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N-methyl-3-(pyridin-2-yl)-N-[2-(pyridin-2-yl)ethyl]-1H-pyrazole-5-carboxamide
7,8-dimethyl-2-(1-methyl-1H-pyrazol-4-yl)-4-(piperidine-1-carbonyl)quinoline
3-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-1-[3-(propan-2-yl)phenyl]urea
[1-(dimethyl-1,3-thiazol-4-yl)ethyl][(3-ethyl-1,2-oxazol-5-yl)methyl]methylamine
1-(2-methoxyethyl)-3-(2-phenylethyl)-8-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-methoxy-1-{4-[4-(piperazine-1-carbonyl)phenoxy]piperidin-1-yl}propan-1-one
8-(5-propylfuran-2-yl)-2H,5H,6H,7H,8H-[1,3]dioxolo[4,5-g]quinolin-6-one
2-(2H-1,3-benzodioxol-5-yl)-N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
2-({2-[(cyclopropylmethyl)sulfanyl]acetamido}methyl)-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
4-{4-[4-methoxy-4-(prop-2-en-1-yl)piperidin-1-yl]piperidin-1-yl}-2-methyl-6-propylpyrimidine
N,6-dimethyl-2-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyrimidin-4-amine
2-ethyl-N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-4-methyl-1,3-oxazole-5-carboxamide
N-cyclopropyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-(5-methylfuran-2-yl)benzamide
4-(2-methoxyethoxy)-1-{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidine
2-(2,3-dihydro-1H-inden-1-yl)-N-{2-[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]ethyl}acetamide
1-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidin-1-yl]-2-(4-methyl-1H-pyrazol-1-yl)ethan-1-one
N-[2-(cyclohex-1-en-1-yl)ethyl]-3-[2-(furan-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
4-ethyl-1-methyl-3-(1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(5-chloro-2-fluorobenzoyl)-N-(2,3-dihydro-1,4-benzodioxin-6-yl)piperidin-3-amine
4-(5-methyl-4H-1,2,4-triazol-3-yl)-N-[3-(methylsulfanyl)propyl]aniline
(2R,3R)-3-[4-(3,5-difluorophenyl)-1H-1,2,3-triazol-1-yl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
[3-(1H-imidazol-1-yl)propyl](oxolan-3-ylmethyl)(pyridin-3-ylmethyl)amine
2-[({1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}oxy)methyl]pyridine
2-[1-(3-phenylpropyl)-4-(quinolin-8-ylmethyl)piperazin-2-yl]ethan-1-ol
2-{4-[(4-fluorophenyl)methyl]-3-oxopiperazine-1-carbonyl}-3,4-dihydroquinazolin-4-one
1-{1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carbonyl}azetidin-3-ol
N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)-2-(pyridin-3-yl)acetamide
N-methyl-1-[2-(morpholin-4-yl)ethyl]-6-oxo-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidine-3-carboxamide
N-ethyl-N-methyl-2-{2-[(5-methylpyrazin-2-yl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}acetamide
3-[5-(hydroxymethyl)-3-(oxan-4-yl)-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl](methyl){[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}amine
(3S,5R)-N3-(4-methylphenyl)-N5-(oxan-4-yl)piperidine-3,5-dicarboxamide
6-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(morpholin-4-yl)pyrimidin-4-amine
4-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-N,N-dimethylpiperazine-1-carboxamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(1-ethyl-1H-pyrazole-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-chloro-N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-5-(piperidin-1-yl)benzamide
2-({4-[2-(propan-2-yl)-1H-imidazol-5-yl]-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)acetic acid
5-({4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}methyl)-2,1,3-benzothiadiazole
ethyl 4-[(4-chlorophenyl)methyl]-1-(2,3-dihydroxypropyl)piperidine-4-carboxylate
(3S,4R)-1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
(3R,5S)-N-[2-(1H-imidazol-4-yl)ethyl]-1-(2-phenylethyl)-5-[3-(trifluoromethyl)phenoxymethyl]piperidine-3-carboxamide
3-chloro-N-{[4-(2-methylpropoxy)phenyl]methyl}-N-(pyridin-4-ylmethyl)benzamide
8-[3-(1H-1,2,3-benzotriazol-1-yl)propanoyl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[(3-hydroxyphenyl)methyl]-N-methyl-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
N-{2-[5-(hydroxymethyl)-1,2,4-oxadiazol-3-yl]ethyl}imidazo[1,2-a]pyridine-6-carboxamide
2-hydroxy-5-methoxy-N-[(1r,4r)-4-methoxycyclohexyl]benzamide
1-(4-phenylpiperazine-1-carbonyl)-6-[3-(prop-2-en-1-yloxy)benzoyl]-6-azaspiro[2.5]octane
2-[4-(2-{[methyl(propyl)amino]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carbonyl)-1H-1,2,3-triazol-1-yl]ethan-1-amine
1-{4-[4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]-1,4-diazepan-1-yl}ethan-1-one
N-methyl-1-(piperidin-3-ylmethyl)-N-(pyridin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide