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methyl (2S,4S)-4-(3-chlorobenzamido)-1-(quinolin-4-ylmethyl)pyrrolidine-2-carboxylate
(2S,4R)-1-[(4-chlorophenyl)methyl]-4-[(2,3-dihydro-1H-inden-2-yl)amino]-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(5-chloropyridin-2-yl)piperazine
N-methyl-N-[1-(pyridin-2-yl)ethyl]-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
N-({5-[4-(methylamino)-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-[4-(4-methoxybenzoyl)piperazin-1-yl]ethan-1-one
5-[(6-ethoxy-2,3-dihydro-1H-inden-5-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
2-(dimethylamino)-2-(4-fluorophenyl)-N-(isoquinolin-5-ylmethyl)-N-methylacetamide
2-(adamantan-1-yl)-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]acetamide
6-[(diethylamino)methyl]-N-(furan-3-ylmethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-N,N-dimethylpyrrolidin-3-amine
2-{2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl}-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
4-(2-methoxyphenoxy)-1-[(5-methylfuran-2-yl)methyl]piperidine-4-carboxylic acid
1-(3-hydroxyphenyl)-4-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]pyrrolidin-2-one
N-(4-ethoxyphenyl)-3-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-yl}-3-oxopropanamide
2-(2H-1,2,3-benzotriazol-2-yl)-1-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]ethan-1-one
benzyl (3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidine-1-carboxylate
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-(2-methoxy-4-methylphenoxymethyl)-1,3-oxazole-4-carboxamide
1-[(2-chloro-6-fluoro-3-methoxyphenyl)methyl]-4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)piperidine
4-(3-fluorophenyl)-N-{[4-(2-methylpropyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}benzamide
(2S,4S)-N-ethyl-4-{[(4-fluorophenyl)methyl]amino}-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
N-ethyl-2-[4-(1H-pyrazol-1-yl)phenyl]benzamide
1-(2-methoxyphenyl)-4-(3-phenyl-1H-pyrazole-4-carbonyl)piperazin-2-one
1-[1-(2-fluorophenyl)cyclopropanecarbonyl]-2-(3-methoxypropyl)piperidine
2-[2-(piperidin-1-ylmethyl)phenoxy]pyridine-4-carbonitrile
(3aS,6aR)-3-[2-(3-chlorophenyl)ethyl]-5-(prop-2-ene-1-sulfonyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
3-[2-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)ethyl]pyridine
2-{4-[(2-chloro-3,4-dimethoxyphenyl)methyl]-1-cyclopentylpiperazin-2-yl}ethan-1-ol
3-methyl-8-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[3-(1H-imidazol-1-yl)propyl]-1,9-dioxaspiro[5.5]undecan-4-amine
3-(4-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)-1,2-dihydropyrazin-2-one
5-methyl-1-(3-{3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}phenyl)-1H-1,2,3,4-tetrazole
N,1-dimethyl-3-(propan-2-yl)-N-[1-(pyrimidin-4-yl)ethyl]-1H-pyrazole-5-carboxamide
N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]-2-(2-phenyl-1,3-thiazol-4-yl)acetamide
1-[(dimethyl-1,3-thiazol-2-yl)methyl]-3-(3-phenyl-1,2,4-thiadiazol-5-yl)urea
7-[1-(furan-2-carbonyl)piperidin-4-yl]-2-oxa-7-azaspiro[4.5]decan-8-one
1-(2H-1,3-benzodioxol-5-yl)-3-cyclopropyl-5-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1H-1,2,4-triazole
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(methylsulfanyl)propyl]acetamide
N,N-dimethyl-2-[2-({[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]carbamoyl}amino)phenyl]acetamide
4-{4-[(4-fluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}-2-methoxypyridine-3-carbonitrile
N-[(2-fluorophenyl)methyl]-2-{[2-(4-hydroxy-3-methoxyphenyl)ethyl]amino}acetamide
1-(1,3-thiazole-4-carbonyl)-4-{[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]methyl}piperidine
N-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-3-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide
N-{[1-(furan-2-ylmethyl)pyrrolidin-3-yl]methyl}-7-methylpyrazolo[1,5-a]pyrimidine-6-carboxamide
3-(1-{[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}piperidin-3-yl)-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
3-amino-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}propanamide
9-[2-(propan-2-yloxy)propanoyl]-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
4-[2-(2,3-dihydro-1-benzofuran-7-yl)pyridine-4-carbonyl]morpholine
ethyl 5-({methyl[1-(1,2-oxazol-3-yl)ethyl]amino}methyl)-1-(4-phenyl-1,3-thiazol-2-yl)-1H-pyrazole-4-carboxylate
(3R,5R)-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide