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6-amino-1-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]hexan-1-one
1-(4,6-dimethylpyrimidin-2-yl)-4'-(2-methylpropyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
(1-{6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carbonyl}pyrrolidin-3-yl)methanol
3-(4-{[(4aS,8aS)-4a-hydroxy-decahydroisoquinolin-2-yl]methyl}-1H-pyrazol-1-yl)propanoic acid
(1S,5R)-6-(cyclopropylmethyl)-3-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}-3,6-diazabicyclo[3.2.2]nonan-7-one
5-oxo-1-(pyridin-2-ylmethyl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]pyrrolidine-3-carboxamide
5-{3-oxo-3-[4-(pyridin-3-ylmethyl)piperazin-1-yl]propyl}imidazolidine-2,4-dione
N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-3,5-dimethylbenzamide
5-(5-ethyl-1,3-oxazol-4-yl)-3-(thiophen-3-ylmethyl)-1,2,4-oxadiazole
(3R,4S)-4-cyclopropyl-1-{6-methylthieno[2,3-d]pyrimidin-4-yl}pyrrolidin-3-amine
(1S,5R)-6-(1-benzothiophene-2-carbonyl)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-(pyridin-3-ylmethyl)-1-[1-(1,3-thiazol-2-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-[(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]-5-methyl-3-phenyl-1,2-oxazole-4-carboxamide
5-cyclohexaneamido-1-(2-methoxyethyl)-N-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
N-benzyl-N,1-dimethyl-5-{4-[(3-methylphenyl)methyl]piperazin-1-yl}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(2R,3R)-3-(dimethylamino)-1'-(4-methyl-1,3-thiazole-5-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-(1-propylpiperidin-4-yl)-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]acetamide
{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(methyl)[2-(morpholin-4-yl)ethyl]amine
1-(propan-2-yl)-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-pyrazole-4-carboxamide
(1R,9S)-5-amino-12-methyl-3-[3-(1H-pyrazol-1-ylmethyl)phenyl]-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]acetamide
2-amino-4-(4,5-dimethylfuran-2-yl)-6-(pyrazine-2-carbonyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[(2,4,6-trimethylphenyl)methyl]amine
methyl 1-ethoxy-2-oxo-8-[3-(2-oxopyrrolidin-1-yl)benzoyl]-1,8-diazaspiro[4.5]decane-4-carboxylate
N-{1-[1-(but-2-ynoyl)piperidin-4-yl]-2-(3-methoxyphenyl)ethyl}-N-methylpyridine-3-carboxamide
N3-ethyl-N5-[1-(furan-2-yl)ethyl]-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
1-[3-(4-fluorophenoxymethyl)piperidin-1-yl]-3-methoxypropan-1-one
1-{2-[1-(2-chloro-5-fluorobenzoyl)piperidin-2-yl]ethyl}pyrrolidin-2-one
N-cyclopentyl-2-[2-(1H-imidazol-4-yl)ethyl]-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
8-(5-hydroxypyridine-2-carbonyl)-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-amino-1-[3-(4-fluorophenoxymethyl)piperidin-1-yl]-2-methylpropan-1-one
1-[3-(4-{1-[(2E)-4-methylpent-2-en-1-yl]pyrrolidin-3-yl}pyridin-2-yl)phenyl]ethan-1-one
7-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(3S,9aR)-8-(2,3-difluorobenzoyl)-3-[(4-methoxyphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-(1-benzyl-5-oxopyrrolidin-3-yl)-3-(3-hydroxy-3-methylbutyl)benzamide
2-(4-methyl-1,2,5-oxadiazol-3-yl)-N-({1-[(3-methylphenyl)methyl]pyrrolidin-3-yl}methyl)acetamide
2-{2-[4-(2-hydroxyethyl)piperidin-1-yl]-4-(morpholin-4-yl)pyrimidin-5-yl}-2-methylpropanoic acid
3-(1H-indol-6-ylmethyl)-1λ6-thiane-1,1-dione
6-(dimethylamino)-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-2-ylmethyl)pyridine-3-carboxamide
N-(1,3-dimethyl-1H-pyrazol-5-yl)-5-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-ylmethyl}-1,3-thiazol-2-amine
(2S)-2-acetamido-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)propanamide
4-(4-ethoxy-3-methylphenyl)-1-{4-[(pyrimidin-2-yl)amino]piperidin-1-yl}butan-1-one
methyl 3-[(2-fluoro-5-methoxyphenyl)methyl]-9-[(1-methyl-5-oxopyrrolidin-3-yl)methoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-ethyl-4-({1-[(2-fluorophenyl)methyl]-2-(propane-2-sulfonyl)-1H-imidazol-5-yl}methyl)piperazin-2-one
2-amino-4-[2-(prop-2-en-1-yloxy)phenyl]-5H,7H,8H-pyrano[4,3-b]pyridine-3-carbonitrile
benzyl 3-({[(1-methyl-1H-1,2,3-triazol-4-yl)carbamoyl]amino}methyl)piperidine-1-carboxylate
N-{1-[1-(2-amino-2-methylpropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-methoxybenzamide
N-methyl-4-{[(4-methylphenyl)amino]methyl}-N-(oxan-2-ylmethyl)benzamide
6,7-dimethoxy-2-[2-(pyridin-4-yl)pyrimidine-5-carbonyl]-1,2,3,4-tetrahydroisoquinoline
1-(2-{[4-(furan-2-carbonyl)piperazin-1-yl]methyl}phenoxy)-3-(piperidin-1-yl)propan-2-ol