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1-[(2E)-3-(2-chlorophenyl)prop-2-enoyl]-4-[2-(pyrrolidin-1-yl)ethyl]-1,4-diazepan-5-one
(1R,3S)-3-(2-aminoethoxy)-7-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)-7-azaspiro[3.5]nonan-1-ol
1-{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-(methoxymethyl)-1H-1,2,4-triazole
1-(1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-1H-pyrazole-4-carbonyl)-4-(propan-2-yl)piperazine
2-(2-ethyl-1H-1,3-benzodiazol-1-yl)-N-{imidazo[1,2-a]pyridin-2-ylmethyl}butanamide
6-fluoro-2-oxo-N-[1-(pyrazin-2-yl)piperidin-4-yl]-1,2,3,4-tetrahydroquinoline-4-carboxamide
(2R,3S,6R)-3-(3,5-difluorophenyl)-5-(3-methyl-1H-pyrazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(3aS,6aS)-2-{[4-(carbamoylmethoxy)-3-chlorophenyl]methyl}-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-(2-methoxyquinolin-3-yl)thiophene-2-carboxamide
(4aS,7aR)-1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-ethyl-3-methoxy-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)propanamide
N-(2-methoxyethyl)-3,5,7-trimethyl-N-(pyridin-2-ylmethyl)-1H-indole-2-carboxamide
3-[(3R,4S)-1-[(3-chloro-2,6-difluorophenyl)methyl]-4-(dimethylamino)piperidin-3-yl]propan-1-ol
N-(1H-indol-2-ylmethyl)-5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-amine
1-[({2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]cyclohexan-1-ol
3-{2-oxo-2-[4-(2-phenoxyethyl)piperazin-1-yl]ethyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
N-(4-{[2-(2-methoxyphenyl)-8-methyl-2,3,4,5-tetrahydro-1,5-benzothiazepin-5-yl]methyl}phenyl)acetamide
2-[6-oxo-4-(piperidin-1-yl)-1,6-dihydropyridazin-1-yl]-N-[1-(thiophen-3-yl)propan-2-yl]acetamide
1-{[5-(hydroxymethyl)furan-2-yl]methyl}-4-(naphthalen-2-yloxy)piperidine-4-carboxylic acid
N-(furan-2-ylmethyl)-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)-N-(pyridin-2-ylmethyl)acetamide
5-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1,2-dihydropyridin-2-one
8-[3-(pyridin-4-yl)-1H-pyrazole-5-carbonyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
3-{1-[(5-acetylthiophen-3-yl)methyl]piperidin-3-yl}-N-[(2,4-dimethoxyphenyl)methyl]propanamide
(5S,9aS,9bS)-2-(2,3-dihydro-1H-inden-2-yl)-5-(2-fluoro-4-methoxyphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
(4-{6-chloro-3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}-1,4-oxazepan-6-yl)methanol
2-(cyclohexylmethyl)-4-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)morpholine
(3S,4R)-1-[3-(4-methoxyphenyl)-1H-pyrazole-5-carbonyl]-N,N-dimethyl-4-propylpyrrolidin-3-amine
6-chloro-N-(1-methyl-5-oxopyrrolidin-3-yl)imidazo[1,2-a]pyridine-2-carboxamide
6-methoxy-3-methyl-N-[(6-oxo-1,6-dihydropyrimidin-4-yl)methyl]-1-benzofuran-2-carboxamide
5-{[(5-methyl-1,2-oxazol-3-yl)methyl]amino}-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
(3S)-3-{[2-amino-6-(morpholin-4-yl)pyrimidin-4-yl]amino}azepan-2-one
N-[2-(4,6-dihydroxypyrimidin-2-yl)ethyl]-4-(piperidin-1-yl)butanamide
(4aS,7aR)-1-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-{[methyl(2-methylprop-2-en-1-yl)amino]methyl}-N-(5-methyl-1,3,4-thiadiazol-2-yl)benzamide
N-(3-phenylprop-2-yn-1-yl)-3-(propan-2-yl)-N-propyl-1H-pyrazole-5-carboxamide
2-{4-[2-(2-ethylphenoxy)ethyl]piperazin-1-yl}phenol
3-{3-methyl-4-[2-(methylamino)ethoxy]phenyl}benzoic acid
N-[(4-methoxyphenyl)methyl]-1-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}piperidine-4-carboxamide
2-[3-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]quinoxaline
1-{[1-(4-methoxyphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]methyl}-1,2-dihydropyrimidin-2-one
N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-3-[4-(3-methylphenyl)piperazin-1-yl]propanamide
(4aR,8aR)-4-[(3-chloro-4,5-dimethoxyphenyl)methyl]-octahydro-2H-1,4-benzoxazine
1-{[(2-fluorophenyl)carbamoyl]methyl}-3-(2-methylpropyl)-2-oxo-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
2-[3-(2-fluorophenyl)pyrrolidin-1-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
1'-[(2-phenyl-1,3-oxazol-4-yl)methyl]-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-(2,5-dioxoimidazolidin-1-yl)-N-(pyridin-3-ylmethyl)acetamide
2-(2H-1,3-benzodioxol-5-yloxy)-N-[(2-methylphenyl)methyl]-N-(prop-2-en-1-yl)acetamide
3-(dimethyl-1,2-oxazol-4-yl)-1-[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]urea
N-cyclopropyl-5-(4-phenylazepane-1-carbonyl)pyridin-2-amine
N,7-dimethyl-2-(1-methyl-1H-pyrazol-4-yl)-N-[1-(3-methylpyridin-2-yl)propan-2-yl]quinoline-4-carboxamide