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N-[3-(azepan-1-yl)propyl]-N-methyl-4-(4H-1,2,4-triazol-4-yl)benzamide
ethyl 4-[(4-chlorophenyl)methyl]-1-[(2-ethylphenyl)carbamoyl]piperidine-4-carboxylate
3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)-N-[1-(2-phenylethyl)piperidin-3-yl]propanamide
N-[2-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-4-methylbenzamide
N-butyl-2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
1-methyl-N-(3-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)-1H-imidazole-4-sulfonamide
1-{[6-(4-fluorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-2-methyl-1,4-diazepan-5-one
3-methoxy-1-{4-[4-(1,2-oxazinane-2-carbonyl)phenoxy]piperidin-1-yl}propan-1-one
1-cyclopropanecarbonyl-N-[1-(pyridin-4-yl)propyl]piperidine-4-carboxamide
1-[1-(3,4-difluoro-5-hydroxyphenyl)-1H-pyrazol-3-yl]ethan-1-one
4-(1H-pyrazol-4-yl)-N-[(1s,4s)-4-aminocyclohexyl]butanamide
[(4aS,8aR)-6-[4-(methylsulfanyl)benzoyl]-decahydro-1,6-naphthyridin-4a-yl]methanol
2-(4-cyclopentyl-3-oxopiperazin-1-yl)-2-[4-(hydroxymethyl)phenyl]acetic acid
2-(2,5-difluorophenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}pyrrolidin-1-yl]ethan-1-one
methyl({[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}){[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
methyl (2S)-2-{[1-(4-benzenesulfonamidophenyl)piperidin-4-yl]amino}-3-methylbutanoate
N-(1-hydroxybutan-2-yl)-3-(5-methyl-1,2,4-oxadiazol-3-yl)-N-(pyridin-2-ylmethyl)benzamide
N-[4-(3-cyanopiperidine-1-carbonyl)phenyl]ethane-1-sulfonamide
4-methyl-6-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}-2-(propan-2-yl)pyrimidine
5-[1-(3,4-difluorophenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]-4-methylpyrimidin-2-amine
ethyl 3-[(2,4-difluorophenyl)methyl]-1-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)piperidine-3-carboxylate
2-[4-ethyl-4-(hydroxymethyl)piperidine-1-carbonyl]-6-methyl-4H-pyran-4-one
2-[4-(2-benzyl-1,3-thiazole-4-carbonyl)-1-methylpiperazin-2-yl]ethan-1-ol
1-[(2R,3S,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(4H-1,2,4-triazol-4-yl)propan-1-one
1-[1-methyl-5-({4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)-1H-pyrrol-3-yl]ethan-1-one
(1R,5R)-6-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
2-{1-[(4-methoxy-3-methylphenyl)methyl]-4-[(2-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
3-chloro-N-(2-methoxyethyl)-4-({1-[(4-methoxyphenyl)methyl]piperidin-4-yl}oxy)benzamide
9-(3,5-dichloro-4-methylbenzoyl)-3-oxa-9-azaspiro[5.5]undecane
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-2-(3-fluorophenyl)azepane
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-1-(furan-2-ylmethyl)-N-methylpiperidin-4-amine
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]piperazin-2-one
1-(2-methylpyridin-4-yl)-4-[3-(thiophen-3-yl)-1H-pyrazole-5-carbonyl]-1,4-diazepane
1-[4-(dimethylamino)azepan-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one
1-(3-{3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}-3-oxopropyl)piperidin-2-one
9-[2-(4,5-dimethyl-1H-imidazol-1-yl)acetyl]-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
(3S,4S)-1-[2-(benzenesulfonyl)ethyl]-4-cyclopropylpyrrolidine-3-carboxylic acid
(1R,5R)-3-(6-methoxy-1-methyl-1H-indole-2-carbonyl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
2-{[6-(2-fluoro-4-methoxyphenyl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazin-2-yl]formamido}-N,N-dimethylacetamide
(3S,4R)-1-(1-aminocyclopropanecarbonyl)-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
1-[3-(hydroxymethyl)-3-propylpiperidin-1-yl]-4-(2-methyl-1H-imidazol-1-yl)butan-1-one
8-[2-(dimethyl-1H-1,2,4-triazol-1-yl)acetyl]-2-ethyl-2,8-diazaspiro[4.5]decan-3-one
N,7-dimethyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}-2,3-dihydro-1,4-benzodioxine-6-carboxamide
1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-8-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[2,4-bis(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
3-(morpholine-4-carbonyl)-N-[(4-phenyloxan-4-yl)methyl]-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-benzyl-2-methyl-5-(2-methylpropanamido)-N-[(5-oxopyrrolidin-2-yl)methyl]-N-(propan-2-yl)-1H-1,3-benzodiazole-7-carboxamide
N-[3-(4-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}phenoxy)propyl]-1,3-thiazole-5-carboxamide
6-{[4-(1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]methyl}-1H-indole
(1S,5R)-6-benzyl-3-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one