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[(3R,4R)-4-[(4-ethylpiperazin-1-yl)methyl]-1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]methanol
3-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)-1-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}urea
3-chloro-4-({1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}oxy)-N-(2-methoxyethyl)benzamide
[(5-tert-butyl-1H-pyrazol-3-yl)methyl](methyl)[(2-methyl-2,3-dihydro-1H-isoindol-5-yl)methyl]amine
3-({2-[5-methyl-2-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}methyl)-4-propyl-4H-1,2,4-triazole
2-(2,4-dichlorophenoxy)-1-[3-(pyridin-2-yl)azetidin-1-yl]ethan-1-one
2-{[6-(2-fluoro-3-methoxyphenyl)pyridazin-3-yl](methyl)amino}ethan-1-ol
3-(3-chloro-1H-1,2,4-triazol-5-yl)-N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}propanamide
4-(cyclopropylmethyl)-3-(propan-2-yl)-1-(pyridin-4-ylmethyl)-1,4-diazepan-5-one
2-[methyl(phenyl)amino]-1-[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]ethan-1-one
5-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-N-phenyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N-(2-oxo-2,3-dihydro-1H-indol-5-yl)-2-(pyridin-3-yl)piperidine-1-carboxamide
4-{[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]amino}-N,5-dimethyl-N-[2-(4-methylphenoxy)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide
2-(2H-1,2,3-benzotriazol-2-yl)-1-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]ethan-1-one
8-[4-(4-ethoxy-3-methylphenyl)butanoyl]-2,8-diazaspiro[4.5]decan-3-one
2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]-N-[(1-hydroxycyclohexyl)methyl]acetamide
ethyl 1-{5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-6-yl}cyclobutane-1-carboxylate
3-(4-{1-[3-(dimethylamino)-2,2-dimethylpropyl]pyrrolidin-3-yl}pyridin-2-yl)phenol
1-{1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-(piperidin-1-yl)piperidine-4-carboxamide
3-methyl-7-[2-(5-oxo-2-phenylcyclopent-1-en-1-yl)acetyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-2-(methylamino)pyridine-4-carboxamide
N3-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-1-(butan-2-yl)-N5-(furan-2-ylmethyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-(2H-1,3-benzodioxol-5-yl)-2-(2-{[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}-4-phenylphenoxy)acetamide
N2-[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-N1-(3-methylpyridin-2-yl)ethane-1,2-diamine
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-3-ethyl-5-hydroxy-N-methyladamantane-1-carboxamide
N-[(2-aminopyrimidin-5-yl)methyl]-N,6-dimethylimidazo[1,2-a]pyridine-2-carboxamide
4-(4-methyl-1,3-oxazole-5-carbonyl)-2-(4-methylpentyl)morpholine
1-(6-cyanopyridin-2-yl)-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
9-[2-(benzyloxy)acetyl]-2-cyclopropyl-2,9-diazaspiro[5.5]undecan-3-one
[(3R,4R)-1-(2,3-dihydro-1H-indene-5-carbonyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
2-amino-4-(furan-3-yl)-6-(2,3,4-trimethoxyphenyl)pyridine-3-carbonitrile
1-[1-(1,2-oxazol-3-ylmethyl)piperidin-3-yl]-4-phenylpiperazine
(3R,4S)-4-[4-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-1,4-diazepan-1-yl]oxolan-3-ol
2-(3-methoxypropyl)-8-(4-methyl-1H-pyrrole-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
6-(azepan-1-yl)-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methyl-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
(3S,4S)-1-[(2-cyanophenyl)methyl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
3-[4-(3,6-dimethyl-1-benzofuran-2-carbonyl)-2-oxopiperazin-1-yl]benzonitrile
5-{[cyclopropyl(pyridin-4-ylmethyl)amino]methyl}-2-methoxybenzoic acid
1-(1-methyl-1H-indole-3-carbonyl)-4-(pyrimidin-2-yl)piperazine-2-carboxylic acid
({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)[(4-fluorophenyl)methyl]methylamine
3-(2-fluorophenoxymethyl)-1-(2-propyl-1,3-thiazole-4-carbonyl)piperidine
3-[2-(2-fluorophenyl)ethyl]-1-[4-(1H-pyrazol-3-yl)benzoyl]piperidine
{2-[methyl({[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl})amino]-1,3-thiazol-4-yl}methanol
1-[4-(2-fluorophenyl)pyrimidin-2-yl]-N-[2-methyl-2-(morpholin-4-yl)propyl]-5-(propan-2-yl)-1H-pyrazole-4-carboxamide
1-benzyl-8-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[1-(thian-4-yl)piperidin-3-yl]-4-[3-(trifluoromethyl)phenyl]piperazine
1-(3-propyl-1H-pyrazole-5-carbonyl)-4-(pyridin-3-yl)piperazine
N-[2-(methylsulfanyl)ethyl]-6-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
ethyl 1-({5-[(adamantan-2-yl)carbamoyl]-6-oxo-1,6-dihydropyridin-2-yl}methyl)piperidine-4-carboxylate
1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine