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1-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-(3-methylphenyl)piperidine
1-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-4-ethyl-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]-3-(piperazine-1-sulfonyl)benzamide
methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl](3-phenylpropyl)amine
1-({4-[3-(azepan-1-yl)-2-hydroxypropoxy]-3-methoxyphenyl}methyl)piperidine-4-carbonitrile
2-[1-(3,5-dimethylbenzoyl)pyrrolidin-3-yl]benzoic acid
3-(2-{2-[4-chloro-2-(dimethylamino)-1,3-thiazol-5-yl]-1H-imidazol-1-yl}ethyl)-1,3-oxazolidin-2-one
N-[(2R)-1-oxo-1-[3-oxo-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-9-yl]butan-2-yl]acetamide
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-1-[2-(pyridin-2-yl)piperidin-1-yl]propan-1-one
4-{[5-(2,3-dihydro-1,4-benzodioxin-2-yl)-1-methyl-1H-1,2,4-triazol-3-yl]methyl}-1-methylpiperidine
2-chloro-N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-5-acetamidobenzamide
N-(5-cyanopyridin-2-yl)-3-{[methyl(oxan-2-ylmethyl)amino]methyl}benzamide
2-(dimethylamino)-2-(4-fluorophenyl)-1-[4-(thiomorpholin-4-yl)piperidin-1-yl]ethan-1-one
7-cyclopentanecarbonyl-N,N-dimethyl-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
8-(butan-2-yl)-1-(3-methylbutyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl 3-[ethyl({[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl})carbamoyl]benzoate
N-[(3S)-1-benzylpyrrolidin-3-yl]-3-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]propanamide
1-ethyl-N,3,5-trimethyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1H-pyrazole-4-carboxamide
(1R,3S)-7-(5-ethyl-1,3-oxazole-4-carbonyl)-3-methoxy-3-methyl-7-azaspiro[3.5]nonan-1-ol
N-(7-methoxy-2,2-dimethyl-3,4-dihydro-2H-1-benzopyran-4-yl)-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
2-(4-{[(3R)-3-hydroxypyrrolidin-1-yl]methyl}phenyl)-6-(4-methoxyphenyl)-3,4-dihydropyrimidin-4-one
2-methyl-4-(5-{[4-(pyridin-4-yl)piperidin-1-yl]methyl}thiophen-2-yl)but-3-yn-2-ol
methyl[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl][1-(pyridin-3-yl)ethyl]amine
(4aS,7aS)-6-(2-methyl-1-benzofuran-5-carbonyl)-octahydro-1H-pyrrolo[3,4-b]pyridine
{5-[3,5-difluoro-4-(pyrrolidin-1-ylmethyl)phenoxy]-2,3-dihydro-1-benzofuran-2-yl}methanamine
3-{2-[3-(dimethylamino)pyrrolidin-1-yl]ethyl}-8-(3-hydroxybenzoyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(4S)-4-phenyl-3-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-1,3-oxazolidin-2-one
1-[(1R,5R)-6-[(2-methoxy-4-methylphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
(3S,9aR)-3-(4-aminobutyl)-8-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-[4-({4-[(2-fluoro-4-methoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenyl]but-3-yn-1-ol
5-[(4-chloro-1-methyl-1H-pyrazol-3-yl)methyl]-N-phenyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
8-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
4-(cyclohex-3-ene-1-carbonyl)-1-[(4-methoxyphenyl)methyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
1-[4-(2,2-dimethylpent-4-en-1-yl)-1-methyl-1,4,9-triazaspiro[5.5]undecan-9-yl]-2-methoxyethan-1-one
N-ethyl-6-hydroxy-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2,5,7,8-tetramethyl-3,4-dihydro-2H-1-benzopyran-2-carboxamide
3-{5-[(4-phenylphenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-[1-(thiophen-2-yl)ethyl]propanamide
4-(5-hydroxypyridine-2-carbonyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-(3-{1-[(5-fluoro-2-methylphenyl)methyl]-1H-pyrazol-3-yl}phenyl)pyrimidine
(4aR,7aS)-1-(cyclopropylmethyl)-4-(3-hydroxy-2-methylbenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(2-methylphenyl)-4-(oxolan-3-ylmethyl)-1,4-diazepane
2-ethyl-9-(3-methoxypropanoyl)-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
(4-benzyl-1-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl)methanol
4-{[1-(4-chlorophenyl)cyclobutyl]methyl}-1λ6-thiomorpholine-1,1-dione
1-{1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]piperidin-4-yl}-3-(pyrrolidine-1-carbonyl)piperidine
2-(dimethyl-1,3-thiazol-5-yl)-1-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]ethan-1-one
1-ethyl-N-(furan-2-ylmethyl)-5-methyl-N-(pyridin-2-ylmethyl)-1H-pyrazole-4-carboxamide
[(2-methoxyphenyl)methyl](methyl)[(5-{[(2-methylphenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)methyl]amine
{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}(methyl)[(7-methyl-1H-1,3-benzodiazol-2-yl)methyl]amine
(1-{1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-3-propylpiperidin-3-yl)methanol
4-(3-methoxyphenyl)-2-[5-methyl-4-(4-propylpiperazine-1-carbonyl)-1H-pyrazol-1-yl]pyrimidine