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3-[4-(2,4-dimethylphenyl)piperazine-1-carbonyl]-2-ethyl-6-methyl-1-(thiophen-2-ylmethyl)-1,4-dihydropyridin-4-one
N-[2-(1-ethyl-1H-1,3-benzodiazol-2-yl)ethyl]-4-(4-oxo-3,4-dihydroquinazolin-3-yl)butanamide
1-cyclopentanecarbonyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}piperidine-4-carboxamide
3-{[4-(dimethylamino)azepan-1-yl]methyl}-5,6,7-trimethoxy-1,2-dihydroquinolin-2-one
2-(pyridin-3-yl)-N-(1,2,3,4-tetrahydronaphthalen-2-yl)pyrimidine-5-carboxamide
N-(1-methoxypropan-2-yl)-3-[(oxan-4-ylmethyl)sulfamoyl]benzamide
methyl 5-[(4-hydroxybutan-2-yl)amino]-3-(2-methoxyacetamido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N3-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-N5-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
(2S,4R)-4-amino-N-methyl-1-{3-[5-(4-methylphenyl)furan-2-yl]propanoyl}pyrrolidine-2-carboxamide
1-[4-(3-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-3,3,3-trifluoropropan-1-one
[(3R,4R)-1-(3-chloro-4-propoxybenzoyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-[(8-{2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-1-oxa-8-azaspiro[4.5]decan-2-yl)methyl]acetamide
2-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]quinoline
5-[3-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]-2,3-dimethyl-1H-indole
[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl](furan-2-ylmethyl)[2-(morpholin-4-yl)ethyl]amine
4-(1-benzothiophen-2-ylmethyl)-11-{[(3-methoxyphenyl)methyl]amino}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-methyl-5-{2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}-1,3-benzothiazole
(1R,5R)-3-methanesulfonyl-6-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
4-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-1,4-oxazepan-6-ol
N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}-2-phenyl-2-(1H-1,2,3,4-tetrazol-1-yl)acetamide
3-[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-3-yl]-N-[(5-methylfuran-2-yl)methyl]propanamide
4-(2-{[1-(3-ethanesulfonamidophenyl)piperidin-4-yl]amino}ethyl)benzene-1-sulfonamide
N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
2-methyl-8-({2-[(oxolan-2-ylmethyl)amino]pyrimidin-5-yl}methyl)-2,8-diazaspiro[4.5]decan-3-one
methyl 2-{[(4-chlorophenyl)methyl]sulfamoyl}-6-(pyridin-4-ylmethyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-(2-{3-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}-2-oxoethyl)-2-azaspiro[4.4]nonan-3-one
2-methanesulfonyl-N-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]acetamide
1-[3-(2-methylphenoxy)azetidin-1-yl]-3-(pyridin-3-yl)propan-1-one
N-(cyclopropylmethyl)-N-propyl-2-(pyridazine-3-carbonyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
4-(2,5-dimethylpyrimidin-4-yl)-2-(6-methoxynaphthalen-2-yl)morpholine
1-[4-(3-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-(1H-pyrrol-1-yl)ethan-1-one
1-[(3S,4R)-1-[2-(2,5-dimethoxyphenyl)acetyl]-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
5-{1-[(4-fluorophenyl)methyl]-4-hydroxypiperidin-4-yl}-N-methyl-N-[2-(pyridin-2-yl)ethyl]-1-benzofuran-2-carboxamide
6-{2-[(3aS,6aS)-1-cyclohexanecarbonyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]-2-oxoethyl}-2-amino-3,4-dihydropyrimidin-4-one
N-methyl-5-(phenoxymethyl)-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-1H-pyrazole-3-carboxamide
6,8-dimethyl-2-{[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]methyl}quinolin-4-ol
{2-[5-(piperidine-1-carbonyl)pyridin-2-yl]phenyl}methanol
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-methyl-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
1,3-dimethyl-N-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
(2S,4S)-4-amino-1-[(6-methoxy-1-methyl-1H-indol-3-yl)methyl]-N-methylpyrrolidine-2-carboxamide
6-fluoro-8-(5-fluoro-4-methoxypyrimidin-2-yl)quinoline
3-methyl-3-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}-1-[3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]urea
N-{imidazo[1,2-a]pyridin-2-ylmethyl}-1-(1-methylpiperidin-4-yl)piperidine-3-carboxamide
2-[(3S,4R)-3-methanesulfonamido-4-propylpyrrolidin-1-yl]-1,3-thiazole-4-carboxamide
1-{1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-3-yl}-4-(2-methylphenyl)piperazine
2-(4-acetylpiperazin-1-yl)-N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)acetamide
1-[(4-methylphenyl)methyl]-4-(2-oxo-1-phenylpyrrolidine-3-carbonyl)piperazin-2-one
2-{2-[2-(1H-imidazol-4-yl)ethyl]-3-oxo-2,9-diazaspiro[5.5]undecane-9-carbonyl}benzonitrile
3-{1-[6-(3-fluorophenyl)imidazo[2,1-b][1,3]thiazol-3-yl]-N-(propan-2-yl)formamido}propanamide
(2S,4S)-4-(2-cyanobenzamido)-1-cyclobutanecarbonyl-N-ethylpyrrolidine-2-carboxamide