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N-[1-(2-{4-[(2-methylphenyl)sulfanyl]piperidin-1-yl}-2-oxoethyl)-1H-pyrazol-4-yl]-3-phenoxypropanamide
N-{[3-(methylsulfanyl)phenyl]methyl}-1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
4-{4-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrol-2-yl]piperidin-1-yl}-N,N,6-trimethylpyrimidin-2-amine
2-[(3,4-difluorophenyl)methyl]-8-(pyrazin-2-yl)-2,8-diazaspiro[4.5]decan-3-one
1-[6-hydroxy-4-(3-methylbut-2-en-1-yl)-1,4-diazepan-1-yl]-2-[4-(hydroxymethyl)phenyl]ethan-1-one
N-(1-benzothiophen-5-ylmethyl)-1,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-(1-cycloheptylpiperidin-3-yl)-4-oxo-4-phenylbutanamide
3-({4-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]piperazin-1-yl}methyl)benzonitrile
1-[(4-methylphenyl)methyl]-4-{4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carbonyl}piperazin-2-one
1-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-yl]-2-phenoxyethan-1-one
2-{1-[1-(4-tert-butylcyclohexanecarbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-2-amine
2-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-N-(2-phenylethyl)acetamide
2-methyl-8-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-cyclopropyl-4-[4-hydroxy-4-(pyridin-3-yl)piperidine-1-carbonyl]pyrrolidin-2-one
(3R,4R)-3-cyclopropyl-4-methyl-1-(pyrrolidine-1-sulfonyl)pyrrolidin-3-ol
1-(4-chlorophenyl)-N-(2-{4-methyl-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)cyclopropane-1-carboxamide
1-ethyl-3-[2-(oxolan-2-ylmethoxy)phenyl]-1-(pyridin-4-ylmethyl)urea
N-[(2-chlorophenyl)methyl]-3-[1-(2-methyl-1H-pyrrole-3-carbonyl)piperidin-3-yl]propanamide
7-[(2S)-2-amino-3-methoxypropanoyl]-2,3-dimethyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
N-[3-(diethylamino)propyl]-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
3-{3-[methyl(2-methylpropyl)amino]propyl}-8-(1-methylcyclopropanecarbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-{1-[4-(1H-pyrazol-3-yl)benzoyl]piperidin-3-yl}-1H-1,3-benzodiazole
N-{5H,6H,7H-cyclopenta[b]pyridin-7-yl}-1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-{4-[1-(furan-2-ylmethyl)piperidine-3-carbonyl]piperazin-1-yl}pyridine-3-carbonitrile
(3aR,6aR)-2-(2-methoxyethyl)-5-{[5-(2-methylpropyl)thiophen-2-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(2-ethoxyethyl)-N,3-dimethyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1H-pyrazole-5-carboxamide
1-[cyclopropyl(4-methylpyridin-2-yl)methyl]-3-(4,5-dimethyl-1H-1,3-benzodiazol-6-yl)urea
N-[2-(3-ethylphenoxy)ethyl]-N-methyl-2-oxo-1-oxaspiro[4.5]decane-4-carboxamide
1-[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-(methylsulfanyl)propan-1-one
N-benzyl-N-methylpiperidin-3-amine
(5S,9aS,9bS)-5-(4-ethylphenyl)-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
5-{1-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]piperidin-4-yl}-5-(pyridin-3-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
4-methoxy-3-[3-methyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]benzene-1-sulfonamide
5-(3-phenylpropyl)-5-(piperidin-4-yl)-3-[2-(pyridin-2-yl)ethyl]imidazolidine-2,4-dione
4-[3-cyclopropyl-1-(2-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]-2,6-dimethoxypyrimidine
{1-[(4,6-dimethylpyrimidin-2-yl)methyl]-3-(2-methoxyethyl)piperidin-3-yl}methanol
6-[(8-fluoro-4-hydroxyquinolin-2-yl)methyl]-1-methyl-1H,4H,5H,6H,7H-pyrrolo[2,3-c]pyridine-2-carboxamide
2-[4-(2,5-difluorophenyl)-1H-pyrazol-1-yl]-N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]acetamide
3-phenyl-N-{1-[1-(pyridine-3-sulfonyl)piperidin-4-yl]-1H-pyrazol-5-yl}propanamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-5-methanesulfonyl-N,2-dimethylpyrimidin-4-amine
4-{[(2-hydroxyethyl)({[4-(methylsulfanyl)phenyl]methyl})amino]methyl}-N-methylbenzene-1-sulfonamide
5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-[1-(pyrazin-2-yl)propan-2-yl]pyridin-2-amine
N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-1-methyl-6-oxo-1,6-dihydropyridazine-3-carboxamide
2-amino-N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-4-methyl-1,3-benzothiazole-6-carboxamide
5-tert-butyl-3-{[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1H-pyrazole
{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
7,7-dimethyl-2-[2-(4-methylpiperidin-1-yl)ethyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-(3-cyano-4-methoxyphenyl)-1-{[1-(morpholin-4-yl)cycloheptyl]methyl}urea
8-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-1-oxa-8-azaspiro[4.6]undecan-9-one