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methyl 3-{[4-(3-{[4-(pyridin-3-ylmethyl)piperazin-1-yl]methyl}phenoxy)piperidin-1-yl]sulfonyl}thiophene-2-carboxylate
4-{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-1-methyl-2-phenylpiperazine
N-[1-(4-methoxyphenyl)-4-(morpholin-4-yl)-1H-indazol-3-yl]-2-(methylsulfanyl)acetamide
3-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridin-2-ol
2-{5-[(2-fluorophenyl)methyl]-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-1-yl}pyridine
(2R)-2-[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyrrolidine
4-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(methylsulfanyl)pyrimidine
1-ethyl-3-methyl-N-[3-(4-methylpiperazin-1-yl)butyl]-1H-pyrazole-4-carboxamide
3-[2-(2-phenylpyrrolidine-1-carbonyl)phenyl]-1H-1,2,4-triazole
3-cyclobutyl-1-[2-(propan-2-ylsulfanyl)phenyl]urea
N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}cyclopropanecarboxamide
4-(4-fluoro-2-methylphenoxy)-1-(pyridin-3-ylmethyl)piperidine-4-carboxylic acid
7-{[4-(pyrrolidine-1-carbonyl)phenyl]methyl}-2-oxa-7-azaspiro[4.5]decan-8-one
5,6-dimethyl-2-oxo-N-[1-(phenylcarbamoyl)piperidin-4-yl]-1,2-dihydropyridine-3-carboxamide
5-(dimethylamino)-2-(3,3,4,4,4-pentafluorobutyl)-2,3-dihydropyridazin-3-one
5-[1-({2-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)pyrrolidin-2-yl]-3-methyl-1H-1,2,4-triazole
2-{4-[(1,3-diphenyl-1H-pyrazol-4-yl)methyl]-1-methylpiperazin-2-yl}ethan-1-ol
N-(2-methylpropyl)-4-{[2-(pyridin-3-yl)ethyl]sulfamoyl}benzamide
4-cyclobutyl-2-[(4-methoxyphenyl)methyl]morpholine
N-[(3-methyl-1,2-oxazol-5-yl)methyl]-3-[(2R)-2-methylpiperazine-1-carbonyl]benzene-1-sulfonamide
N-benzyl-3-({[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}methyl)-N-methylpyridin-2-amine
4-[(3S)-3-aminopiperidine-1-carbonyl]-N-(3-methoxypropyl)benzene-1-sulfonamide
dimethyl({3-[2-(1-{6-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-3-yl)-1H-imidazol-1-yl]propyl})amine
4-{[(2-methanesulfonylethyl)carbamoyl]amino}-N-(2-methoxyethyl)benzamide
N-{3-[4-(morpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]propyl}-1-phenylcyclohexane-1-carboxamide
2-(2,3-dihydro-1H-inden-5-yloxy)-2-methyl-N-[(1-methylpiperidin-4-yl)methyl]propanamide
3-(1H-imidazol-1-ylmethyl)-1-[(4-methanesulfonylphenyl)methyl]piperidine
N-[(1-benzylpyrrolidin-3-yl)methyl]-1-[(4-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
4-(3-methyl-1H-pyrazol-5-yl)-6-(4-methylpiperazin-1-yl)pyrimidin-2-amine
5-({4-[(3-fluorophenyl)methyl]piperazin-1-yl}methyl)-2-phenylpyrimidine
N-(1-{1-[(2-fluoro-5-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)oxolane-3-carboxamide
8-(1,3-thiazol-4-ylmethyl)-1,3-dioxa-8-azaspiro[4.5]decan-2-one
2-(adamantan-1-yl)-N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}acetamide
2-(quinolin-4-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-{3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}-3-(1-methyl-1H-imidazol-2-yl)piperidine
5-(4-acetyl-2-methoxyphenoxymethyl)-N-ethyl-N-[2-(1H-pyrazol-1-yl)ethyl]-1,2-oxazole-3-carboxamide
1-(azepan-1-yl)-4-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}butane-1,4-dione
4-(3-methylthiophen-2-yl)-1-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]-1H-1,2,3-triazole
(3aR,6aR)-N-[(5-ethylpyridin-2-yl)methyl]-2-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
(2S,4R)-N,N-diethyl-1-methyl-4-(thiophene-3-amido)pyrrolidine-2-carboxamide
1-(4-fluorophenyl)-4-[1-(1-phenylcyclopropanecarbonyl)piperidin-3-yl]piperazine
5-methyl-2-[2-methyl-1-(4H-1,2,4-triazol-4-yl)propyl]-1H-1,3-benzodiazole
6-{4-[1-(2,2-dimethylpropyl)pyrrolidin-3-yl]piperidin-1-yl}-9H-purine
1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethan-1-amine
4-(4-methanesulfonyl-1,4-diazepane-1-carbonyl)-1,2-dihydroisoquinolin-1-one
N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
1-ethyl-3-methyl-N-{2-[(3-methylpyridin-4-yl)amino]ethyl}piperidine-3-carboxamide
1-{3-[9-methoxy-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]phenyl}imidazolidin-2-one
2-[3-(1H-pyrazol-3-yl)phenyl]benzonitrile
7-cyclobutaneamido-1-methyl-2-(pyridin-4-yl)-N-{spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-5-ylmethyl}-1H-1,3-benzodiazole-5-carboxamide