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1-[4-(1H-1,3-benzodiazol-1-yl)phenyl]-N-[2-(methylsulfanyl)ethyl]piperidin-4-amine
2-(dimethylamino)-2-(3-fluorophenyl)-N-[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]acetamide
N-(oxolan-2-ylmethyl)-2-propyl-N-(pyridin-2-ylmethyl)-1,3-thiazole-4-carboxamide
2-{2-[1-(5-ethyl-2,6-dimethylpyrimidin-4-yl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
N-{2-[4-(4-methyl-1,4-diazepane-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}-2-(naphthalen-2-yl)acetamide
N-[2-(1-ethyl-1H-1,3-benzodiazol-2-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-{5-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-1H-pyrazol-3-yl}ethan-1-one
2-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
N-[2-(1H-imidazol-4-yl)ethyl]-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-2-(3-oxo-3,4-dihydro-2H-1,4-benzothiazin-4-yl)acetamide
N-[(3-methyloxetan-3-yl)methyl]-6-(thiomorpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
9-methoxy-7-(4-methylphenyl)-4-(thiophen-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
6-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidine-1-carbonyl]-2-methyl-2,3-dihydropyridazin-3-one
2-fluoro-N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-5-sulfamoylbenzamide
4-(1H-imidazole-4-carbonyl)-2-(2-phenylethyl)morpholine
N-[2-(N-methylmethanesulfonamido)ethyl]pyridine-3-carboxamide
(4S,4aS,8aS)-1-(morpholine-4-carbonyl)-4-phenyl-decahydroquinolin-4-ol
2-(2-methoxy-5-methylphenyl)-4-(piperidine-1-carbonyl)pyridine
N,N-dimethyl-7-(oxolane-3-carbonyl)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
methyl 2-({9-methyl-10-oxo-3,9-diazaspiro[5.6]dodecane-3-carbonyl}amino)benzoate
5-(2,5-dimethylfuran-3-yl)-1-[(2-methylphenyl)methyl]-3-(oxan-4-yl)-1H-1,2,4-triazole
(1S,4S)-2-(2-methoxy-5-phenylphenyl)-5-(1H-pyrazole-3-carbonyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
5-[(4-chlorophenyl)methyl]-5-{3-oxo-3-[3-(3-phenylpropanoyl)piperidin-1-yl]propyl}pyrrolidin-2-one
5-{2-oxo-2-[2-(2-phenylethyl)piperidin-1-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
methyl 2-(2,3-dihydroxypropyl)-1-oxo-1,2-dihydroisoquinoline-7-carboxylate
2-{4-[(4-fluoropiperidin-1-yl)methyl]phenyl}-6-[2-(1H-pyrazol-1-yl)ethyl]-3,4-dihydropyrimidin-4-one
1-[4-(hydroxymethyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-1-yl]-2-(pyrimidin-2-ylsulfanyl)ethan-1-one
1-cyclopentyl-4-{[4-phenyl-5-(pyridin-3-yl)-1H-imidazol-1-yl]methyl}pyrrolidin-2-one
N-[2-(2-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-(3-methoxyphenyl)-6-methyl-4-(oxolane-3-carbonyl)piperazin-2-one
4-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-1λ6-thiane-1,1-dione
2-butyl-8-(2,6-dimethylpyrimidine-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]-2-(2-phenylethyl)-1,3-benzoxazole-5-carboxamide
(2R,3S,6R)-3-(3-methoxyphenyl)-5-(pyridine-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-{4-[5-fluoro-4-(methylamino)pyrimidin-2-yl]piperazin-1-yl}-1-(piperidin-1-yl)ethan-1-one
3-{3-[methyl(2-methylpropyl)amino]propyl}-8-(oxolan-3-ylmethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
[(1-ethyl-1H-pyrazol-4-yl)methyl][1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]amine
7-(3-methylbut-2-enoyl)-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-(4-hydroxyphenyl)-N-{[1-(pyridin-4-ylmethyl)piperidin-3-yl]methyl}acetamide
1-(cyclopropylmethyl)-N-[(1-ethylpyrrolidin-3-yl)methyl]-5-(quinolin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-(3-{4-[(4-fluorophenyl)sulfanyl]piperidin-1-yl}-3-oxopropyl)-5-methylpyrrolidin-2-one
(1R,6S)-N-{1-[(2-methoxyphenyl)methyl]-1H-pyrazol-5-yl}-9-methyl-3,9-diazabicyclo[4.2.1]nonane-3-carboxamide
N-[2-(2-methoxyphenyl)ethyl]-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
2-(2-fluorophenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]ethan-1-one
1-methyl-3-phenyl-8-(2-phenylacetyl)-1,8-diazaspiro[4.5]decan-2-one
3-(2,5-dioxoimidazolidin-4-yl)-N-[2-(pyridin-4-yl)ethyl]propanamide
(3R,4R)-4-(azepan-1-yl)-1-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}piperidin-3-ol
(3R,5S)-N3-(4-fluorophenyl)-N5-(oxolan-2-ylmethyl)-1-(pyridin-4-ylmethyl)piperidine-3,5-dicarboxamide
3-{1-[(2-ethoxyphenyl)methyl]piperidin-4-yl}-1-(4-phenylpiperazin-1-yl)propan-1-one
N-methyl-1-(3-phenylphenyl)-N-[2-(1H-pyrazol-4-yl)ethyl]piperidin-4-amine