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1-[2-ethyl-5-(4H-1,2,4-triazol-4-yl)phenyl]-3-methyl-3-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]urea
methyl({[2-(pyrrolidin-1-yl)pyrimidin-5-yl]methyl})(quinolin-5-ylmethyl)amine
N-(9H-fluoren-9-yl)-3-fluoroimidazo[1,2-a]pyridine-2-carboxamide
(1-{[(6-amino-2-{[(4-methylphenyl)methyl]sulfanyl}pyrimidin-4-yl)amino]methyl}cyclobutyl)methanol
8-(1H-indol-2-ylmethyl)-3-(2-methoxyethyl)-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[4-phenyl-5-(2-phenyl-1,3-thiazol-5-yl)-1H-imidazol-1-yl]ethan-1-ol
(3aS,6aR)-5-cyclopentyl-3-[2-(pyridin-2-yl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
4-[4-(1-benzyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-3-fluoropyridine
N-(furan-2-ylmethyl)-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
4-[(3,4-dimethoxyphenyl)methyl]-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]piperazin-2-one
(3S)-N-tert-butyl-2-[(4-hydroxy-3-methylphenyl)methyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
[(2S)-1-{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl]methanol
N-{2-[(1R,3S)-1-hydroxy-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-7-yl]-2-oxoethyl}methanesulfonamide
1-benzyl-5-(5-fluoro-2-methoxyphenyl)-3-methyl-1H,4H-pyrazolo[3,4-d]imidazole
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-1-methyl-1H-imidazole-4-sulfonamide
2-(4-{3-[5-(thiophen-2-yl)furan-2-yl]propanoyl}morpholin-3-yl)acetamide
2-ethyl-N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N,4-dimethyl-1,3-thiazole-5-carboxamide
N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-5-methylpyrazine-2-carboxamide
4-[4-(thiomorpholin-4-yl)piperidin-1-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
7-(cyclopropylmethyl)-2-[2-(2,3-difluorophenyl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
{[(3S,4R)-1-(2H-1,3-benzodioxole-5-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl}dimethylamine
5-acetamido-1-ethyl-2-(3-methoxyphenyl)-N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
2-(3-{[methyl(thiophen-2-ylmethyl)amino]methyl}phenyl)-6-(oxan-4-yl)-3,4-dihydropyrimidin-4-one
N4-(1H-1,3-benzodiazol-2-ylmethyl)-6-ethyl-5-methylpyrimidine-2,4-diamine
1-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}cyclopropan-1-amine
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-(1,3-benzothiazol-2-yl)-3-{ethyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amino}propanamide
N-[1-(benzenesulfonyl)piperidin-4-yl]-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(pyridin-2-ylmethyl)acetamide
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-({[(1r,4r)-4-hydroxycyclohexyl]amino}methyl)piperidin-2-one
1-[1-(methoxymethyl)cyclopropanecarbonyl]-4-(pyridin-4-yl)-1,4-diazepan-6-ol
2-methyl-8-[6-methyl-1-(propan-2-yl)-1H-pyrazolo[3,4-b]pyridine-4-carbonyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
1-(4-{1-azabicyclo[2.2.2]octan-3-yl}piperazin-1-yl)-3-(2,4-difluorophenyl)propan-1-one
(3aR,6aR)-2-acetyl-5-{[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-{4-[(4,8-dimethoxynaphthalen-1-yl)methyl]piperazin-1-yl}propan-1-ol
1-[(furan-2-ylmethyl)carbamoyl]-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
3-methyl-3-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1-(5,6,7,8-tetrahydronaphthalen-1-yl)urea
2-{[4-cyclohexyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}quinolin-4-ol
2-{4-[2-(2-amino-4,6-dimethylpyrimidin-5-yl)acetyl]piperazin-1-yl}-N-ethylacetamide
9-(2-hydroxyethyl)-1-methyl-4-(pyrazin-2-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
8-(2,3-dihydro-1H-inden-2-yl)-1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(ethoxymethyl)-1-(5-propyl-1,3,4-oxadiazol-2-yl)piperidine
4-(4-benzyl-1H-1,2,3-triazol-1-yl)-1-(1,3-thiazole-4-carbonyl)piperidine
6-(1-phenylpropyl)-3-(propan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
2-methyl-4-{4-[(2-propylpyrrolidin-1-yl)methyl]phenyl}butan-2-ol
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
2-[6-(4-phenylazepan-1-yl)pyrimidin-4-yl]ethan-1-amine
N,N-dimethyl-6-{[1-(thiomorpholin-4-yl)hex-5-en-2-yl]oxy}pyridazin-3-amine
2-butoxy-N-(2-methoxyethyl)-N-(thiophen-2-ylmethyl)acetamide
N-cyclopropyl-N-({4-methoxy-3-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)thiophene-2-carboxamide