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6-(2-aminoethyl)-N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]pyrimidin-4-amine
5-[(4-benzylpiperidin-1-yl)methyl]-N-methyl-N-[(3-methylpyridin-2-yl)methyl]-1,2-oxazole-3-carboxamide
N,2,7-trimethyl-N-[3-(oxolan-2-yl)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetamide
4-[2-oxo-2-(5,6,7,8-tetrahydro-1,6-naphthyridin-6-yl)ethyl]-1-phenyl-3-propyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4-(4-chlorophenyl)-1-[1-(methoxymethyl)cyclobutanecarbonyl]piperidin-4-ol
4-[5-(2-chlorophenyl)furan-2-carbonyl]-1,4-oxazepane
ethyl 4-[4-(4-{[(3-methyl-1,2-oxazol-5-yl)methyl]amino}piperidin-1-yl)benzoyl]piperazine-1-carboxylate
(3S,5S)-5-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)-1-methylpyrrolidin-3-amine
1-(1-benzothiophene-2-carbonyl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
N-cyclopropyl-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)-1,2,5-thiadiazole-3-carboxamide
3-[(4,4-difluoropiperidin-1-yl)sulfonyl]-N-[(1-methyl-1H-pyrazol-4-yl)methyl]benzamide
3-[1-cyclohexyl-5-(methoxymethyl)-1H-1,2,4-triazol-3-yl]pyridine
3-(1-ethyl-1H-1,2,3-triazol-4-yl)-1-{[1-(4-fluorophenyl)cyclopentyl]methyl}urea
ethyl 4-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)piperidine-1-carboxylate
3-({[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}amino)butan-1-ol
3-benzyl-8-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{[2-(dimethylamino)-7-methoxyquinolin-3-yl]methyl}-N-(2-methoxyethyl)-3-(3-methyl-1H-pyrazol-1-yl)propanamide
1-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]-3-ethylurea
3-{2-[2-(propan-2-yl)-1H-imidazol-1-yl]ethyl}-1H-indole
ethyl 2-{1-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]piperidin-2-yl}acetate
4-[1-(5,6-dimethylpyrimidin-4-yl)azetidin-3-yl]morpholine
(3S)-1-{[7-methyl-2-(3-methylphenyl)quinolin-3-yl]methyl}pyrrolidin-3-ol
3-(2-ethoxyethoxy)-N-[1-(3-methylbutan-2-yl)-1H-pyrazol-5-yl]benzamide
8-methyl-N-(propan-2-yl)-2-[2-(pyridin-2-yl)pyrimidin-5-yl]quinoline-4-carboxamide
ethyl[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)amine
1-[(2-chloro-5-fluorophenyl)methyl]-4-cyclopropyl-4-methylpyrrolidin-2-one
N-(isoquinolin-5-ylmethyl)-N-methyl-5-(naphthalen-1-yl)-1,2,4-triazin-3-amine
8-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
8-(1,3-benzothiazol-2-ylmethyl)-1-ethyl-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{[2-(cycloheptanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-3-methylpiperidine
4-[1-(7-fluoro-2-methylquinoline-4-carbonyl)piperidin-3-yl]benzoic acid
2-(2H-1,2,3-benzotriazol-2-yl)-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]acetamide
1-[(2,3-dichloro-6-fluorophenyl)methyl]pyrrolidin-2-one
N4-[(1-benzylpyrrolidin-3-yl)methyl]-N4,6-dimethylpyrimidine-2,4-diamine
N-(2-methoxypyridin-3-yl)-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
2-({1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-4-yl}oxy)pyrimidine
N-[(7S,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1,8-naphthyridine-2-carboxamide
N-methyl-3-[3-(2-methylpiperidin-1-yl)azetidine-1-carbonyl]pyridin-2-amine
4-({1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}carbamoyl)pyridin-1-ium-1-olate
5-cyclopropyl-N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-1,3-oxazole-4-carboxamide
N-cyclohexyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-5-phenyl-1,2-oxazole-3-carboxamide
3-amino-1-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}propan-1-one
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-2-(1H-pyrazol-1-yl)benzamide
3-({[(3-chlorophenyl)methyl]amino}methyl)-N,N-dimethylpyridin-2-amine
5-{3-[2-(4-methoxyphenyl)ethyl]piperidine-1-carbonyl}-2-methylpyridine
N-ethyl-3-methoxy-N-[2-(1H-pyrazol-1-yl)ethyl]pyridine-2-carboxamide
5-{[4-(adamantan-1-yl)piperazin-1-yl]methyl}-2-(methoxymethyl)pyrimidine
N-{[2-(3-hydroxypiperidin-1-yl)-7-methylquinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1,3-thiazole-5-carboxamide
3-{[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]methyl}-3-hydroxy-1-(2-methoxyethyl)piperidin-2-one