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1-{4-[(1S,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]piperidin-1-yl}ethan-1-one
4-hydroxy-N-[(3R,4R)-4-(piperidin-1-yl)oxolan-3-yl]-2-(pyridin-2-yl)pyrimidine-5-carboxamide
2-{1-[2-(4-fluorophenyl)imidazo[1,2-a]pyridine-6-carbonyl]piperidin-2-yl}ethan-1-ol
[1-(1-{[3-(2-methylphenyl)phenyl]methyl}piperidin-3-yl)piperidin-4-yl]methanol
(3aR,6aS)-5-(2-chlorobenzenesulfonyl)-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(1-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}pyrrolidin-3-yl)acetamide
(3S)-3-benzyl-4-[2-methyl-2-(morpholin-4-ylmethyl)propyl]piperazin-2-one
2-[(5-ethyl-1,3,4-oxadiazol-2-yl)sulfanyl]-1-[1-(4-ethylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]ethan-1-one
1-{1-[4-(2,4-dimethylbenzamido)phenyl]piperidin-4-yl}-N,N-diethylpiperidine-4-carboxamide
3-{3-[3-(pyrimidin-5-yl)phenyl]-1H-pyrazol-1-yl}propan-1-ol
N-(2H-1,3-benzodioxol-5-yl)-3-[methyl(2-phenylethyl)amino]piperidine-1-carboxamide
2-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-1H-pyrrole
{3-ethyl-1-[(3-fluoro-4-methoxyphenyl)methyl]piperidin-3-yl}methanol
1-(2-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-oxoethyl)-1,2-dihydropyridin-2-one
3-(1-methyl-1H-imidazol-2-yl)-1-(3-phenoxybenzoyl)piperidine
ethyl 4-[(3R,4R)-3-hydroxy-4-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidin-1-yl]piperidine-1-carboxylate
4-(1H-imidazol-1-ylmethyl)-1-(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)piperidin-4-ol
2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-{[1-(4-methoxyphenyl)cyclopentyl]methyl}acetamide
N3-ethyl-N5-[(2-fluorophenyl)methyl]-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
3-({[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)amino)propan-1-ol
2-ethyl-1-[(2-methoxyphenyl)methyl]-N,6-dimethyl-4-oxo-N-(thiophen-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
2-amino-3-ethyl-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-3H-imidazo[4,5-b]pyridine-6-carboxamide
N-{3-[(3S,4R)-3-ethyl-4-hydroxy-4-methylpiperidine-1-carbonyl]-2-methylphenyl}furan-2-carboxamide
2-[3-(pyridin-3-yl)azetidin-1-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxylic acid
N-(5-fluoro-2-methylphenyl)-2-[2-(1H-imidazol-1-yl)ethyl]piperidine-1-carboxamide
3-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[2-(4-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-4-hydroxy-2-methylpyrimidine-5-carboxamide
3-(2-hydroxyphenyl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-1H-pyrazole-5-carboxamide
methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)amine
2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-1-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]ethan-1-one
2-[4-(4-chlorophenoxy)piperidine-1-carbonyl]pyridin-3-ol
4-(3,4,7-trimethyl-1H-indole-2-amido)oxane-4-carboxylic acid
N-{2-[4-(furan-2-ylmethyl)morpholin-2-yl]ethyl}-3-hydroxybenzamide
1-[3-({[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
3-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-3-methyl-1-(1,2,3-thiadiazol-5-yl)urea
2-(methylsulfanyl)-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}-1,3-thiazole-4-carboxamide
1-{2-[ethyl(methyl)amino]acetyl}-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperazine
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-{[methyl(oxan-4-yl)amino]methyl}piperidin-2-one
5-methyl-1-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]-5-phenylpiperidin-2-one
9-(3-methoxybenzenesulfonyl)-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
7-fluoro-4-[2-(3-methyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]-2-(pyrimidin-5-yl)quinoline
4-[(2-methylpyridin-3-yl)oxy]-N-[2-(3-methylthiophen-2-yl)ethyl]piperidine-4-carboxamide
5-ethyl-2,3-dimethyl-N-[(5-methylthiophen-2-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
N-(4-methyl-1,3-thiazol-2-yl)-4-(1H-pyrazol-3-yl)benzamide
1-methyl-N-[(5-methylfuran-2-yl)methyl]-5-({[1-(morpholin-4-yl)cyclopentyl]methyl}amino)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-methyl-N-[2-(pyrrolidine-1-sulfonyl)ethyl]-1H-indole-4-carboxamide
ethyl 4-[(4-chlorophenyl)methyl]-1-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}piperidine-4-carboxylate
1-[1'-(3-hydroxy-4-methylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
N-{2-[4-(1-tert-butyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]ethyl}benzamide