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(2S,4S)-4-amino-1-[3-(2-chlorophenyl)-5-methyl-1,2-oxazole-4-carbonyl]-N-methylpyrrolidine-2-carboxamide
(3aS,6aR)-5-(1-benzothiophen-2-ylmethyl)-3-[2-(pyridin-2-yl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-(1-benzothiophene-5-carbonyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
1-{[3-(difluoromethoxy)phenyl]methyl}-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
methyl 3-(2-methoxyacetamido)-1-(3-phenylpropyl)-5-{[4-(1H-pyrazol-1-yl)butan-2-yl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-cyclopentyl-3-fluoro-N-({3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)benzamide
methyl (1R,3S,3aR,6aS)-1,5-dimethyl-4,6-dioxo-3-[2-(propylamino)pyrimidin-5-yl]-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
1-{1-[(5-ethylfuran-2-yl)methyl]piperidin-3-yl}-4-(2-fluorophenyl)piperazine
2-[1-benzyl-4-(2,2-dimethylpropyl)piperazin-2-yl]ethan-1-ol
N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-{[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}cyclopropanamine
3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)-N-methyl-N-(oxan-2-ylmethyl)propanamide
N-({1-[(3-fluoro-4-methoxyphenyl)methyl]piperidin-4-yl}methyl)-1-methylcyclopropane-1-carboxamide
3-cyclopropyl-N-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}-1H-pyrazole-5-carboxamide
4-(cyclohexylmethyl)-1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-1,4-diazepan-5-one
4-[3-(1H-imidazol-2-yl)piperidin-1-yl]-2-methoxypyridine-3-carbonitrile
1-[(3aS,6aS)-5-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-octahydropyrrolo[2,3-c]pyrrol-1-yl]propan-1-one
N-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-3-methyl-2-oxo-1-oxa-3,7-diazaspiro[4.5]decane-7-carboxamide
1-{[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-2-one
N-[(5-methylthiophen-2-yl)methyl]-2-propyl-N-(pyridin-2-ylmethyl)-1,3-thiazole-4-carboxamide
4-(2-chlorophenoxy)-1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidine
N,1-diethyl-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-1H-pyrazole-3-carboxamide
N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]imidazo[1,2-a]pyrimidine-2-carboxamide
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]acetamide
4-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-2-ethyl-1-(propan-2-yl)piperazine
3-[(3R,4R)-3-hydroxy-4-methyl-3-(propan-2-yl)pyrrolidine-1-carbonyl]benzene-1-sulfonamide
2-(morpholin-2-yl)-N-[2-(2-phenoxyphenyl)ethyl]acetamide
methyl 3-(2-methoxy-2-phenylacetyl)-7-oxo-9-(pyridin-4-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-({3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}methyl)-4-methoxyphenol
1-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-4-(1,2,4-oxadiazol-3-yl)piperidine
4-{2-[2-(1H-imidazol-2-yl)-6-methoxyphenoxy]ethyl}morpholine
2,2-diethyl-4-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}morpholine
2-(3-fluorophenoxymethyl)-N-{[1-(morpholin-4-yl)cyclopentyl]methyl}-1,3-oxazole-4-carboxamide
4-(cyclopropylmethyl)-1-[5,6-dimethyl-2-(trifluoromethyl)pyrimidin-4-yl]-3-(propan-2-yl)-1,4-diazepan-5-one
1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(oxolane-2-carbonyl)piperazine
8-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]-1-oxa-8-azaspiro[4.5]decane
1-(1-{5-[4-(trifluoromethyl)phenyl]-1,2,4-triazin-3-yl}piperidin-4-yl)piperidin-4-ol
(3R,4R)-1-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}-4-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidin-3-ol
1-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-4-[(2-methylphenyl)sulfanyl]piperidine
N-({7-[4-(1H-imidazol-1-yl)benzoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-5-methylthiophene-2-carboxamide
4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidine
8-[2-(3,4-dimethyl-6-oxo-1,6-dihydropyridazin-1-yl)acetyl]-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one
2-{[(2-chlorophenyl)methyl](methyl)amino}-2-[4-fluoro-3-(hydroxymethyl)phenyl]acetic acid
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-(2-oxo-1,2-dihydropyridin-1-yl)propanamide
1-(2-methylphenyl)-3-{[1-(pyrrolidin-1-yl)cyclopentyl]methyl}urea
2-(2-{5-[(4-methylphenyl)sulfanyl]furan-2-yl}-1H-imidazol-1-yl)ethan-1-ol
(1R,3S)-3-{1-[(3-chlorophenyl)methyl]-3-methyl-1H-1,2,4-triazol-5-yl}cyclopentan-1-amine
N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]imidazo[1,2-a]pyrimidine-2-carboxamide
3-[(1S,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]propanamide
N-propyl-2-(pyridin-3-yl)pyridine-3-carboxamide
1-[1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)piperidin-4-yl]-N-(oxolan-2-ylmethyl)piperidine-4-carboxamide