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7-(pyridin-3-yl)-4-(pyridin-3-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-{1-[2-(2-chlorophenyl)acetyl]piperidin-3-yl}-N-methyl-N-(1-methylpiperidin-4-yl)propanamide
N-(2-cyclopropanecarbonyl-1,2,3,4-tetrahydroisoquinolin-7-yl)-4-(trifluoromethyl)benzamide
1-[1-(2-methylpropyl)-1H-pyrazol-5-yl]-3-[(1R,2S)-2-phenylcyclopropyl]urea
2-(5-fluoro-2-methoxyphenyl)-6-(4-methylpiperazine-1-carbonyl)pyrazine
(4aS,7aR)-1-[(2,5-dimethylphenyl)methyl]-4-[(5-methylfuran-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-{1-[(3,5-dimethyl-1-benzofuran-2-yl)methyl]pyrrolidin-2-yl}-3-methyl-1,2-oxazole
1-(3-fluoro-4-methylphenyl)-3-[1-(4-propyl-4H-1,2,4-triazol-3-yl)ethyl]urea
3-(2-fluoro-6-methoxyphenyl)-5-(thiomorpholine-4-sulfonyl)benzoic acid
4-ethyl-1-methyl-3-[(1-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}piperidin-4-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(2-methoxyphenyl)methyl]-N-methyl-6-oxo-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethan-1-one
4-benzyl-3-[1-(4-methylbenzoyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
[1-(4-aminopyrimidin-2-yl)-4-[(3-fluorophenyl)methyl]piperidin-4-yl]methanol
3-[3-(1H-imidazol-2-yl)piperidine-1-carbonyl]-6-phenyl-1,2-dihydropyridin-2-one
9-[2-(5-methyl-1H-pyrazol-1-yl)acetyl]-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
2-[3-(4-methoxyphenyl)propanamido]-N,N-dimethylpropanamide
3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]-1-(thiophen-2-ylmethyl)piperidine
2-(propan-2-yloxy)-N-{2-[(pyridin-3-yl)amino]ethyl}propanamide
N-[(4-benzyl-5-{[(2-chlorophenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl)methyl]propanamide
5-phenyl-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-1,2-oxazole-3-carboxamide
5-{[3-(piperidin-1-yl)pyrrolidin-1-yl]methyl}-2-(pyridin-2-yl)pyrimidine
7-methoxy-3-({methyl[2-(pyridin-4-yl)ethyl]amino}methyl)-1,2-dihydroquinolin-2-one
2-(3,4-dimethoxyphenyl)-7-methyl-3-[(4-methyl-1,4-diazepan-1-yl)methyl]quinoline
4-(prop-2-en-1-yl)-1-{[4-(trifluoromethoxy)phenyl]methyl}-1,4-diazepan-5-one
4-{4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-6-methylpyrimidine
N-[(5-chloro-2-propoxyphenyl)methyl]morpholine-2-carboxamide
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-1-[2-(methylsulfanyl)pyrimidin-4-yl]piperidin-4-amine
2-methoxy-5-{[(oxolan-2-ylmethyl)(pyridin-4-ylmethyl)amino]methyl}benzoic acid
4-[(4-oxo-3,4-dihydrophthalazin-1-yl)methyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-[1-cyclopentyl-3-(4-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-(oxan-4-yl)acetamide
2-cyclopropyl-N-[2-(propylsulfanyl)ethyl]pyrimidine-5-carboxamide
(1-benzothiophen-2-ylmethyl)(methyl)[(4-{2-[4-(2-methyl-1,3-thiazole-4-carbonyl)piperazin-1-yl]ethoxy}phenyl)methyl]amine
3-(1-ethyl-1H-pyrazol-4-yl)-4-(1-phenylethyl)-4H-1,2,4-triazole
3-methoxy-5-[3-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]pyridine
1-(3-fluorobenzoyl)-3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}[4-(1H-pyrazol-1-yl)butan-2-yl]amine
methyl 4-(5-{[2-(1,3-thiazol-2-yl)piperidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoate
5-{3-[2-(3-methoxyphenyl)ethyl]piperidine-1-carbonyl}-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
4-[(dimethylamino)methyl]-1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]azepan-4-ol
N3-(3-methoxypropyl)-N1,N1-dimethyl-N3-[(4-methylphenyl)methyl]piperidine-1,3-dicarboxamide
{1-methyl-5-[6-(4-methylphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}methanol
(3S,4R)-4-(pyridin-4-yl)-1-[2-(pyrrolidin-1-yl)benzoyl]pyrrolidine-3-carboxylic acid
5-methyl-1-(3-methylphenyl)-4-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]piperazin-2-one
(2S,4R)-4-(4-chlorobenzamido)-N-ethyl-1-(3-hydroxypropanoyl)pyrrolidine-2-carboxamide
methyl[(5-{[(2-methylphenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)methyl][(6-methylpyridin-2-yl)methyl]amine
4-[5-(propan-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl]-4-azaspiro[2.5]octane
N-[(3-hydroxypiperidin-3-yl)methyl]-2-(thiophen-2-yl)acetamide
4-(4-fluorophenyl)-1-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]butan-1-one
1,2-dimethyl-5-[(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)methyl]-1H-1,3-benzodiazole