-methoxyphenyl)-3-{[methyl(propan-2-yl)amino]methyl}benzamide
4-(3-fluoropyridin-4-yl)-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
5-{1-ethyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-2-methoxypyridine
1,3-dimethyl-6-[4-(pyridin-3-ylmethyl)piperazine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}(ethyl)[2-(1H-pyrazol-1-yl)ethyl]amine
N-(2-methoxyethyl)-N-(pyridin-3-ylmethyl)-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
3-{4-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-6-hydroxy-1,4-diazepan-1-yl}pyrazine-2-carbonitrile
4-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridin-2-amine
2,6-difluoro-3-methoxy-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]benzamide
3-{2-[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]-2-oxoethyl}-3,4-dihydroquinazolin-4-one
1-{3-[(4-methoxypiperidin-1-yl)methyl]-7-methylimidazo[1,2-a]pyridine-2-carbonyl}azepane
4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-(propane-1-sulfonyl)piperidine
4-{4-[(3-methylphenyl)methyl]piperazin-1-yl}-2-(oxolan-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
ethyl 4-[3-({[2-(4-chlorophenyl)ethyl]amino}methyl)-6-methylquinolin-2-yl]piperazine-1-carboxylate
5-{3-[2-(pyridin-4-yl)pyridin-4-yl]pyrrolidine-1-carbonyl}pyridin-2-amine
benzyl(methyl)[(3-{octahydro-1H-pyrido[1,2-a]piperazine-2-carbonyl}-1,2-oxazol-5-yl)methyl]amine