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2-(3-chloro-2,6-difluorophenyl)-1-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]ethan-1-one
methyl 4-[4-(pyrrolidin-3-ylmethyl)piperazin-1-yl]benzoate
8-{1-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}quinoline
3-amino-N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-2-methylpropanamide
1-({6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperidin-4-ol
4-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}-5-methyl-1-(2-methylphenyl)piperazin-2-one
1-(thiophen-2-ylmethyl)-4-[4-(1H-1,2,4-triazol-3-yl)benzoyl]-1,4-diazepane
1-(4-{[4-(2-methoxyphenyl)piperidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
1-(2-{3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}-2-oxoethyl)pyrrolidin-2-one
1-{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}-4-[(4-fluorophenyl)methyl]-1,4-diazepan-5-one
1-(adamantan-1-yl)-4-{pyrazolo[1,5-a]pyridine-7-carbonyl}piperazine
[(2S,4R)-1-{3-azaspiro[5.5]undecan-9-yl}-4-(dimethylamino)pyrrolidin-2-yl]methanol
N-[(4-methoxynaphthalen-1-yl)methyl]-N-(propan-2-yl)-2-(1,2,3,6-tetrahydropyridin-4-yl)acetamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[1-(1,3-thiazole-4-carbonyl)piperidin-3-yl]piperazine
1-{3-[(methylsulfanyl)methyl]piperidin-1-yl}-4-(1H-pyrazol-4-yl)butan-1-one
ethyl 4-(1-cycloheptyl-1H-1,2,3-triazole-4-carbonyl)piperazine-1-carboxylate
ethyl 1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-3-(3-phenylpropyl)piperidine-3-carboxylate
N-[(5-chloro-2-ethoxyphenyl)methyl]-3-(2,5-dioxoimidazolidin-4-yl)-N-methylpropanamide
ethyl 2-[4-({[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]carbamoyl}amino)phenyl]acetate
N-[2-(2-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
4-methyl-3-(pyridin-3-yl)-1H-indazole
2-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-6-methylpyridine-3-carboxylic acid
4-(2-amino-4-phenylpyrimidine-5-carbonyl)-3-methyl-1-(2-methylpropyl)piperazin-2-one
9-(but-3-yn-1-yloxy)-4-(3,5-dimethoxybenzoyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-(morpholin-4-yl)propanamide
(2S)-2-(hydroxymethyl)-N-[4-(3-methylphenyl)phenyl]pyrrolidine-1-carboxamide
(4aS,8aR)-6-methanesulfonyl-1-[2-(5-methylfuran-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
N-(cyclohex-1-en-1-ylmethyl)-8-methyl-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-[2-(pyrazin-2-yl)ethyl]pyridin-2-amine
N,N-dimethyl-6-[3-(propoxymethyl)pyrrolidin-1-yl]pyrimidin-4-amine
4-[({[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}amino)methyl]-1,2-dihydrophthalazin-1-one
2-(2,2-diphenylethyl)-4-(1H-imidazol-4-ylmethyl)morpholine
1-[(4aS,8aS)-4a-hydroxy-7-(pyridin-3-ylmethyl)-decahydro-2,7-naphthyridin-2-yl]-3-methylbut-2-en-1-one
methyl[(3-methyl-1,2-oxazol-5-yl)methyl]({6-methyl-2-[(2-methylphenyl)methoxy]quinolin-3-yl}methyl)amine
1-(2-{[3-(3-chlorophenyl)pyrrolidin-1-yl]methyl}-4-methoxyphenyl)-1H-pyrazole
(2,2-difluoroethyl)({[3-(4-fluorophenyl)oxolan-3-yl]methyl})amine
(3-{5-[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}phenyl)methanol
2-(2H-1,2,3-benzotriazol-2-yl)-N-({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)acetamide
8-[(4-methanesulfonylphenyl)methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-[4-(2-fluorophenoxy)phenyl]-1-(2-methylpropyl)piperidine-4-carboxamide
2-{1-[(4-methylphenyl)methyl]-4-(oxan-4-yl)piperazin-2-yl}ethan-1-ol
7-(9H-fluoren-2-ylmethyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(morpholin-4-yl)benzamide
2-[2-(morpholin-4-ylmethyl)phenyl]pyridin-4-amine
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
ethyl 4-[5-(2-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]piperazine-1-carboxylate
N,4-dimethyl-3-(2-oxoimidazolidin-1-yl)-N-[1-(1,3-thiazol-2-yl)ethyl]benzamide
1-[(2-chloro-4,5-dimethoxyphenyl)methyl]-3-[4-(2,6-difluorophenyl)-1H-pyrazol-5-yl]piperidine
2-(5,5-dimethyl-2,4-dioxo-1,3-oxazolidin-3-yl)-N-methyl-N-{[4-(trifluoromethyl)phenyl]methyl}acetamide