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8-(5-hydroxy-1,2-dimethyl-1H-indole-3-carbonyl)-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
3,4-dimethoxy-2-({4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}methyl)pyridine
4-(benzyloxy)-1-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}piperidine
1-(piperazin-1-yl)-2-[(1R,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
methyl 3-(cyclobutylmethoxy)-5-[4-(methylamino)piperidine-1-carbonyl]benzoate
N-[1-({[(3-methoxyphenyl)methyl]carbamoyl}methyl)-1H-pyrazol-4-yl]-3-phenoxypropanamide
N-[(5-chloro-2-ethoxyphenyl)methyl]-N,1-dimethylazepane-2-carboxamide
7-methoxy-N,N-dimethyl-2-[2-(pyridin-2-yl)pyrimidin-5-yl]quinoline-4-carboxamide
3-{1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
3-{1-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1-(pyrrolidin-1-yl)propan-1-one
ethyl 4-{3-[(thiophen-2-ylformamido)methyl]piperidin-1-yl}piperidine-1-carboxylate
[(2E)-2-methyl-3-phenylprop-2-en-1-yl]({3-[4-(morpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]propyl})amine
9-(3-methoxy-4-methylbenzoyl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-5-methyl-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
3-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]azepan-2-one
methyl 5-[(2,2-dimethylpropyl)amino]-3-(oxolane-2-amido)-1-(2-phenylethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-3,5-bis(trifluoromethyl)benzamide
N-ethyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
N-[(5-methoxy-1,3-benzoxazol-2-yl)methyl]-2,3-dimethylquinoxaline-6-carboxamide
N-(2-{[3-(pyridin-4-yl)-1H-pyrazol-5-yl]formamido}ethyl)pyridine-3-carboxamide
4-[(dipropylamino)methyl]-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]benzamide
(1S,5R)-6-[4-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)benzoyl]-3-methyl-3,6-diazabicyclo[3.2.2]nonane
N-[(4-methyl-1H-imidazol-2-yl)methyl]-2-(methylsulfanyl)benzamide
2-(butan-2-ylsulfanyl)-5-{[4-(1,2,4-oxadiazol-3-yl)piperidin-1-yl]methyl}pyrimidine
2-{5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
[(2S,6S)-4-(1-ethylpiperidin-4-yl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
1-[2-(3,3-dimethylbutanamido)ethyl]-N-(3-methoxyphenyl)-1H-1,2,3-triazole-4-carboxamide
2-{1-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]piperidin-3-yl}-1H-1,3-benzodiazole
1-methyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-1H-pyrazole-4-sulfonamide
(3S,4R)-1-(morpholine-4-carbonyl)-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
9-ethyl-1-methyl-4-{[5-(pyridin-3-yl)-1,3,4-oxadiazol-2-yl]methyl}-1,4,9-triazaspiro[5.6]dodecan-10-one
1-(4-methyl-2-{[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]amino}pyrimidin-5-yl)ethan-1-one
3-[(2R,3R,6R)-5-(dimethyl-1,2-oxazole-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
3-(2-ethyl-5-oxopyrrolidin-2-yl)-N-[(4-phenyloxan-4-yl)methyl]propanamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)piperidin-3-ol
N-[2-(2,5-dimethylphenoxy)ethyl]-N-methylquinoxaline-5-carboxamide
1-[1-(thiophene-2-carbonyl)piperidin-3-yl]-4-[3-(trifluoromethyl)phenyl]piperazine
N,3-dimethyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-1-propyl-1H-pyrazole-4-carboxamide
(2R)-2-[({4-[1-(dimethylamino)ethyl]phenyl}methyl)amino]propanamide
[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl][1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amine
1-(2H-1,3-benzodioxole-5-carbonyl)-4-{[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine
1-{2,7-dimethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-4-(3-methylpyridin-4-yl)piperazine
1-(4-{4-cyclopropyl-5-[(dimethylamino)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-3-(ethylsulfanyl)propan-1-one
2-(2,5-dioxoimidazolidin-4-yl)-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]acetamide
2-{ethyl[3-(morpholin-4-yl)propyl]amino}-2-[4-(propan-2-yloxy)phenyl]acetic acid
4-(cyclopropylmethyl)-1-[2-(2,3,6-trifluorophenyl)acetyl]-1,4-diazepan-5-one
[3-(2-fluoro-4-methoxybenzoyl)-9-propyl-3,9-diazaspiro[5.5]undecan-1-yl]methanol
2-benzyl-9-[(2-ethyl-1,3-thiazol-4-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[(3R,4S)-4-cyclopropyl-1-{[4-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl]-2-hydroxyacetamide
N-{[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl}-N-[(trimethyl-1H-pyrazol-4-yl)methyl]cyclopropanamine