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4,6-dimethoxy-2-[3-(pyridin-3-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]pyrimidine
methyl 3-[2-amino-3-cyano-6-(3,5-dimethyl-1H-pyrazol-4-yl)pyridin-4-yl]benzoate
5-{[(3S,4R)-3-cyclopropyl-4-(dimethylamino)pyrrolidin-1-yl]sulfonyl}-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-4-(1H-1,2,4-triazol-1-yl)butan-1-one
2-methyl-1-[9-(oxolan-3-ylmethoxy)-7-{8-thiatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-4-yl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propan-1-one
N-{[1-(2,1,3-benzoxadiazol-4-ylmethyl)piperidin-3-yl]methyl}-2,3-dimethoxybenzamide
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
1-(4-{[3-(2-hydroxyethyl)-4-[(6-methylpyridin-2-yl)methyl]piperazin-1-yl]methyl}thiophen-2-yl)ethan-1-one
N-[2-(N-methylmethanesulfonamido)ethyl]-4-[(2-methylprop-2-en-1-yl)oxy]benzamide
3-{[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-1-yl]methyl}piperidin-3-ol
3-[benzyl({[4-(pyrimidin-2-yloxy)phenyl]methyl})amino]-2-methylpropan-1-ol
{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}(methyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
4-(4-methyl-1H-pyrazol-1-yl)-1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}piperidine-4-carboxylic acid
N,4-dimethyl-2-(methylamino)-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1,3-thiazole-5-carboxamide
4-{4-[methyl(oxan-2-ylmethyl)amino]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl}benzamide
7-(1,3-benzothiazol-2-yl)-4-(furan-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-(4-fluorophenoxy)-1-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperidine
(3S,4R)-1-{3-[(2R,6S)-2,6-dimethylmorpholin-4-yl]propanoyl}-4-phenylpyrrolidine-3-carboxylic acid
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-1,3-dimethyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-methyl-N-{4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]phenyl}methanesulfonamide
3-{[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}-3,4-dihydro-1,2,3-benzotriazin-4-one
N-{1-[1-(1-benzofuran-2-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopropanecarboxamide
3-(1,4-diazepane-1-carbonyl)-N-[2-(1H-pyrazol-1-yl)ethyl]benzene-1-sulfonamide
N,N-dimethyl-1-{2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}pyrrolidin-3-amine
2-oxo-N-[4-(thiophen-2-ylmethoxy)phenyl]-1,3-dioxa-8-azaspiro[4.5]decane-8-carboxamide
(3R,4R)-N-benzyl-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidine-1-carboxamide
N'-cyclopentyl-N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]butanediamide
methyl({4-methyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)[3-(5-methylfuran-2-yl)butyl]amine
N-[2-(morpholin-4-yl)ethyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
3-chloro-5-[2-(dimethylamino)-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-1,2-dihydropyridin-2-one
(3-{2-[1-(4,6-dimethylpyridin-2-yl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)dimethylamine
2-{4-[(6-methoxy-2H-chromen-3-yl)methyl]-1-(thiophen-2-ylmethyl)piperazin-2-yl}ethan-1-ol
2-[methyl({4-methyl-5-[1-(4-methylpyridine-3-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)amino]ethan-1-ol
N-(2H-1,3-benzodioxol-5-ylmethyl)-3-(1,2-oxazolidin-2-yl)-N-(pentan-3-yl)propanamide
3-[2-(benzyloxy)ethyl]-3,9-diazaspiro[5.5]undecane
3-methyl-N-[4-(morpholin-4-yl)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide
4-[(3,5-difluorophenyl)methyl]-1-[(3-methoxyphenyl)methyl]piperazin-2-one
4-(hydroxymethyl)-N-(4-methylphenyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-1-carboxamide
8-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
1-({6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
(3aS,6aR)-3-[3-(morpholin-4-yl)propyl]-5-(2-phenoxyethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(4-methyl-1,3-thiazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-{1-[2-(2-fluorophenoxy)ethyl]-4-phenyl-1H-imidazol-5-yl}pyridine
2-(5-methyl-1,2-oxazol-3-yl)-N-[2-(prop-2-en-1-yloxy)phenyl]piperidine-1-carboxamide
1-(2-{4-[1-(2-fluorophenyl)propan-2-yl]piperazin-1-yl}ethyl)-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
N-[2-(1H-indol-3-yl)ethyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
4-[(4-pentyl-1H-1,2,3-triazol-1-yl)methyl]pyridine
2-(5-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl)ethan-1-ol
1-({5-[1-(azetidine-3-carbonyl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
6-ethyl-2-methoxy-3-({[2-(methylsulfanyl)pyrimidin-4-yl]amino}methyl)-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one